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methyl (2S,4R)-4-(2-cyclopropylquinoline-4-amido)-1-(3-phenylpropyl)pyrrolidine-2-carboxylate
8-[(3-methylphenyl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
N-methyl-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}-N-(pyrazin-2-ylmethyl)acetamide
2-(3-fluorophenoxymethyl)-4-[3-(1H-pyrazol-1-yl)azetidine-1-carbonyl]-1,3-oxazole
(2-{[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl][(2-methylphenyl)methyl]amino}ethyl)dimethylamine
1-[5-(furan-2-ylmethyl)-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-1,4-diazepan-5-one
methyl 2-[2-(3,5-dimethyl-1-benzofuran-2-yl)-1H-imidazol-1-yl]acetate
4-({5-[1-(oxolan-2-ylmethyl)-1H-1,2,3-triazol-4-yl]-1,2,4-oxadiazol-3-yl}methyl)-1-propylpiperidine
(1R,5R)-3-benzoyl-6-(4-phenoxybutyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(2R,3R)-2-methoxy-1'-[(2E)-3-phenylprop-2-en-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
3-{4-[1-ethyl-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}-1λ6-thiolane-1,1-dione
3-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}propan-1-one
1-(3-phenylpropyl)-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-{2-[1-(2H-1,3-benzodioxol-5-ylmethyl)-1H-1,2,4-triazol-5-yl]ethyl}-N-methylmethanesulfonamide
2-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-5-methoxy-4H-pyran-4-one
5-({3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}methyl)-N-methylfuran-2-carboxamide
3-[5-(pyridin-3-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-4-methyl-N-(oxolan-2-ylmethyl)-1,2,5-oxadiazole-3-carboxamide
2-(3,5-difluorophenyl)-1-[3-(1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
N-{[6-chloro-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}-2,3-dimethoxybenzamide
4-{methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]sulfamoyl}-N-propylbenzamide
3-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3,5-dimethylphenyl)urea
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]acetamide
6-(cyclopropylmethoxy)-1-[(3-methoxyphenyl)methyl]-4-(thiophene-3-carbonyl)-1,4-diazepan-2-one
4-[(3,4-dimethoxyphenyl)methyl]-3-[2-oxo-2-(3-oxopiperazin-1-yl)ethyl]piperazin-2-one
2-{[(3-ethoxyphenyl)methyl][(2E)-3-(furan-2-yl)prop-2-en-1-yl]amino}ethan-1-ol
2-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-4-methylphenol
(1S,5R)-6-(cyclobutylmethyl)-3-(3,5-difluoropyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{2-[(4-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-3-yl}-5-methylpyrimidin-2-yl)sulfanyl]ethyl}morpholine
1-[({[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}amino)methyl]cyclohexan-1-ol
4-{5-[2-(1H-1,2,4-triazol-1-yl)ethyl]-1,2,4-oxadiazol-3-yl}-1H-indole
N-(furan-2-ylmethyl)-7-(2-methoxyacetamido)-N-methyl-1-(2-phenylethyl)-1H-1,3-benzodiazole-5-carboxamide
methyl 5-{2-[(1R,4R)-2-azabicyclo[2.2.1]heptan-2-yl]acetyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
5-methyl-3-[2-(morpholin-4-ylmethyl)phenyl]pyridin-2-amine
2-{[3-(pyridin-3-yl)azetidin-1-yl]methyl}-1H-indole
1-{3-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(1-methyl-1H-pyrazole-4-carbonyl)piperidine
4-{4-[(2,3-dimethoxyphenyl)methyl]piperazin-1-yl}-2-{[4-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
N-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-[3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propyl]-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(2R,6R)-4-(2,5-dimethylbenzoyl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-(1-{1-[(3-chloro-4-hydroxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxybenzamide
methyl 4-({1-ethyl-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-8-yl}methyl)thiophene-2-carboxylate
N-methyl-3-[(1,4-oxazepan-6-ylmethyl)sulfamoyl]benzamide
ethyl 5-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylate
4-{3-[2-(3,4-difluorophenyl)ethyl]piperidine-1-carbonyl}-2-methylphenol
methyl 2-[(cyclohexylmethyl)sulfamoyl]-6-(6-methylpyridine-2-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-[(1S,5R)-6-[(2-cyanophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
1-[4-(3-methoxyphenoxy)phenyl]-3-methyl-3-(1-methylpiperidin-4-yl)urea
N-[(2-methyloxolan-2-yl)methyl]-2-[(prop-2-en-1-yl)amino]benzamide