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1-methyl-4-[1-(1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)ethyl]piperazine
dimethyl({5-[2-(pyrrolidine-1-carbonyl)piperazine-1-carbonyl]furan-2-yl}methyl)amine
N-benzyl-2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-hydroxyethyl)acetamide
6-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-N-(propan-2-yl)pyrimidin-4-amine
2-(4-chloro-2-{[(1,4-dioxan-2-ylmethyl)(methyl)amino]methyl}phenoxy)acetamide
N-(4-fluoro-2-methylphenyl)-3-[1-(1,3-oxazole-5-carbonyl)piperidin-3-yl]propanamide
3-[6-hydroxy-4-(1H-imidazole-5-carbonyl)-1,4-diazepan-1-yl]pyrazine-2-carbonitrile
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-methylbenzamide
1-cyclopentyl-4-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}pyrrolidin-2-one
3-[1-(3-fluorobenzoyl)piperidin-3-yl]benzoic acid
1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
N,8-dimethyl-N-(2-phenylethyl)-3-({[2-(propan-2-yloxy)ethyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
N-{2-[2-(trifluoromethoxy)phenyl]ethyl}oxane-2-carboxamide
2-cyclopropyl-6-methyl-3-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-1-(thiophen-2-ylmethyl)-1,4-dihydropyridin-4-one
N-[3-(4-chlorophenoxy)propyl]-1-cyclopropyl-N-methyl-5-oxopyrrolidine-3-carboxamide
6-methoxy-N-methyl-N-[3-(3-methylphenoxy)propyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-ethyl-N-(furan-2-ylmethyl)-N-methyl-5-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
methyl(oxolan-2-ylmethyl)[(2-phenyl-1H-imidazol-4-yl)methyl]amine
1-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-5-methyl-5-phenylpiperidin-2-one
2-({4-[4-(1H-pyrazol-1-yl)phenyl]phenyl}sulfanyl)acetamide
1,5-dimethyl-4-{[2-oxo-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]methyl}-1H-pyrrole-2-carbonitrile
1-(2-{1-[3-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl}ethyl)-1H-1,2,3,4-tetrazole
6-methoxy-N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
methyl N-(2-oxo-2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)carbamate
1-[(3-methylpyridin-2-yl)methyl]-4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperazine
3-(2-fluorophenyl)-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]propanamide
1-cyclohexyl-4-({4-[3-(dimethylamino)-2-hydroxypropoxy]phenyl}methyl)piperazin-2-one
2-[1-(oxolan-2-ylmethyl)-4-phenyl-1H-imidazol-5-yl]benzoic acid
(1s,4s)-4-{4-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carbonyl]-1H-1,2,3-triazol-1-yl}cyclohexan-1-amine
(2S,4R)-4-amino-N-methyl-1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]pyrrolidine-2-carboxamide
N-[(2R,3R)-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]cyclopropanecarboxamide
N,N-dimethyl-6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridazin-3-amine
N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-(2-methyl-1H-1,3-benzodiazol-1-yl)acetamide
2-amino-4-(3,4-dihydroxyphenyl)-6-(2-methylbutan-2-yl)pyridine-3-carbonitrile
6-ethyl-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
1-(oxolane-3-carbonyl)-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
2-[(adamantan-1-ylmethyl)(oxolan-3-ylmethyl)amino]ethan-1-ol
1-{1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
1-cyclopropyl-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
4-[2-(2-cyclopropyl-1H-imidazol-1-yl)ethyl]-1-ethyl-3,5-dimethyl-1H-pyrazole
N-(2-methoxyethyl)-6-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-1,6-dimethyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
N-[(2-fluorophenyl)methyl]-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(1-{5-[(2E)-but-2-en-1-yl]-1,3,4-oxadiazole-2-carbonyl}-3-(2-methylpropyl)piperidin-3-yl)methanol
(1S,5R)-3-[2-(benzyloxy)benzoyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
(1S,5R)-3-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(pyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
1-(2,5-dimethylphenyl)-5-(1,4-dioxan-2-yl)-3-(2-methylpropyl)-1H-1,2,4-triazole