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1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(thiophene-2-carbonyl)piperazine
3-(7-chloro-4-hydroxyquinoline-3-carbonyl)-3,9-diazaspiro[5.6]dodecan-10-one
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-[(2-ethyl-6-methylpyridin-3-yl)oxy]ethan-1-one
N-(3-chloro-4-fluorophenyl)-3-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)propanamide
1-(adamantan-1-yl)-4-[(2-methyl-1,3-oxazol-4-yl)methyl]piperazine
5-[cyclohexyl(pyridin-3-ylmethyl)carbamoyl]thiophene-2-carboxylic acid
1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2-(methoxymethyl)piperidine
N,6-dimethyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1,3-benzothiazol-2-amine
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-3-methoxy-N-methylpropanamide
1-(2-phenylethyl)-4-(pyridin-3-yl)piperazine
N,N-diethyl-1-[(1s,4s)-4-(thiophene-2-amido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-[4-(2-aminopyrimidin-4-yl)-1-[(4-ethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
1-[(2-ethylpyrimidin-5-yl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
1-methyl-4-{3-methyl-5-[4-(1H-pyrazol-3-yl)phenyl]-1H-1,2,4-triazol-1-yl}piperidine
1-[benzyl(methyl)amino]-3-[4-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
2-cyclopropyl-9-[(6-methylpyridin-2-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
2-(2,3-dihydro-1H-inden-1-yl)-N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-1-(carbamoylmethyl)piperidine-4-carboxamide
N-{1-[1-(1,4-dithiepan-6-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
3-[2-(azepan-1-yl)-2-oxoethyl]-4-[(2-chloro-4-fluorophenyl)methyl]piperazin-2-one
6-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
1-(3-{7-methyl-4-oxo-3H,4H-thieno[3,2-d]pyrimidin-3-yl}propyl)piperidine-3-carboxamide
3-(1-cyclohexylpiperidin-3-yl)-N-(3,5-dimethoxyphenyl)propanamide
1-(2-methoxy-4-{[(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)amino]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
1-[(1R,5S,6R)-6-[({[4-(methylsulfanyl)phenyl]methyl}(prop-2-en-1-yl)amino)methyl]-3-azabicyclo[3.1.0]hexan-3-yl]ethan-1-one
2-(4-chloro-2-methylphenoxy)-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]acetamide
(3aS,6aS)-2-[(benzylcarbamoyl)methyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[3-(azepan-1-yl)propyl]-N,2-dimethyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-cyclohexyl-N3-cyclopropyl-N5-[(2,3-dimethoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-{4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
5-methoxy-3-methyl-2-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}-1H-indole
2,2-dimethyl-N-(5-methyl-3-{4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}thiophen-2-yl)propanamide
N,N-dimethyl-5-[(2-phenylethyl)amino]-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-5-[4-(trifluoromethyl)phenyl]-1,2,4-triazin-3-amine
N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N,3-dimethylfuran-2-carboxamide
2-[2-(1-methyl-1H-imidazol-4-yl)ethyl]-1-oxo-N-(pyridin-2-ylmethyl)-2,3-dihydro-1H-isoindole-4-carboxamide
(1S,4S)-2-{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}-2-azabicyclo[2.2.1]heptane
1-ethyl-3-(pyridin-2-ylmethyl)-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]-1-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]urea
3-[3-(dimethylamino)propyl]-8-[2-(4-methyl-1H-pyrazol-1-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(4aR,7aS)-1-(cyclopropylmethyl)-4-[2-(methylamino)-1,3-thiazole-4-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[(2-fluorophenyl)methyl]-N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-1,3-benzoxazole-6-carboxamide
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(2-fluorophenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
(1R,5R)-3-(3-chloro-4-fluoro-1-benzothiophene-2-carbonyl)-3,9-diazabicyclo[3.3.2]decan-10-one
methyl 2-[1-(2-methoxyethyl)-2,4-dioxo-8-[(3-phenoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-[2-(1H-imidazol-1-yl)ethyl]piperazine
5-(2,4-difluorophenoxymethyl)-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1,2-oxazole-3-carboxamide
5-[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidine-1-carbonyl]-3,4-dihydropyrimidin-4-one
(2S,4R)-4-amino-1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-{[(1R,3S,5S)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octan-8-yl]methyl}-1,5-dimethyl-1H-pyrrole-2-carbonitrile