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3-methyl-1-[1-(6-{[(3-methyl-1,2-oxazol-5-yl)methyl]amino}pyridine-3-carbonyl)piperidin-3-yl]butan-1-one
3-chloro-4-({4-[2-(methylsulfanyl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)pyridine
3-benzyl-8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1,6-dimethyl-N-[1-(thiophen-3-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-4-(1H-imidazol-2-yl)piperidine
N-[(3-hydroxypyrrolidin-3-yl)methyl]-2-methyl-4-phenylpyridine-3-carboxamide
3-methyl-1-(2-methyl-1-benzofuran-5-yl)-3-[(trimethyl-1H-pyrazol-4-yl)methyl]urea
7-[(3,4-difluorophenyl)methyl]-2-(pyrimidin-2-yl)-2,7-diazaspiro[4.5]decane
N-[(2-methylphenyl)methyl]-N-(prop-2-en-1-yl)isoquinoline-5-carboxamide
3-(2-methoxyethyl)-3H,4H-thieno[3,2-d]pyrimidin-4-one
9-[6-(dimethylamino)pyridine-3-carbonyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(2-methoxyethyl)-5-(1H-1,2,3-triazol-1-ylmethyl)-1-[3-(trifluoromethyl)phenyl]-1H-1,2,4-triazole
ethyl 1-{[7-fluoro-2-oxo-1-(pyridin-2-ylmethyl)-1,2-dihydroquinolin-3-yl]methyl}piperidine-4-carboxylate
methyl 5-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-5-oxopentanoate
3-({5-[1-(furan-2-ylmethyl)-1H-imidazol-2-yl]furan-2-yl}sulfanyl)-4-methyl-4H-1,2,4-triazole
8-acetyl-2-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-{[5-(2,2-dimethyloxan-4-yl)-1,2,4-oxadiazol-3-yl]methyl}-4-methylpiperazine
1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]-2-(thiophen-3-yl)ethan-1-one
5-{[2-(2-ethyl-1H-1,3-benzodiazol-1-yl)butanamido]methyl}-1,2,4-oxadiazole-3-carboxamide
2-{4-[(8-methoxyquinolin-2-yl)methyl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
2-amino-1-{4-[(2,5-dimethoxyphenyl)methyl]piperazin-1-yl}-2-(3,5-dimethyl-1H-pyrazol-4-yl)ethan-1-one
3-(1-{1-[(3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methylphenyl)urea
8-[(dimethyl-1,2-oxazol-4-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
1-methyl-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}azepane-2-carboxamide
1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-3,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
(3aS,6aR)-5-(2-amino-6-methylpyrimidin-4-yl)-3-[3-(4-fluorophenyl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
3-(1-methylpiperidin-3-yl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)propanamide
6-fluoro-N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-methyl-N-[2-(morpholin-4-yl)ethyl]benzamide
4-[(4-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}furan-2-yl)methyl]morpholine
5-[(2,3-dihydro-1-benzofuran-5-ylmethyl)amino]-4,6-dimethyl-1,2-dihydropyridin-2-one
(2S)-2-[(5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)amino]propanamide
2-(azepan-1-yl)-N-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]acetamide
N-(1H-1,3-benzodiazol-2-yl)-2-{[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]amino}acetamide
1-{[3-(1-methyl-1H-1,2,4-triazol-5-yl)phenyl]methyl}azepane
8-chloro-2-ethyl-4-(4-fluorobenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-phenoxy-1-(4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperazin-1-yl)ethan-1-one
1-(2-chloro-4-fluoro-5-methylphenyl)-3-[(1-ethylpyrrolidin-2-yl)methyl]urea
2-(2-methoxyethyl)-N-methyl-N-(naphthalen-1-ylmethyl)-1,3-benzoxazole-6-carboxamide
4-benzyl-1-[(1-methyl-1H-pyrazol-5-yl)methyl]piperidine
4-methyl-1-{2-[(1S,5R)-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-1,2-dihydroquinolin-2-one
8-methoxy-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[(3,4-difluorophenyl)methyl]-3-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}propanamide
9-(2-methylpyrimidine-5-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
[(2-phenoxypyridin-3-yl)methyl]({[3-(1H-pyrazol-1-yl)phenyl]methyl})amine
4-(2,4-dimethoxyphenyl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N4-[1-(benzenesulfonyl)piperidin-4-yl]-5-methylpyrimidine-2,4-diamine