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N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
4-{1-[2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]piperidin-3-yl}benzoic acid
N-[4-(furan-2-yl)phenyl]-4-[(3S,4R)-4-hydroxyoxolan-3-yl]-1,4-diazepane-1-carboxamide
3-{2-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-4-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-one
7-[2-(methylsulfanyl)acetyl]-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
methyl 2-{8-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-1-(2-methoxyethyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl}acetate
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-[(3-methylphenyl)methyl]-N-(oxolan-2-ylmethyl)acetamide
2-methyl-6-[4-(pyrrolidine-1-carbonyl)piperidine-1-carbonyl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
N-[(1-cyclopentylpiperidin-3-yl)methyl]-N-[2-(piperidin-1-yl)ethyl]-1H-imidazole-2-carboxamide
2-(3-{1-[3-(piperidin-1-yl)propyl]-1H-pyrazol-3-yl}phenyl)pyrazine
3-[5-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
(1H-imidazol-2-ylmethyl)(methyl){4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
N,N-dimethyl-4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperazine-1-carboxamide
6-(furan-2-yl)-3-(oxolan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
1-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-3-(thiophen-3-yl)propan-1-one
2-methoxy-3-{1-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-1H-imidazol-2-yl}quinoline
2-[(4aR,7aS)-4-[(2-chloro-5-fluorophenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
3-(1,3-benzothiazol-2-yl)-N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]propanamide
1-(2-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1'-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-(1-benzofuran-2-yl)-N-[2-(morpholin-4-yl)ethyl]-1,2,4-triazin-3-amine
1-methyl-N-(morpholin-2-ylmethyl)-1H-indole-4-carboxamide
5-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]-2,3-dihydro-1H-pyrazol-3-one
1-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-3-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)urea
N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-3-(5-methylthiophene-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2,3-dihydro-1H-inden-2-yl)-3-({[5-(methoxymethyl)furan-2-yl]methyl}amino)-5-[(propan-2-yl)sulfamoyl]benzamide
4-{7-cyclopentyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl}-1λ6-thiane-1,1-dione
4-(oxolane-3-carbonyl)-7-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
dimethyl({4-[(6-phenylpyridazin-3-yl)oxy]phenyl}methyl)amine
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-2-(1H-1,2,4-triazol-1-yl)propanamide
2-(1H-indazol-3-yl)-N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]acetamide
1-{[2-(2-butyl-1H-imidazol-4-yl)-1H-imidazol-1-yl]methyl}cyclohexan-1-ol
2-(4-benzyl-2-oxopyrrolidin-1-yl)-N-(3-cyclopentylpropyl)-N-methylacetamide
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-methylfuran-3-carboxamide
methyl[(3-methylpyridin-4-yl)methyl]{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}amine
7-[(2-fluorophenyl)methyl]-2-(2-methoxyacetyl)-2,7-diazaspiro[4.5]decan-6-one
3-(2-ethylbutyl)-8-[2-(methylsulfanyl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[2-(2-propyl-1,3-thiazole-4-carbonyl)-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-1-yl]pyridine
5-(3-methoxyphenoxymethyl)-3-{octahydro-1H-pyrido[1,2-a]piperazine-2-carbonyl}-1,2-oxazole
4-{1-[1-(4-methyl-1,3-thiazol-2-yl)piperidin-4-yl]ethyl}morpholine
(2R)-2-amino-N-(1H-imidazol-2-ylmethyl)-N-methyl-2-phenylacetamide
4-{1-[1-(2-methyl-1-benzofuran-7-carbonyl)piperidin-4-yl]ethyl}morpholine
(1R,3S)-3-{[(4,6-dimethylpyridin-2-yl)methyl](methyl)carbamoyl}cyclopentane-1-carboxylic acid
5-methoxy-9-(4-methylpyrimidin-2-yl)-1-oxa-9-azaspiro[5.5]undecane
[2-(1H-imidazol-1-yl)ethyl]({[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl})methylamine
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
{2-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-8-methylquinolin-3-yl}methanol
1-cyclopropyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-5-oxopyrrolidine-3-carboxamide