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N-[3-(piperidin-1-ylmethyl)phenyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2-(3,5-dimethyl-1H-pyrazol-1-yl)acetamide
7-[(3-methoxy-2-propoxyphenyl)methyl]-2-oxa-7-azaspiro[4.5]decan-8-one
3-(3,5-dimethylphenyl)-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]propan-1-one
N-(4-methylpentan-2-yl)-1-[4-(1,3-thiazol-4-yl)phenyl]piperidin-4-amine
1-[2-(methylamino)pyridine-4-carbonyl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
3-[(2R,3R,6R)-5-(5-methyl-1,2-oxazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N2-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-N4,N4,5-trimethylpyrimidine-2,4-diamine
5-(5-methylfuran-2-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,2,4-triazin-3-amine
3-(dimethylsulfamoyl)-5-{[(4-ethoxyphenyl)methyl]amino}-N-[3-(1H-imidazol-1-yl)propyl]benzamide
[(3-methyl-1H-pyrazol-5-yl)methyl][(1-methylpiperidin-3-yl)methyl](2-phenylethyl)amine
3-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-6-methyl-1,2-dihydropyridin-2-one
1-[1-ethyl-3-(4-phenylpiperazine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(2-fluorophenyl)ethan-1-one
7-(2-methoxyacetamido)-N,1-dimethyl-N-[2-(4-methylphenoxy)ethyl]-2-phenyl-1H-1,3-benzodiazole-5-carboxamide
2-{[5-(1-methoxyethyl)-4-(4-methylphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
2-(2-fluorophenyl)-4-(pyridin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(4-methoxyphenyl)-2,2-dimethyl-N-[(1r,4r)-4-hydroxycyclohexyl]cyclopropane-1-carboxamide
7-amino-4-[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]-1,2,3,4-tetrahydro-1,8-naphthyridin-2-one
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-5,6-dimethylpyridine-3-carboxamide
N-{[2-chloro-5-(trifluoromethyl)phenyl]methyl}-1-methylazepane-2-carboxamide
7-(2-methoxyethyl)-2-[(5-phenylthiophen-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2,8-dimethyl-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]quinoline-4-carboxamide
3-chloro-N-({4-[(4-fluorophenyl)methoxy]phenyl}methyl)-N-(pyridin-3-ylmethyl)benzamide
3-(1H-1,3-benzodiazol-5-yl)-1-ethyl-1-(oxan-4-ylmethyl)urea
2-methyl-4-(2-methylpropyl)-3-oxo-N-[4-(trifluoromethyl)phenyl]piperazine-1-carboxamide
3-[5-(1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)-1,2,4-oxadiazol-3-yl]pyridine
2-(2,3-dihydro-1H-inden-1-yl)-N-[1-(furan-2-carbonyl)piperidin-4-yl]acetamide
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3-[4-methyl-3-(2-oxopyrrolidin-1-yl)phenyl]urea
3-benzyl-1,8-dimethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-({[2-(cyclohexylsulfanyl)ethyl]carbamoyl}amino)-N,4-dimethylbenzamide
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(4-methylpiperazin-1-yl)ethyl]amine
N-[2-(ethylsulfanyl)ethyl]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-({4-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}amino)-3-methylbutan-1-ol
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-3-(4-methylphenyl)propan-1-one
4-[(2-fluorophenyl)methyl]-1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-(1-phenylbutyl)butanamide
8-cyclohexyl-1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{2-[4-(3-fluorophenoxy)piperidin-1-yl]pyrimidin-4-yl}pyrrolidin-3-ol
4-(1H-indazol-5-yl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
5-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)carbamoyl)-1H-imidazole-4-carboxylic acid
[(3-{2-[1-(3,5-dimethoxybenzoyl)piperidin-2-yl]ethoxy}phenyl)methyl](methyl)(quinolin-8-ylmethyl)amine
1-methyl-4-(1-{1-[2-(phenylsulfanyl)ethyl]piperidin-4-yl}ethyl)piperazine
N-(5-methylpyridin-3-yl)-3-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}benzamide
5-(propan-2-yl)-3-{1-[3-(1H-pyrazol-1-yl)benzoyl]pyrrolidin-2-yl}-1,2-oxazole
2-{3-[methyl(2-phenylethyl)amino]piperidine-1-carbonyl}pyridin-3-ol
N-{3-[5-methyl-4-({[3-(prop-2-en-1-yloxy)phenyl]formamido}methyl)-1,3-oxazol-2-yl]phenyl}oxane-4-carboxamide
N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
1-benzyl-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]piperidine-2-carboxamide
1-(benzenesulfonyl)-4-(pyrrolidin-3-ylmethyl)piperazine
ethyl 3-({3-[methyl(2-phenylethyl)amino]piperidine-1-carbonyl}amino)propanoate