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2-[3-(cyclopropylmethyl)-1-ethyl-1H-1,2,4-triazol-5-yl]-N,N-dimethylaniline
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2,4-dimethyl-1,3-oxazole-5-carboxamide
1-methyl-3-{2-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-2-oxoethyl}-3-(4-phenylphenyl)pyrrolidine-2,5-dione
2-{5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}acetic acid
1-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-hydroxypropan-1-one
2-(ethylamino)-4-methyl-N-[(2,3,4-trifluorophenyl)methyl]-1,3-thiazole-5-carboxamide
3-{5-[2-(1-methyl-1H-pyrrol-2-yl)-2-oxoacetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
3-{1-[1-(9H-purin-6-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-1-ol
1-(2-{1-[(4-fluorophenyl)methyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl}ethyl)-1H-1,2,3,4-tetrazole
2-(3-cyclopropanecarbonyl-1H-indol-1-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}acetamide
1-{1-[(2-fluorophenyl)methyl]-1H-pyrazol-4-yl}-3-[(1-methyl-1H-imidazol-2-yl)methyl]-3-propylurea
2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]benzamide
1-(3,5-difluorophenyl)-N-(1-ethylpiperidin-4-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-(1H-imidazol-1-yl)-1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]propan-1-one
4-chloro-3-({1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}carbonyl)-1H-pyrazol-5-amine
2-ethyl-9-(2-phenoxypropanoyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(4-methylphenyl)-1-(1,4-oxazepan-6-ylmethyl)urea
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
1-(6-methyl-2-phenylpyrimidin-4-yl)-N-[3-(1H-1,2,4-triazol-1-yl)propyl]piperidin-4-amine
1-methyl-4-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[2-(1,3-thiazol-4-yl)ethyl]-1H-1,2,3-benzotriazole-5-carboxamide
1-(cyclopropylmethyl)-4-[(3,5-dimethoxyphenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
2-(1,7-dimethyl-1H-indole-2-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,5,7-trimethylquinoline-4-carboxamide
N-({1-[5-(2,6-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-3-yl}methyl)acetamide
3-{6-hydroxy-4-[2-(1H-imidazol-1-yl)acetyl]-1,4-diazepan-1-yl}pyrazine-2-carbonitrile
4-[4-(4-fluorophenoxy)piperidin-1-yl]-4-oxobutane-1-sulfonamide
dimethyl(2-{2-[1-(oxane-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)amine
2-[(3R,4S)-3-[1-(1H-imidazol-1-ylmethyl)cyclopropaneamido]-4-propylpyrrolidin-1-yl]acetic acid
N-[(4-ethoxyphenyl)methyl]-4-methyl-5-[1-(thiophen-3-ylmethyl)-1H-pyrazol-3-yl]-1,3-thiazol-2-amine
2-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-1-(piperazin-1-yl)ethan-1-one
N-[(3S,4R)-1-(2,1,3-benzothiadiazol-5-ylmethyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
1-ethyl-4,6-dimethyl-2-oxo-N-(pyridin-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
N,N-dimethyl-5-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-(pyridin-3-yl)-N-{1-[2-(trifluoromethyl)phenyl]ethyl}pyrimidin-2-amine
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-[2-(3-fluorophenyl)ethyl]-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
N-[(4-chlorophenyl)methyl]-1-(2-ethoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
5-(1-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1H-1,2,3-triazol-4-yl)pyrimidine
methyl 3-{[1-(cyclopropylmethyl)-5-(3-methylpentanoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-2-(2-methoxyphenyl)acetamide
3-hydroxy-3-{[methyl(propan-2-yl)amino]methyl}-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
3-(1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-2-yl)pyridine
N-(2-fluorophenyl)-3-(2-methoxybenzoyl)piperidine-1-carboxamide
2-{6-[4-(1-cyano-1-methylethyl)phenyl]pyridin-3-yl}acetic acid
dimethyl({3-[2-(1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidin-4-yl)-1H-imidazol-1-yl]propyl})amine
N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)-5-(oxolan-2-yl)thiophene-2-carboxamide
N-{4-[4-({[2-(trifluoromethyl)phenyl]methyl}amino)piperidin-1-yl]phenyl}pyrazine-2-carboxamide
N-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
[1-(cyclopent-1-ene-1-carbonyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
3-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-1-(4-oxo-4H-chromen-6-yl)urea