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N,N-dimethyl-3-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]propane-1-sulfonamide
N-(1,4-dioxan-2-ylmethyl)-N,5-dimethyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-(1-ethylcyclopropyl)-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
4-(5-fluoropentyl)-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
[(3R,4R)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-[(5-methylfuran-2-yl)methyl]pyrrolidin-3-yl]methanol
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propylacetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-[4-({2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}amino)piperidin-1-yl]benzamide
{1-[2-methyl-2-(morpholin-4-yl)propyl]piperidin-4-yl}(thiophen-2-yl)methanol
2-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-N-[2-(4-methoxyphenyl)ethyl]acetamide
N-[2-chloro-5-(methylcarbamoyl)phenyl]-9-oxa-2-azaspiro[5.5]undecane-2-carboxamide
2-(3-{[4-(oxan-4-yl)piperazin-1-yl]methyl}phenoxy)acetamide
2-[4-(4H-1,2,4-triazol-4-yl)phenoxymethyl]pyridine
2-[1-(3-methylbutyl)-4-{[4-(methylsulfanyl)phenyl]methyl}piperazin-2-yl]ethan-1-ol
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-(6-methylpyridine-3-carbonyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
2-(4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1H-imidazol-2-yl}phenoxy)pyrimidine
2-(4-fluorophenoxy)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-[(2-methoxyphenyl)methyl]piperidine
3-(3,5-dimethoxyphenyl)-6-(1-methyl-1H-imidazol-2-yl)pyridazine
3-{[4-(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl)piperidin-1-yl]methyl}pyridine
4-benzyl-3-ethyl-1-[2-(1H-pyrazol-1-yl)acetyl]-1,4-diazepan-5-one
4-methyl-N-[2-(oxolan-2-ylmethoxy)phenyl]-1,4-diazepane-1-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-2-(pyridin-3-yl)ethane-1,2-dione
3-{1-[2-(4-chlorophenoxy)acetyl]piperidin-4-yl}-N-(3-methylphenyl)propanamide
2-({4-[(2-methoxyphenyl)methyl]piperazin-1-yl}methyl)-6-methylquinolin-4-ol
N-(1-{7-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)pyridine-2-carboxamide
ethyl 4-benzyl-1-(2,3-dihydroxypropyl)piperidine-4-carboxylate
(2R,3S,6R)-5-(dimethyl-1,3-thiazole-5-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(1-{[ethyl(oxolan-2-ylmethyl)carbamoyl]methyl}-1H-pyrazol-4-yl)pyridine-2-carboxamide
4-[4-(2,3-dihydro-1,4-benzodioxin-6-yl)phenyl]piperidin-4-ol
methyl 1-methyl-5-({[4-(methylsulfanyl)phenyl]methyl}amino)-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-(2-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)piperidin-2-one
N,N-bis(propan-2-yl)-2-[5-(trifluoromethyl)-1H-1,2,4-triazol-3-yl]benzamide
4-(5-methyl-1H-indol-3-yl)-6-(morpholin-4-yl)pyrimidin-2-amine
N-(1-{7-[(2-hydroxy-5-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
4-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-({[1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidin-3-yl]oxy}methyl)pyridine
2-(6-fluoro-4-methylquinolin-2-yl)benzamide
1-(5-methanesulfonyl-2-methylphenyl)-3-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}urea
1-[(3-methoxyphenyl)methyl]-4-[6-(trifluoromethyl)pyridin-2-yl]piperazin-2-one
6-methoxy-2-[3-(methylsulfanyl)propyl]-1,2,3,4-tetrahydroisoquinoline
5-methyl-N4-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]pyrimidine-2,4-diamine
7-{[2-(2-methoxyethyl)piperidin-1-yl]methyl}-1H-indole
2-({4-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)acetic acid
methyl 6-methyl-2-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyrimidine-4-carboxylate
2-phenyl-N-[1-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]acetamide
N-(pyridin-2-ylmethyl)-1-{1-[2-(pyrrolidin-1-yl)acetyl]piperidin-4-yl}piperidine-3-carboxamide
4-[5-({3-[(2-oxopyrrolidin-1-yl)methyl]piperidin-1-yl}methyl)-1,2,4-oxadiazol-3-yl]benzoic acid
2-phenyl-2-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,3-dihydro-1H-indene-1,3-dione
(1R,5R)-3-(3-chloro-2-fluorobenzoyl)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane