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3-{1-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-1-oxopropan-2-yl}-2,3-dihydro-1,3-benzoxazol-2-one
N-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-4-hydroxy-2-(phenoxymethyl)pyrimidine-5-carboxamide
N-[(8-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]furan-2-carboxamide
2-acetyl-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
(3S)-N-[3-(3-chlorophenyl)phenyl]-3-(dimethylamino)pyrrolidine-1-carboxamide
1-[4-(furan-2-yl)benzoyl]-4-(pyrrolidine-1-carbonyl)piperidine
N2-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}pyrimidine-2,4-diamine
1-[4-(3-{[methyl(quinolin-5-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
N-(1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
N,1-dimethyl-5-phenyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-3-carboxamide
4-(2-methyl-1H-imidazol-1-yl)-1-(quinolin-8-ylmethyl)piperidine-4-carboxylic acid
4-[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl]-1-(oxan-4-ylmethyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
1-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
4-(2-benzyl-1,3-thiazole-4-carbonyl)morpholine-2-carboxamide
4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}-N-[1-(pyridin-2-yl)propan-2-yl]benzamide
1-[2-(4-chlorophenyl)ethyl]-N-(cyclopropylmethyl)-6-oxo-N-propylpiperidine-3-carboxamide
N-(cyclopropylmethyl)-5-(morpholin-4-ylmethyl)-N-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-cyclopropyl-2,2-dimethyl-N-{[3-(2-methylpropoxy)phenyl]methyl}oxane-4-carboxamide
9-{2-[(cyclopropylmethyl)sulfanyl]acetyl}-2-[3-(1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
N-ethyl-4-methyl-5-[4-(9H-purin-6-yl)piperazine-1-carbonyl]-1,3-thiazol-2-amine
3-chloro-4-fluoro-N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)benzene-1-sulfonamide
N-{1-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]ethyl}-2-(trifluoromethyl)pyrimidin-4-amine
1-(2-fluorophenyl)-3-phenyl-5-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-5-methylpiperidin-2-one
5-{2-[4-(1-hydroxy-3-methylbutyl)piperidin-1-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
6-methyl-2-(3-{[4-(thiophene-2-carbonyl)piperazin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(9H-purin-6-yl)piperazin-2-one
5-(methoxymethyl)-N-{4-[5-methyl-4-({[2-(methylsulfanyl)phenyl]formamido}methyl)-1,3-oxazol-2-yl]phenyl}furan-2-carboxamide
(1R,3S)-7-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carbonyl]-7-azaspiro[3.5]nonane-1,3-diol
(3S,4R)-1-(2-aminopyrimidin-4-yl)-3-ethyl-4-methylpiperidin-4-ol
N-(1,3-benzoxazol-2-ylmethyl)-6-(2-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
(2R,3S,6R)-5-(3-methoxybenzoyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
5-{1-[(4-hydroxyphenyl)methyl]piperidin-4-yl}-5-(2-methylpropyl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
6-phenyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(methylsulfanyl)ethan-1-one
3-methyl-N-({5-methyl-2-[2-(3-phenoxypropanamido)phenyl]-1,3-oxazol-4-yl}methyl)butanamide
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-3-(4-methylphenyl)-1H-pyrazole-5-carboxamide
2-(4-phenyl-1,3-thiazol-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-{3-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(2S)-2-aminopropanoyl]-N-[4-(2-fluorophenoxy)phenyl]piperidine-4-carboxamide
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-[2-(3-methoxyphenyl)ethyl]benzamide
N-[(4-phenyloxan-4-yl)methyl]-1-propyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-2-(methylsulfanyl)acetamide
N-[3-(methylcarbamoyl)-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
1-{4-[(2-fluorophenyl)methyl]piperidin-1-yl}-2-(oxan-2-ylmethoxy)ethan-1-one
4-fluoro-1-({3-methoxy-4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}methyl)piperidine
methyl (2S,4R)-4-(dimethylamino)-1-[(3E)-4-phenylbut-3-enoyl]pyrrolidine-2-carboxylate
2-{4-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidine-1-carbonyl]phenoxy}acetamide
4-[5-(4,6-dimethoxypyrimidin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]morpholine
3-(4-methyl-1,3-thiazol-5-yl)-N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}propanamide