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3-[(2R,3R,6R)-5-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
4-{[5-(methylsulfanyl)-4-phenyl-4H-1,2,4-triazol-3-yl]methyl}-1-(oxolan-3-ylmethyl)piperidine
N-[1-(3-fluoro-4-hydroxyphenyl)ethyl]-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-methyl-N-(oxan-4-yl)acetamide
1-(4-fluorophenyl)-3,5-dimethyl-N-[2-(6-oxo-1,6-dihydropyrimidin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
8-[(3-methoxyphenyl)carbamoyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[4-(4-methylphenoxy)piperidine-1-carbonyl]cyclopropane-1-carboxamide
N-(1-{1-[(2-hydroxy-6-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]ethan-1-one
2-methyl-N-{[1-(4-methylpiperazin-1-yl)cyclopentyl]methyl}-1-benzofuran-5-carboxamide
2-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidine-1-carbonyl]naphthalen-1-ol
6-(4-methoxy-2-methylphenyl)-1H-1,3-benzodiazole
4-{[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)piperidin-4-yl]oxy}pyridine
1-(1-benzylpiperidin-4-yl)-3-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}piperidine
(2S,4R)-4-[2-(5-chloro-6-methyl-1-benzofuran-3-yl)acetamido]-N-ethyl-1-methylpyrrolidine-2-carboxamide
2-[(2R)-2-aminopropanoyl]-N-[2-(pyridin-2-yl)ethyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
N-[3-(azepan-1-yl)-2-hydroxypropyl]-5-chloro-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
[(4-fluoro-3-methoxyphenyl)methyl]({1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl})amine
3-(1,3-benzothiazol-6-yl)-1-(thiolan-3-yl)urea
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-3-chloropyridin-2-amine
N-[(3S)-1-benzylpiperidin-3-yl]-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
1-(5-methyl-1,2-oxazole-4-carbonyl)-3-(2-methylphenyl)piperidine
4-(4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]amino}piperidin-1-yl)-6-methylpyrimidin-2-amine
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amine
N-benzyl-N-(3-hydroxy-2-methylpropyl)pyrazolo[1,5-a]pyridine-3-carboxamide
{1-[6-(dimethylamino)pyrazin-2-yl]-3-ethylpiperidin-3-yl}methanol
2-[2-(dimethylamino)ethyl]-9-[(3-hydroxy-4-methoxyphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
4-({1-[1-(2-methylpyridin-4-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)thiomorpholine
1-{[1-(7-chloroquinolin-4-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
1-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-4-(2-fluorophenyl)piperazine
2-[2-({2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}amino)pyrimidin-4-yl]pyridine-4-carboxylic acid
N-benzyl-N-methyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
(3R,4S)-N,N-dimethyl-1-[4-(piperidine-1-carbonyl)pyridin-2-yl]-4-(propan-2-yl)pyrrolidin-3-amine
2-({[2-(dimethylamino)ethyl][(2-methylphenyl)methyl]amino}methyl)-6-methoxyphenol
N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]piperidin-3-amine
3-(4-methoxyphenyl)-N-methyl-N-[1-(1,3-thiazol-5-yl)ethyl]-1H-pyrazole-5-carboxamide
2-(2-fluoro-3-methoxyphenyl)-6-methylpyridine
4-(1-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)thiomorpholine
(1S,3R)-3-amino-N-(3-{[(2-chlorophenyl)methyl]sulfanyl}propyl)cyclopentane-1-carboxamide
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-3-(4-fluorophenyl)-1H-pyrazole-5-carboxamide
N-[2-(pyridin-3-ylformamido)ethyl]oxane-4-carboxamide
1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methoxybenzoyl)piperazine
1-{[5-(2-chlorophenyl)furan-2-yl]methyl}-3-(pyrrolidine-1-carbonyl)piperazine
2-(3,4-dichlorophenyl)-N,N-diethylmorpholine-4-sulfonamide
methyl 3-benzamido-6-{[(2-ethoxy-2-oxoethyl)(methyl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-methyl-4-{[(4-phenylphenyl)methyl]amino}pyrrolidine-2-carboxamide
2-(3-methoxypropyl)-8-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
N-({7-[2-(2-chloro-4-fluorophenyl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
ethyl 2-(1-{[(4-methoxyphenyl)methyl]carbamoyl}piperidin-2-yl)acetate