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N-(furan-3-ylmethyl)-5-(2-methoxyphenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
1'-(cyclohex-3-en-1-ylmethyl)-5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-methyl-4-{[4-(pyridin-4-yl)piperazin-1-yl]methyl}quinoline
{3-ethyl-1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]piperidin-3-yl}methanol
2-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-N-methylpyrimidin-4-amine
N-[(3S,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-tert-butyl-1-methyl-1H-pyrazole-5-carboxamide
3-methyl-4-{[3-(2-methylphenoxy)azetidin-1-yl]methyl}-1-(prop-2-en-1-yl)-1H-pyrazole
3-propoxy-1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine
N-(butan-2-yl)-5-methoxy-N-(pyridin-4-ylmethyl)-1H-indole-2-carboxamide
N-[(butylcarbamoyl)methyl]-2-(dimethylamino)-2-(4-fluorophenyl)-N-methylacetamide
3-hydroxy-N-[(1-{[1-(propan-2-yl)-1H-pyrrol-3-yl]methyl}pyrrolidin-3-yl)methyl]benzamide
4-{2-[(1-{4-[2-oxo-2-(pyrrolidin-1-yl)ethyl]phenyl}piperidin-4-yl)amino]ethyl}benzene-1-sulfonamide
N-[(1-hydroxycyclohexyl)methyl]-6-(2-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
(2S,4S)-N-ethyl-4-[(9H-purin-6-yl)amino]-1-(pyridin-2-ylmethyl)pyrrolidine-2-carboxamide
3-(oxolan-3-yl)-5-{pyrazolo[1,5-a]pyrimidin-2-yl}-1,2,4-oxadiazole
6-[(5-ethylpyrimidin-2-yl)amino]-2-methylheptan-2-ol
4-benzyl-3-ethyl-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-1,4-diazepan-5-one
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-[3-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]urea
N-(1-hydroxy-2-methylpropan-2-yl)-4-{[(3-methoxyphenyl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
N-tert-butyl-4-oxo-1-(propan-2-yl)-5-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
N-[1-(furan-2-carbonyl)piperidin-3-yl]-2-(1H-1,2,4-triazol-3-yl)benzamide
(2S)-N-[6-(dimethylamino)-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl]-2-(hydroxymethyl)pyrrolidine-1-carboxamide
(1S,5R)-3-methyl-6-{2-[(4-methylphenyl)methyl]benzoyl}-3,6-diazabicyclo[3.2.2]nonane
2-(dimethylamino)-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-2-(3-methylphenyl)acetamide
1-(2-ethylpyrimidine-5-carbonyl)-4-(2-methylquinolin-6-yl)piperidin-4-ol
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
8-(2,5-dimethylfuran-3-carbonyl)-2-(2-methylpropyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N,2-dimethyl-N-{2-phenyl-1-[1-(quinoxaline-6-carbonyl)piperidin-4-yl]ethyl}furan-3-carboxamide
1-[3-(pyridin-3-yl)azetidin-1-yl]-2-(3,4,5-trimethoxyphenyl)ethan-1-one
ethyl 4-(cyclopropylmethyl)-1-[2-(2,3,6-trifluorophenyl)acetyl]piperidine-4-carboxylate
N-(2-hydroxyethyl)-3,6-dimethyl-N-[(2E)-3-phenylprop-2-en-1-yl]-1-benzofuran-2-carboxamide
3-(2,4-difluorophenyl)-4-{[3-(2-fluorophenyl)pyrrolidin-1-yl]methyl}-1H-pyrazole
N-[2-(azepan-1-yl)ethyl]-6-methyl-4-oxo-N-(propan-2-yl)-1,4-dihydroquinoline-3-carboxamide
3-(2-hydroxyphenyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1H-pyrazole-5-carboxamide
2-[3-(1,3-benzoxazol-2-yl)piperidine-1-carbonyl]-8-fluoroquinoline
9-(2-methoxyethyl)-1-methyl-4-(thiophen-3-ylmethyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N,N-dimethyl-2-({[4-(3-methylphenyl)phenyl]carbamoyl}amino)butanamide
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methyl-N-[(5-phenyl-1H-pyrazol-4-yl)methyl]benzamide
(2R,3R,6R)-3-(4-fluorophenyl)-5-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-(oxan-4-ylmethyl)benzamide
N-[3-(1H-indazol-1-yl)propyl]-1-(2-methoxyethyl)-6-oxopiperidine-3-carboxamide
(2S)-2-[(4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}phenyl)formamido]-4-methylpentanamide
1-{1-azabicyclo[2.2.2]octan-3-yl}-3-(1-propyl-1H-1,2,3,4-tetrazol-5-yl)urea
2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-{[4-(trifluoromethoxy)phenyl]methyl}acetamide
(1R,5R)-6-benzyl-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(4aS,7aR)-1-[(3,4-dimethoxyphenyl)methyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-[cyclohexyl(methoxy)methyl]-4-(1-methyl-1H-pyrazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(methylsulfanyl)ethan-1-one
2-(thiophen-3-ylmethyl)-3-({trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)propan-1-ol