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2-[(4aS,8aR)-1-[2-(methylamino)ethyl]-2-oxo-decahydro-1,6-naphthyridin-6-yl]-1,3-thiazole-4-carboxamide
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(8-methoxy-2H-chromen-3-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-N,N-diethyl-5-(furan-2-yl)-1H-pyrazole-4-carboxamide
dimethyl[(4-{1-[(5-methylfuran-2-yl)methyl]piperidin-2-yl}phenyl)methyl]amine
1-[2-(1-ethyl-3-oxopiperazin-2-yl)acetyl]-4-phenylpiperidine-4-carbonitrile
1-({3-[2-hydroxy-3-(4-methylpiperazin-1-yl)propoxy]-4-methoxyphenyl}methyl)piperidine-4-carbonitrile
5-[4-(1,3-benzothiazol-2-yl)piperazine-1-carbonyl]-N-butyl-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
(3S,5S)-5-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine-3-carbonyl)-1-methylpyrrolidin-3-amine
2-(4-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperazin-1-yl)-1-(pyrrolidin-1-yl)ethan-1-one
2-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
2-amino-N-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-6-(propan-2-yl)pyrimidine-4-carboxamide
{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}(methyl)[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amine
[5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]methanol
N,N-dimethyl-4-[2-(2,4,7-trimethyl-1H-indol-3-yl)acetamido]butanamide
3-[(3R,4S)-4-(dimethylamino)-1-[3-(dimethylamino)benzoyl]piperidin-3-yl]propan-1-ol
1-(3-{[3-(2-chlorophenoxy)azetidin-1-yl]methyl}phenyl)ethan-1-one
2-{3-[4-(methylsulfanyl)phenyl]-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl}-1,2,3,4-tetrahydroisoquinoline
2-{2-[methyl(pyridin-2-ylmethyl)amino]acetyl}-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-{4-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]morpholin-3-yl}-N-phenylacetamide
4-(3-hydroxy-3-methylbutyl)-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}benzamide
2,5-dimethoxy-N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzene-1-sulfonamide
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-2-(3-methoxyphenyl)azetidine
1-(1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carbonyl)azepane
N-cyclopentyl-3-fluoro-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}benzene-1-sulfonamide
1-({5-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
3-(2-oxo-2-{7-[(4-phenylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}ethyl)-1,3-thiazolidine-2,4-dione
4-methyl-2-({methyl[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]amino}methyl)phenol
(1S,4S)-2-(2-methoxy-5-phenylphenyl)-5-[2-(5-methyl-1H-pyrazol-1-yl)ethyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
N-[(1-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carbonyl}piperidin-3-yl)methyl]furan-2-carboxamide
1-(pyridin-4-ylmethyl)-4-(thiophen-3-ylmethyl)-1,4-diazepane
ethyl({[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl})(pyridin-4-ylmethyl)amine
6-{[benzyl(butyl)amino]methyl}-N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
3-{2-[1-(2-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-oxoethyl}-3,4-dihydroquinazolin-4-one
2-(2-methoxyethyl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1,3-benzoxazole-6-carboxamide
N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
7-[(2,3-difluorophenyl)methyl]-2-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-2,7-diazaspiro[4.5]decane
1-[2-(4-fluorophenyl)ethyl]-4-[(propan-2-yl)amino]pyrrolidin-2-one
1-{3-oxo-3-[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]propyl}-1,2-dihydropyridin-2-one
3-benzyl-8-(1H-indol-2-ylmethyl)-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{2-[(6-methyl-2-propylpyrimidin-4-yl)amino]ethyl}pyrrolidine-2,5-dione
4-(5-{1-oxa-8-azaspiro[4.5]decane-8-carbonyl}-1H-pyrazol-3-yl)phenol
5-{7-[(4-phenylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl}pyrrolidin-2-one
3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)-N-[1-(thiophen-2-yl)ethyl]propanamide
[(2-ethyl-3-methyl-1H-indol-5-yl)methyl][(3-phenyl-1H-pyrazol-4-yl)methyl]amine
[1-(1-{[2-(trifluoromethoxy)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]methanamine
2-amino-4-ethyl-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-1,3-thiazole-5-carboxamide
5-[2-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-1,3,4-thiadiazol-2-amine
9-[6-(morpholin-4-yl)pyrimidin-4-yl]-3-oxa-9-azaspiro[5.5]undecane
2-{[2-(2-ethoxyphenoxy)ethyl](methyl)amino}acetic acid
methyl 4-[4-(1H-pyrazole-3-carbonyl)piperazin-1-yl]benzoate