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N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
(4aR,8aR)-2-methanesulfonyl-7-[(2-methyl-1-benzothiophen-3-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
2-cyclopentyl-1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)[(6-fluoroquinolin-2-yl)methyl]methylamine
3-(2,5-dioxoimidazolidin-4-yl)-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}propanamide
2-({[1-(methoxymethyl)cyclopropyl]methyl}sulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-(dimethylamino)-N-{[3-(3-fluorophenyl)-1,2-oxazol-5-yl]methyl}-2-(2-methylphenyl)acetamide
1-(7-ethyl-1-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indol-3-yl)ethan-1-one
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-[2-(1H-imidazol-1-yl)ethyl]piperidine
2,6-dimethyl-4-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyridine
1-(4-methoxyphenyl)-4-[3-(phenylamino)piperidin-1-yl]butane-1,4-dione
2-cyclopropanecarbonyl-8-[3-(dimethylamino)pyrazin-2-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N,2,8-trimethyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]quinoline-4-carboxamide
2-(3,4-dimethoxyphenyl)-5-fluoro-1-[1-(furan-3-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
3-(pyrrolidine-1-carbonyl)-2-(2,4,6-trimethylphenyl)pyridine
methyl (2S)-2-[(2-butyl-1,3-benzoxazol-5-yl)formamido]-3-phenylpropanoate
(4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}morpholin-2-yl)methanamine
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}(pyridin-2-ylmethyl)amine
4-({1-[(2-aminopyridin-3-yl)methyl]pyrrolidin-3-yl}methyl)benzoic acid
N-(1-{7-[(3,4-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-3,5-dimethylbenzamide
2-cyclopentyl-N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)acetamide
8-[(5-chlorothiophen-2-yl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-hydroxy-N,2-dimethyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrimidine-5-carboxamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1-(5-propylpyrimidin-4-yl)piperidin-4-amine
1-[1-(3-phenyl-1H-1,2,4-triazol-5-yl)ethyl]pyrrolidin-2-one
6-methyl-1-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4-(trifluoromethyl)-1,2-dihydropyridin-2-one
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N-cyclopropyl-N-[(3-ethoxyphenyl)methyl]-3-(1H-imidazol-1-yl)propanamide
(3aS,6aS)-2-benzyl-5-{[(furan-2-ylmethyl)carbamoyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(1r,4r)-4-hydroxycyclohexyl]-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
methyl 8-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
1-(2,3-dihydro-1H-inden-5-yl)-5-[(2S)-1-methanesulfonylpyrrolidin-2-yl]-1H-1,2,4-triazole
3-{2-[1-(propan-2-yl)piperidin-2-yl]ethyl}-8-(trifluoromethyl)-3,4-dihydroquinazolin-4-one
1-[4-(furan-2-yl)benzoyl]-2-(3-methoxypropyl)piperidine
1-[4-(3-fluorophenyl)phenyl]-3-[4-(morpholin-4-yl)butan-2-yl]urea
1-({5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}amino)butan-2-ol
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-(thiophen-3-ylmethyl)acetamide
methyl 4-(3-{2-[(3,5-dimethoxyphenyl)carbamoyl]ethyl}piperidin-1-yl)-4-oxobutanoate
2-({4-[(prop-2-en-1-yl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}methyl)benzoic acid
3-methyl-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}-1H-pyrazole-4-carboxamide
2-[2-(morpholin-4-ylmethyl)piperidin-1-yl]-N-(pyridin-2-ylmethyl)acetamide
(4aS,8aR)-6-[3-(2-methylphenoxy)propanoyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
2,3-dimethyl-6-(1-propanoylpiperidine-3-carbonyl)-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
4-ethyl-1-methyl-3-(1-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(2-phenyl-1,3-thiazol-5-yl)methyl]-3-(pyrrolidin-1-yl)piperidine
1-[(4-methyl-1H-imidazol-5-yl)methyl]spiro[azepane-4,2'-chromene]
3-[(3R,4S)-1-(6-methyl-4-oxo-4H-pyran-2-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
(3aR,6aR)-2-methanesulfonyl-5-[2-(phenylsulfanyl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-methyl-N-[(5-{[methyl({[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl})amino]methyl}furan-2-yl)methyl]methanesulfonamide
(furan-3-ylmethyl)(methyl){[5-(oxolane-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}amine