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N-(2-hydroxyethyl)-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
4-[({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)amino)methyl]-1H-pyrrole-2-carbonitrile
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(3R,5S)-5-[4-(4-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]pyrrolidin-3-ol
N-{3-[({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}carbamoyl)methoxy]phenyl}propanamide
methyl (2S)-2-{[2-(phenoxymethyl)-1,3-oxazol-4-yl]formamido}-2-phenylacetate
(cyclopropylmethyl)({[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})(oxolan-2-ylmethyl)amine
3-(2-ethyl-1H-1,3-benzodiazol-1-yl)-1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]propan-1-one
(3aR,6aS)-2-ethyl-1-oxo-5-[(2-phenylethyl)carbamoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-(dimethylamino)ethyl]-3-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}propanamide
1-[(3,5-dimethylphenyl)methyl]-4-[3-(hydroxymethyl)-8-methylquinolin-2-yl]piperazin-2-one
(1R,3S,5S)-8-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)-8-azabicyclo[3.2.1]octan-3-ol
2-cyclopropyl-6-[4-(2-phenylethyl)piperidine-1-carbonyl]-1,3-benzoxazole
4-fluoro-3-{5-[1-hydroxy-3-(methylsulfanyl)propyl]-3-methyl-1H-1,2,4-triazol-1-yl}benzene-1-sulfonamide
7-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-(6-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}pyridin-2-yl)ethan-1-ol
6-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
1-{3-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{3-[(4-methoxyphenyl)methyl]-5-{[(4-methyl-1,3-thiazol-2-yl)sulfanyl]methyl}-1H-1,2,4-triazol-1-yl}ethan-1-ol
3-({5-[1-(1,3-dihydro-2-benzofuran-5-yl)-1H-imidazol-2-yl]furan-2-yl}sulfanyl)-4-methyl-4H-1,2,4-triazole
(3S,4S)-3-[({3-[(3-fluorophenyl)methoxy]-4-methoxyphenyl}methyl)amino]-4-hydroxy-1λ6-thiolane-1,1-dione
(4S)-N-[2-(2-fluorophenyl)ethyl]-4-hydroxy-3,3,4-trimethylpiperidine-1-carboxamide
N-(2-methoxyethyl)-5-{1-[(2E)-3-phenylprop-2-enoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
4-(benzyloxy)-1-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
N-[1-(2,4-dimethoxyphenyl)ethyl]-2-(1H-imidazol-2-yl)-N-methylbenzamide
1-[2-(4-chlorophenyl)morpholin-4-yl]-2-(methylamino)ethan-1-one
4-{4-[(2-methylphenyl)methyl]piperazin-1-yl}-6-(pyrrolidin-1-yl)pyrimidin-2-amine
4-[(5-{1-[(5-ethylpyridin-2-yl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]morpholine
N,N-dimethyl-2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carboxamide
N-(1-carbamoylcyclopentyl)-3-(1H-pyrazol-4-yl)benzamide
3-(5-{imidazo[1,2-a]pyrimidin-2-yl}-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl)-1λ6-thiolane-1,1-dione
4-chloro-5-{[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-3-methyl-1H-pyrazole
dimethyl[2-({[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}(thiophen-3-ylmethyl)amino)ethyl]amine
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylpyrazine-2-carboxamide
2,7,8-trimethyl-4-[3-(piperidin-1-yl)azetidine-1-carbonyl]quinoline
N-[(3-ethoxyphenyl)methyl]-2-(2-hydroxyphenoxy)-N-(prop-2-en-1-yl)acetamide
3-[2-(2-methylpropanesulfonyl)ethyl]-1-[2-(trifluoromethoxy)phenyl]urea
1-{1-[3-(5-methylfuran-2-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]ethyl}pyrrolidin-2-one
N-{2-[7-(1H-indol-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-4-methoxybenzamide
1-[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N2-(1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)-N1-(pyridin-3-yl)ethane-1,2-diamine
3-cyclopropyl-1-[4-ethoxy-3-(1H-pyrrol-1-yl)phenyl]-3-[(1-methyl-1H-imidazol-2-yl)methyl]urea
methyl 4-{2-chloro-4-[(2-methoxyethyl)carbamoyl]phenoxy}piperidine-1-carboxylate
2-(5-chloro-6-methyl-1-benzofuran-3-yl)-1-[3-(1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-4-yl}(1-methyl-1H-imidazol-2-yl)methanol
2-{1,9-dimethyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}-N-[2-(4-methoxyphenyl)ethyl]acetamide
6-{1-[1-(oxan-4-yl)piperidine-4-carbonyl]piperidin-3-yl}pyrimidin-4-ol
4-[(dimethylamino)methyl]-1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-ol
4-(4-{[3-(morpholin-4-yl)piperidin-1-yl]methyl}phenyl)but-3-yn-1-ol