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1-(2-hydroxyethyl)-4-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}-1,4-diazepan-6-ol
3-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-1-(5-tert-butyl-2-methoxyphenyl)urea
N-[3-(cyclopentyloxy)propyl]-2,6-dimethylpyridine-4-carboxamide
5-(1-{[4-(dimethylamino)phenyl]methyl}piperidin-4-yl)-5-[(2-fluorophenyl)methyl]imidazolidine-2,4-dione
1-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethan-1-one
(4aS,7aR)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-pentanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-methyl-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1-(pyridin-2-yl)-1H-pyrazole-4-carboxamide
(3R,4R)-3-cyclopropyl-1-(6-methoxypyrimidin-4-yl)-4-methylpyrrolidin-3-ol
3-hexyl-8-(1-methyl-1H-pyrazole-5-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
7-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[(3,4-dimethoxyphenyl)methyl]-1,3-benzoxazole-6-carboxamide
4-methyl-5-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,3-thiazol-2-amine
N-({3,5-dimethoxy-4-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-3,5-dimethyl-N-[(3S)-2-oxoazepan-3-yl]-1,2-oxazole-4-sulfonamide
3-(1-ethyl-1H-pyrazol-4-yl)-1-[3-(1H-imidazol-1-yl)propyl]-1-(pyridin-3-ylmethyl)urea
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-1-methyl-1H-pyrazole-4-sulfonamide
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]pyridine-3-sulfonamide
1,3-dimethyl-6-(pyridin-3-yl)-N-[2-(pyridin-4-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
6-[2-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-imidazol-1-yl]-2,3-dihydro-1,3-benzoxazol-2-one
2-(2-fluorophenyl)-N-{2-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}acetamide
6-fluoro-2-oxo-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-methoxy-N-(1-{7-[(5-methylfuran-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)propanamide
N-[2-(2-ethoxyphenyl)ethyl]-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
1-[4-(furan-2-yl)pyrimidin-2-yl]-N,5-dimethyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1H-pyrazole-4-carboxamide
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[(3-ethoxy-4-methoxyphenyl)methyl]acetamide
N-(3-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-3-oxopropyl)methanesulfonamide
(3S,4S)-1-(1-aminocyclobutanecarbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
1-(4-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}thiophen-2-yl)ethan-1-one
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-(2-methoxyethyl)-N-(pyridin-4-ylmethyl)acetamide
1-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}-4-methylpentane-1,2-dione
1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-[2-(4-chloro-3-methyl-1H-pyrazol-1-yl)acetyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-[3-(piperidin-3-yl)benzoyl]-4-(1H-pyrazol-1-ylmethyl)piperidine
1-ethyl-N,6-dimethyl-2-oxo-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,2-dihydropyridine-3-carboxamide
3-methyl-5-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)cinnoline
1-(carbamoylmethyl)-N-[(5-chloro-1-benzothiophen-3-yl)methyl]piperidine-4-carboxamide
4-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrole-2-carbonyl]-N-(2,2-difluoroethyl)benzene-1-sulfonamide
6-ethoxy-3-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-1,2-dihydroquinolin-2-one
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-2-(2,5-dioxoimidazolidin-4-yl)acetamide
3-(4-cyano-2-ethylphenyl)-1-[1-(pyrazin-2-yl)piperidin-3-yl]urea
1-(2,3-dihydro-1-benzothiophene-2-carbonyl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
5-methyl-1-{3-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]phenyl}-1H-1,2,3,4-tetrazole
{1-[(2-chloro-4,5-dimethoxyphenyl)methyl]-3-[(2,4-difluorophenyl)methyl]piperidin-3-yl}methanol
3-[8-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinoline-2-carbonyl]phenol
(4aS,8aR)-6-(isoquinolin-1-yl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N,1-dimethyl-1H-indole-2-carboxamide
2-tert-butyl-5-[3-(2-chlorophenyl)pyrrolidine-1-carbonyl]pyrimidin-4-ol
3-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-5-(propan-2-yl)-1,2-oxazole
2-phenoxy-N-(2-{7-[(2,4,5-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
[(2,3-difluorophenyl)methyl](2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)amine
2-[3-(dimethylamino)propyl]-9-[(4-methyl-1H-imidazol-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one