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4-[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]-3-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-(1-{1-[1-ethyl-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]propan-2-yl}-3,5-dimethyl-1H-pyrazol-4-yl)ethan-1-one
(1S,5R)-6-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[1-(1,3-thiazol-2-yl)propyl]acetamide
2-benzyl-N-({2-[3-(2-methoxyacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-1,3-thiazole-4-carboxamide
N-[3-(4-fluorophenyl)phenyl]-1-(2-methoxypyridine-3-carbonyl)piperidine-3-carboxamide
(3S,4S)-1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}-4-(propan-2-yloxy)pyrrolidin-3-ol
3-{[4-(4-fluorophenoxy)piperidin-1-yl]methyl}piperidin-3-ol
N-{3-[(2-methylpropyl)carbamoyl]phenyl}-4-[2-(methylsulfanyl)ethyl]piperazine-1-carboxamide
3-fluoro-N,2-dimethyl-N-(1H-pyrazol-3-ylmethyl)benzamide
2-[(4-aminoazepan-1-yl)methyl]-8-fluoroquinolin-4-ol
N-[3-(1H-pyrazol-1-yl)phenyl]-1-[2-(pyridin-2-yl)acetyl]pyrrolidine-2-carboxamide
9-(2-methoxypropanoyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-benzyl-8-{[6-(dimethylamino)pyridin-3-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
3-(2-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-oxoethyl)-4-[(4-methylphenyl)methyl]piperazin-2-one
4-{1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carbonyl}thiomorpholine
dimethyl[3-(2-{1-[3-(pyrrolidin-1-yl)pyrazin-2-yl]piperidin-4-yl}-1H-imidazol-1-yl)propyl]amine
(2S)-2-{[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}-2-phenylethan-1-ol
N-(5-fluoro-2-methylphenyl)-2-[2-(morpholin-4-yl)ethyl]piperidine-1-carboxamide
N-(2,4-dimethoxyphenyl)-3-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-4-yl)propanamide
N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)pyrazolo[1,5-a]pyridine-2-carboxamide
6-[(diethylamino)methyl]-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-4-(pyridin-3-ylmethyl)piperazine
2-(4-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-oxopiperazin-1-yl)benzonitrile
2-(1,2-benzoxazol-3-yl)-1-[2-(pyridin-2-yl)piperidin-1-yl]ethan-1-one
N-(furan-3-ylmethyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
(4aS,8aR)-6-{2-methyl-7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carbonyl}-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
4-[1-(furan-3-carbonyl)piperidin-4-yl]-5-(3-methylphenyl)-2-(pyridin-4-yl)pyrimidine
3-phenoxy-1-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
N-cyclopentyl-1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-({[2-(dimethylamino)ethyl][(3-methylthiophen-2-yl)methyl]amino}methyl)-3-methoxyphenol
N-[3-(2-chlorophenoxy)propyl]-1-cyclopropyl-N-methyl-5-oxopyrrolidine-3-carboxamide
1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]-2-{methyl[(4-methylphenyl)methyl]amino}ethan-1-one
2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-4-yl)-1H-1,3-benzodiazole
2-({[(3R,4R)-1-[(3-chloro-2-fluorophenyl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl][(5-methylthiophen-2-yl)methyl]amine
N-(7-{6-azabicyclo[3.2.1]octane-6-carbonyl}-2-benzyl-1-methyl-1H-1,3-benzodiazol-5-yl)propanamide
3-(5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-sulfonyl}thiophen-2-yl)-1,2-oxazole
N-(2-hydroxyethyl)-5-{1H-pyrrolo[2,3-c]pyridin-5-ylmethyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
3-hexyl-8-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
ethyl 1-[(2E)-3-(1-methyl-1H-pyrazol-4-yl)prop-2-enoyl]-3-(2-phenoxyethyl)piperidine-3-carboxylate
N-benzyl-N-(3-hydroxy-2-methylpropyl)imidazo[1,2-a]pyridine-3-carboxamide
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-2-(methylsulfanyl)benzamide
N-(2-methylpropyl)-1-{1-[(3,4,5-trimethoxyphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
3-{2-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}phenol
3-[3-(1-methyl-1H-imidazol-2-yl)phenyl]-1-[2-(1H-pyrazol-1-yl)ethyl]-1H-pyrazole
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-3-hydroxy-N-(oxolan-2-ylmethyl)propanamide
1-[3-(1,2-oxazolidin-2-yl)propanoyl]-4-phenoxypiperidine-4-carboxylic acid
8-(1H-indol-2-ylmethyl)-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(5-acetylthiophen-3-yl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide