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2-[(2,6-dichlorophenyl)methyl]-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-4-hydroxypyrimidine-5-carboxamide
2-methyl-3-phenyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cycloprop-2-ene-1-carboxamide
1-(3-chlorobenzoyl)-N-[3-(furan-2-yl)phenyl]piperidine-4-carboxamide
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-1,4-diazepan-5-one
N-(3,5-dimethylphenyl)-6-(1-methylazepane-2-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[2-(2-fluorophenyl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl 2-chloro-5-({[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]carbamoyl}amino)benzoate
1-phenoxy-2-{4-[(3,4,5-trimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}propan-2-ol
{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}({[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl})methylamine
N-[2-(dimethylamino)ethyl]-2-(3-fluorophenyl)-N-(thiophen-3-ylmethyl)acetamide
(1R,5R)-6-(cyclobutylmethyl)-3-(5-methoxy-3-methyl-1H-indole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(1-methylpyrrolidin-3-yl)-9-(1,3-thiazol-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-[2-(dimethylamino)ethyl]-5-{1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-benzyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-methyl-1H-pyrazole-4-carboxamide
3-methyl-2-oxo-N-[2-(propylsulfanyl)phenyl]-1-oxa-3,8-diazaspiro[4.5]decane-8-carboxamide
(3R,5S)-5-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrrolidin-3-ol
3-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-ol
3-[({[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(thiophen-2-yl)pyrimidine-5-carboxamide
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-5-methyl-1,3-oxazole-4-carboxamide
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
methyl 1-[(3R,5S)-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}-1-cyclopentylpyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
3-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1-(4-methyl-2-oxo-2H-chromen-7-yl)urea
[4-({1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]pyrrolidin-3-yl}methyl)phenyl]methanol
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)thiophene-3-carboxamide
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
N-(1-hydroxybutan-2-yl)-5-[(methylsulfanyl)methyl]-N-(pyridin-2-ylmethyl)furan-2-carboxamide
N-[2-(2-chloro-6-fluorophenyl)ethyl]-1-ethyl-5-oxopyrrolidine-3-carboxamide
3-[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)propanamide
1-(2,1,3-benzothiadiazol-5-ylmethyl)-3-(3-benzyl-1H-1,2,4-triazol-5-yl)-1-methylurea
6-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]pyridine-2-carboxylic acid
N,4-dimethyl-5-[4-(2-methylphenoxy)piperidine-1-carbonyl]-1,3-thiazol-2-amine
3-{2-[2-(4-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-3-(2-methoxyphenyl)-1-(3-methoxypropyl)pyrrolidine-2,5-dione
3-{1-[1-(4-methoxypyrimidin-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-1-ol
ethyl 3-[(2-fluorophenyl)methyl]-1-[3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanoyl]piperidine-3-carboxylate
[2-(4-chlorophenyl)ethyl]({[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
2-(dimethylamino)-2-(2-fluorophenyl)-1-(4-hydroxy-4-phenylpiperidin-1-yl)ethan-1-one
1-{1-[4-(3-fluorophenyl)phenyl]piperidin-4-yl}piperidine-4-carbonitrile
N,2-dimethyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-1,6-naphthyridine-3-carboxamide
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2-(2-oxopiperidin-1-yl)acetamide
1-[4-(ethylamino)pyrimidin-2-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(furan-2-ylmethyl)({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)methylamine
4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-9-methoxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
7-cyclopentyl-2-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
4-[(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]benzonitrile
4-{5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}benzamide
(1-{1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methanamine