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2-(3-{[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
3-fluoro-4-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]pyridine
1-(cyclopropylmethyl)-N-methyl-5-[2-(3-methylphenyl)acetyl]-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(propylsulfanyl)ethan-1-one
(1R,3R,5S)-3-(4-methoxyphenyl)-8-(oxane-4-carbonyl)-8-azabicyclo[3.2.1]octane
2-(3-methyl-1,2-oxazol-5-yl)-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]acetamide
(1R,5S)-6-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
(1-{3-[(6-cyclopropylpyrimidin-4-yl)amino]propyl}piperidin-2-yl)methanol
5-butyl-4-(3-hydroxypropyl)-1-(3-phenylphenyl)piperazin-2-one
N-[(2,3-dimethoxyphenyl)methyl]-3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}propanamide
1-(2-benzylmorpholin-4-yl)-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
N-(1-{7-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
4-methyl-2-(1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperidin-3-yl)-1H-1,3-benzodiazole
4-(2-ethylpyrimidine-5-carbonyl)-3-methyl-1-(2-methylpropyl)piperazin-2-one
3-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanoic acid
N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
5-[2-(2-ethyl-2-methyl-3-oxopiperazin-1-yl)-2-oxoethyl]-2,6-dimethyl-3,4-dihydropyrimidin-4-one
4-{2-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-5-methyl-2,3-dihydro-1H-pyrazol-3-one
2-[5-(6,8-dimethylquinolin-4-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
1-(2,3-difluorobenzoyl)-4-[4-(2-phenylethyl)-1H-pyrazol-5-yl]piperidine
3-amino-1-{[2-(ethylamino)pyrimidin-5-yl]methyl}pyrrolidine-3-carboxylic acid
2-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-S-(4-fluoro-2-methylphenyl)-2-oxoethane-1-sulfonamido
(3S,4S)-4-propyl-1-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]pyrrolidine-3-carboxylic acid
(2S)-2-amino-2-(2-chlorophenyl)-N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]acetamide
8-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-1-oxa-8-azaspiro[4.5]decan-3-ol
(3aS,6aR)-5-(2-methylquinolin-4-yl)-3-[2-(piperidin-1-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
8-(2,2-dimethylpropyl)-3-(2-methoxyethyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[2-(methylsulfanyl)benzoyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
3-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}piperidin-3-ol
6-[4-(benzyloxy)piperidin-1-yl]-9H-purin-2-amine
N-{3-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]phenyl}acetamide
N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanamide
4-[(3R,4R)-4-amino-3-hydroxypiperidine-1-carbonyl]-7-fluoro-1,2-dihydroquinolin-2-one
(2E)-3-(3-fluorophenyl)-1-[3-(3-{[methyl(quinolin-6-ylmethyl)amino]methyl}phenoxymethyl)piperidin-1-yl]prop-2-en-1-one
3-(5-fluoro-2-methoxybenzoyl)-1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidine
N-[(2-chloro-6-fluorophenyl)methyl]-N-ethyl-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
4-[(2-ethyl-1,3-thiazol-4-yl)methyl]-9-(2-methoxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
3-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}(methyl)amino)propan-1-ol
N-(2-hydroxyethyl)-1-methyl-N-[(2-methylphenyl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
3-(5-methylthiophen-2-yl)-N-{3-[(pyridin-3-yl)amino]propyl}-1H-pyrazole-5-carboxamide
1-({5-[1-(5,6-dimethylpyrimidin-4-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1-(furan-2-ylmethyl)piperidine-4-carboxamide
2-(1-benzyl-3-oxopiperazin-2-yl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
(1s,4s)-4-hydroxy-N-[1-(4-methyl-1H-imidazol-2-yl)propyl]cyclohexane-1-carboxamide
4-[(1S,5R)-7-oxo-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]benzene-1-sulfonamide
2-(4-methyl-1H-imidazole-2-carbonyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-methyl-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-ethyl-4-[(2-methylpropyl)amino]pyrrolidine-2-carboxamide