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(2S)-2-({[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)-4-methylpentanamide
2-methoxy-5-oxo-6-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N,5-dimethyl-2-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzamide
6-[4-(pyridin-2-yl)butyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
5-cyclobutanecarbonyl-1'-(1H-pyrrole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-{4-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}pentan-1-ol
2-(2-fluorophenyl)-1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
1-{4-[6-(hydroxymethyl)-1,4-oxazepane-4-carbonyl]phenyl}pyrrolidin-2-one
1-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(2-methoxyphenyl)-1-{6-phenylimidazo[2,1-b][1,3]thiazole-3-carbonyl}pyrrolidine
N-(1-benzothiophen-5-ylmethyl)-3-(1,2-oxazolidin-2-yl)propanamide
5-methyl-N-[2-(4-phenylpyrimidin-2-yl)ethyl]-1,3,4-oxadiazol-2-amine
4-methyl-2-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
4-fluoro-N-({1-[2-(2-methoxyphenoxy)acetyl]piperidin-3-yl}methyl)benzamide
1-[1-butyl-3-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
(4aR,8aS)-6-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1-{[4-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}(methyl)[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]-1-[5-(propan-2-yl)-1,3-oxazole-4-carbonyl]piperidine
1-[(2,6-dimethoxyphenyl)methyl]-3-(4-ethyl-1H-pyrazol-5-yl)piperidine
(3S,4S)-4-(4-fluorophenyl)-1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperidin-3-ol
(2,1,3-benzoxadiazol-5-ylmethyl)({[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl})amine
2-cyclopropyl-4-methyl-5-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrimidine
(3R,4R)-1-{[5-(cyclohexylsulfanyl)furan-2-yl]methyl}-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
6-[(3-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-[3-(pyridin-4-yl)propanoyl]-1,4-diazepan-2-one
N-methyl-2-[(1-methyl-3-propyl-1H-pyrazol-5-yl)formamido]butanamide
2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-methyl-N-(thiophen-3-ylmethyl)acetamide
2-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-1H-indole
3-(methoxymethyl)-1-(3-methyl-5-propyl-1-benzofuran-2-carbonyl)piperidine
N-(3-chloro-4-fluorophenyl)-N'-{2-[(4-methylpyridin-2-yl)amino]ethyl}butanediamide
4-(2-cyclopentylacetyl)-6-[(3-methoxyphenyl)methoxy]-1-(pyridin-2-ylmethyl)-1,4-diazepan-2-one
2-(3-hydroxypropyl)-9-(pyrimidin-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2,2-dimethyloxan-4-yl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
6-chloro-2-{2-[3-(1H-imidazol-1-yl)propoxy]phenyl}-1H-1,3-benzodiazole
2-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-5-fluoro-N,N-dimethylpyrimidin-4-amine
5-cyclopropyl-3-{[2-(oxolan-3-yl)-1H-imidazol-1-yl]methyl}-1,2-oxazole
1-(4-hydroxy-2-phenylpyrimidine-5-carbonyl)piperidine-4-carbonitrile
2-({[(3R,4R)-4-(hydroxymethyl)-1-(3-methyl-1-benzothiophene-2-carbonyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
3-[5-(4-chloro-2-fluorobenzoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
2,6-dimethyl-5-{2-[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]-2-oxoethyl}-3,4-dihydropyrimidin-4-one
3-(pyridin-4-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-pyrazole-5-carboxamide
[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl][1-(2-methyl-1H-imidazol-1-yl)propan-2-yl]amine
3-{methyl[2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}propane-1,2-diol
2-methoxy-6-({4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazin-1-yl}methyl)phenol
2-[3-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]pyridin-3-ol
1-[(2E)-3-phenylprop-2-en-1-yl]-4-[2-(pyrrolidin-3-yl)benzoyl]piperazine
ethyl 1-(2,6-dimethylpyrimidine-4-carbonyl)-3-(2-phenylethyl)piperidine-3-carboxylate
1-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
1-(4-{[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
5-{[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]methyl}-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-4,4,4-trifluorobutanamide