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N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-2-({6-[4-(pyridin-2-yl)piperazin-1-yl]pyridazin-3-yl}oxy)acetamide
N-[1-(cyclopropylmethyl)-1H-indazol-3-yl]-2-[4-(5-methylfuran-2-yl)-1H-pyrazol-1-yl]acetamide
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-(propan-2-yl)acetamide
3-chloro-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}pyridin-2-amine
1-cyclobutanecarbonyl-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]piperidine-4-carboxamide
1-[(5-methylthiophen-2-yl)methyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
5-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-{1-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-4-yl}pyrimidin-2-amine
ethyl 5-(1H-indol-3-ylmethyl)-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-methyl-4-[3-(1H-pyrazol-3-yl)phenyl]pyridine
2-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]acetamide
5-{3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-4-methyl-3-phenyl-1H-pyrazole
3-(3-fluorophenyl)-4-[4-(2-oxopyrrolidin-1-yl)butanoyl]piperazin-2-one
(2S,4S)-4-[(1-benzylpiperidin-4-yl)amino]-N-methyl-1-(propan-2-yl)pyrrolidine-2-carboxamide
(3aS,6aS)-2-methyl-5-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine
2-hydroxy-N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-phenylpyrrolidin-3-yl]acetamide
8-{[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}quinoline
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-methyl-N-[(4-methylphenyl)methyl]benzamide
2-[(8-methoxy-2H-chromen-3-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
2-chloro-5-[1-(2-phenoxyethyl)-1H-1,2,3-triazol-4-yl]pyridine
3-hexyl-8-(4-methylpiperidine-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-5-one
N-(3-ethoxypropyl)-1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-butyl-3-methyl-5-[3-(1H-1,2,4-triazol-1-yl)adamantan-1-yl]-1H-1,2,4-triazole
N-(4-tert-butyl-1,3-thiazol-2-yl)-2-{[1-(1-methyl-1H-pyrazol-5-yl)propyl]amino}acetamide
3-{5-methoxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-1-methyl-1,2-dihydroquinoxalin-2-one
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-methyl-N-(oxan-4-yl)acetamide
methyl 4-({[5-(2-fluorophenyl)-1,2,4-triazin-3-yl]amino}methyl)benzoate
4-(2-methylpropyl)-1-(thiophen-2-ylmethyl)-1,4-diazepan-5-one
7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(2,6-dimethylquinoline-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(3S,4S)-1-{2-methyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl}-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
5-[1-(cyclohexylmethyl)-4-hydroxypiperidin-4-yl]-N-(3,4-dimethoxyphenyl)-1-benzofuran-2-carboxamide
1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-3-(1H-imidazol-1-ylmethyl)piperidine
ethyl 1-(but-2-ynoyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
14-(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-[(5-fluoro-1H-indol-2-yl)methyl]-1-[4-(morpholine-4-carbonyl)phenyl]piperidin-4-amine
1-(4-benzylpiperazin-1-yl)-3-{1-[(2E)-2-methylbut-2-en-1-yl]piperidin-3-yl}propan-1-one
N-[1-(1H-1,2,3-triazole-5-carbonyl)piperidin-4-yl]pyridin-2-amine
1,3,6-trimethyl-5-(3-{1-[(5-methyl-1,2-oxazol-3-yl)methyl]-1H-pyrazol-3-yl}phenyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-cyclopropyl-2-(4-{[(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)carbamoyl]amino}phenyl)acetamide
3-[2-(4-methoxypiperidin-1-yl)-2-oxoethyl]-4-[(3-phenoxyphenyl)methyl]piperazin-2-one
2-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-1,3-benzoxazole
{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}[(3,4-dimethoxyphenyl)methyl]methylamine
ethyl 2-[3-(morpholin-4-yl)piperidin-1-yl]pyridine-3-carboxylate
5-methyl-1-(2-methylphenyl)-4-(2-phenylacetyl)piperazin-2-one
2-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]pyrido[2,3-d]pyrimidin-4-amine
2-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-3-methylquinoxaline
8-(2-methyl-1,3-thiazole-5-carbonyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(1-benzylpiperidin-4-yl)methyl]-2-[3-(3-fluorophenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide