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5-fluoro-2-{1-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
N-cyclooctyl-4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}benzamide
N-cyclopropyl-2-{[2-(4-fluorophenyl)imidazo[1,2-a]pyridin-6-yl]formamido}acetamide
4-{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}-3-ethylpiperazin-2-one
1-[2-(3-benzoylpiperidin-1-yl)pyrimidin-4-yl]piperidin-4-ol
N-{3-oxo-3-[(2R,6S)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]propyl}acetamide
5-[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-4-yl]-3-cyclopentyl-5-[(4-fluorophenyl)methyl]imidazolidine-2,4-dione
2-{6-[4-(benzenesulfonyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}ethan-1-amine
ethyl 4-{1-[(2-fluorophenyl)methyl]-6-oxopiperidine-3-amido}piperidine-1-carboxylate
N-benzyl-3-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]oxy}benzamide
2-[({2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}amino)methyl]-6-methylquinolin-4-ol
N-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-N-methyl-2-(naphthalen-2-yloxy)propanamide
3-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1-[4-(2-methyl-1H-imidazol-1-yl)phenyl]urea
N-[1-(pyrimidin-2-yl)piperidin-3-yl]-2-(pyrimidin-2-ylsulfanyl)acetamide
4-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-2-(4-chlorophenyl)morpholine
(2S)-1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-methyl-2-(propan-2-yl)piperazine
4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-1-(2-methyl-1-benzofuran-5-carbonyl)piperidine
methyl (2S,4S)-1-(2-methylpropyl)-4-{2-[4-(trifluoromethyl)phenyl]benzamido}pyrrolidine-2-carboxylate
2-(4-fluorophenyl)-N-(2-{7-[(2,4,5-trimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
4-[2-(4-fluorophenyl)piperidine-1-carbonyl]benzonitrile
1-[2-(ethanesulfonyl)ethyl]-2-(6-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazole
2-(pyrrolidine-1-carbonyl)-1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperazine
N-(1-{2-oxo-2-[2-(pyridin-2-yl)piperidin-1-yl]ethyl}-1H-pyrazol-4-yl)-2H-1,3-benzodioxole-5-carboxamide
4-[2-(4-fluorophenoxy)ethyl]-1-[5-(4-methoxyphenyl)furan-2-carbonyl]-1,4-diazepan-5-one
1-[4-(5-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-yl]azepane
8-fluoro-N-(2-methoxyethyl)-N-(pyridin-3-ylmethyl)quinoline-2-carboxamide
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
(1S,5R)-6-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-({3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}methyl)phenol
{4-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]morpholin-2-yl}methanamine
(3aS,6aR)-5-(1-benzofuran-2-carbonyl)-3-[(2-methoxyphenyl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-3,9-diazaspiro[5.5]undecane
2-{[4-(4-methoxy-3-methylphenyl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
N-{2-[(6-methyl-2-phenylpyrimidin-4-yl)amino]ethyl}acetamide
9-(propane-2-sulfonyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
8-[6-(propan-2-yl)-2-(trifluoromethyl)pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
6-{4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}quinoxaline
2-{2-[4-(2-chlorophenyl)-4H-1,2,4-triazol-3-yl]ethyl}phenol
1-ethyl-3-(thiomorpholine-4-carbonyl)-N-[2-(thiophen-2-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-{9-[(2-ethylphenyl)carbamoyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
1-(2-methoxy-5-{[methyl(2-methylprop-2-en-1-yl)amino]methyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
2-methoxy-4-({[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}amino)pyridine-3-carbonitrile
2-(hydroxymethyl)-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-1H-1,3-benzodiazole-5-carboxamide
5-[3-(pyridin-3-yl)propanoyl]-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]pyridine-4-carboxamide
N-(1,2-diphenylethyl)-2-(ethylamino)pyrimidine-5-carboxamide
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(2-methoxyethyl)piperidine
{1-[8-chloro-2-(furan-2-yl)quinoline-4-carbonyl]-2,5-dihydro-1H-pyrrol-2-yl}methanol
6-(naphthalene-1-carbonyl)-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
(5S,9aS,9bS)-5-(2-fluoro-4-methoxyphenyl)-2-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one