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8-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
4-(1-methylpiperidin-4-yl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(1H-pyrazole-3-carbonyl)pyrrolidin-3-yl]methanol
9-(cyclopropylmethyl)-1-methyl-4-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]-1,4,9-triazaspiro[5.6]dodecan-10-one
7-(1,3-benzothiazol-2-yl)-4-(oxolan-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-ethyl-N-{[1-(methoxymethyl)cyclopropyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
2-[2-(1H-imidazol-4-yl)ethyl]-8-(5-methylpyridin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-butyl-7-fluoro-2-methyl-N-(pyridin-2-ylmethyl)quinoline-4-carboxamide
(3R,4R)-4-ethyl-1-[5-(1H-indol-1-ylmethyl)furan-2-carbonyl]piperidine-3,4-diol
3-(3-hydroxyquinoxalin-2-yl)-1-[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]propan-1-one
2-[methyl(2-phenylethyl)amino]-N-(oxan-3-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
(2R,3R)-3-[4-(4-fluorophenyl)-1H-1,2,3-triazol-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-(2-fluorophenyl)-1H-pyrazole-5-carboxamide
2-tert-butyl-6-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyloxane-4-carboxamide
2-{4-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]piperazin-1-yl}pyridine-3-carbonitrile
2-{4-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]morpholin-3-yl}acetic acid
2-methoxy-6-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]phenol
4-[(4-methyl-1H-imidazol-5-yl)methyl]-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]acetamide
N-methyl-N-[(5-methylfuran-2-yl)methyl]-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-(2-oxopiperidin-3-yl)benzamide
N-(2-methoxyphenyl)-3-[(1,2-oxazol-5-ylmethyl)sulfamoyl]benzamide
4-benzyl-3-ethyl-1-{[5-(hydroxymethyl)furan-2-yl]methyl}-1,4-diazepan-5-one
3-(1H-pyrazol-1-yl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]benzamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(4-methyl-1H-pyrrole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[2-(2-methoxy-4-methylphenoxy)ethyl]-1-(4-methoxyphenyl)-5-methylpiperazin-2-one
3-ethyl-8-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-methyl-N-[(2-phenoxypyridin-3-yl)methyl]azepane-2-carboxamide
1-[1-(4-fluorobenzoyl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
N-{2-[2-(2,3,4-trifluorophenyl)-1H-imidazol-1-yl]ethyl}acetamide
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(1H-imidazol-1-yl)propan-1-one
5-methyl-3-{3-[3-(1H-pyrazol-3-yl)phenyl]phenyl}-1,2,4-oxadiazole
3-methyl-7-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl](2-methoxyethyl)[(2E)-3-phenylprop-2-en-1-yl]amine
3-(2-methyl-1H-imidazol-1-yl)-N-[1-(3-methylphenyl)piperidin-4-yl]butanamide
2-(3-fluoro-4-hydroxyphenyl)-1-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonan-7-yl]ethan-1-one
(2R,6R)-4-[3-(piperidin-1-yl)propanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[2-(4-methylphenoxy)ethyl]amine
4-(1-{[2-(2-hydroxyethoxy)phenyl]methyl}piperidin-3-yl)benzoic acid
dimethyl[(4-methyl-5-{1-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]piperidin-3-yl}-4H-1,2,4-triazol-3-yl)methyl]amine
2-(1,2-benzoxazol-3-yl)-1-(1,2-oxazinan-2-yl)ethan-1-one
methyl 3-({1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidin-3-yl}formamido)propanoate
1-{4-[4-(pyridin-4-yl)piperidin-1-yl]piperidin-1-yl}butan-1-one
N-{[1-(3,5-dimethylphenyl)cyclopentyl]methyl}-3-(pyridin-4-yl)propanamide
3-{[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl](methyl)amino}-N-methylpropanamide
1-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl]pyrazine-2-carboxamide
6-fluoro-2-{[3-(2-methylpiperidin-1-yl)azetidin-1-yl]methyl}quinolin-4-ol
3-[3-(4-ethylpiperazin-1-yl)propyl]-8-(1,3-thiazol-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one