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N-{1-[3-(3,5-dimethylphenyl)propanoyl]piperidin-4-yl}methanesulfonamide
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-2-(phenylamino)pyrimidine-5-carboxamide
ethyl({[4-methoxy-3-(methoxymethyl)phenyl]methyl})({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)amine
5-{[5-(2,5-dimethyl-1-propyl-1H-pyrrol-3-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1H-1,2,4-triazole
3-{[3-cyclopropyl-1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]methyl}pyridine
3-amino-1-[(3,5-dichlorophenyl)methyl]pyrrolidine-3-carboxylic acid
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-6-(4-ethyl-1,4-diazepane-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N4-[1-(cyclohexylmethyl)piperidin-3-yl]-N1,N1-dimethylpiperidine-1,4-dicarboxamide
4-hydroxy-N-(2-methoxyethyl)-2-(4-methylphenyl)-N-(1-methylpiperidin-4-yl)pyrimidine-5-carboxamide
4-(5-methylpyrazine-2-carbonyl)-7-[(4-phenylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
(3S,4S)-1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
1-(3-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
4-(4-propylpyrimidine-5-carbonyl)-2-(trifluoromethyl)morpholine
5-(4-fluoro-3-methylphenyl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-phenyl-1H-imidazole
3-[({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}amino)methyl]-1-[(3,4-difluorophenyl)methyl]-3-hydroxypiperidin-2-one
6-(pyrrolidin-1-ylmethyl)-4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-1,4-oxazepan-6-ol
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-3-(4-methoxyphenyl)-3-phenylpropanamide
N-butyl-4-{[2-(dimethylamino)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
(3R,9aR)-3-[(benzylsulfanyl)methyl]-8-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]acetamide
8-fluoro-3-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1,4-dihydroquinolin-4-one
5-(2-methoxypyridin-4-yl)-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
(3aS,6aS)-2-(6-ethyl-5-fluoropyrimidin-4-yl)-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopent-1-ene-1-carboxamide
2-(3-hydroxypropyl)-9-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
4-(2-methylquinolin-6-yl)-1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-ol
5-(oxane-4-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
7-(1,3-benzothiazol-2-yl)-4-cyclobutanecarbonyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
[(4aS,8aR)-6-(6-phenylpyridazin-3-yl)-decahydro-1,6-naphthyridin-4a-yl]methanol
N-[3-(4-fluorophenyl)phenyl]-1-(furan-2-carbonyl)piperidine-3-carboxamide
(3aS,6aS)-2-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(furan-2-yl)-1-{3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}propan-1-one
methyl 8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(naphthalen-2-ylmethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
5-(3-acetylphenoxymethyl)-N-(1,3-dihydroxy-2-methylpropan-2-yl)-1,2-oxazole-3-carboxamide
2-tert-butyl-4-hydroxy-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]pyrimidine-5-carboxamide
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-1-(9H-purin-6-yl)piperidin-4-amine
1-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-4-(1H-pyrazol-1-yl)butan-1-one
{4-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]morpholin-2-yl}methanamine
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-methyl-N-[(4-methylphenyl)methyl]piperidine-4-carboxamide
3-methyl-1-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-phenylpiperidine
N-[(2-fluorophenyl)methyl]-5-[(3-hydroxy-2,2-dimethylpropyl)amino]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-(1-{[4-(1H-imidazol-1-yl)phenyl]methyl}pyrrolidin-2-yl)-3-(propan-2-yl)-1,2,4-oxadiazole
1-benzyl-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-2-carboxamide
N,N-dimethyl-2-[(1S,5R)-6-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
N1-[4-(1H-1,2,4-triazol-1-yl)phenyl]piperidine-1,3-dicarboxamide
N-[3-(2-fluorophenyl)propyl]-2-[4-(morpholin-4-yl)-6-oxo-1,6-dihydropyridazin-1-yl]acetamide
3-{[methyl({[2-(methylamino)pyrimidin-5-yl]methyl})amino]methyl}pyrrolidin-3-ol
(1R,2R,6S,7S)-N-[5-(2-methoxyacetamido)-2-methylphenyl]-4-azatricyclo[5.2.1.02,6]decane-4-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-3-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]propanamide