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N-ethyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-(oxolan-2-ylmethyl)-1,3-oxazole-4-carboxamide
1-(1-ethylpiperidin-4-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(3-cyclopentylpropyl)piperidin-3-ol
7-chloro-4-hydroxy-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}quinoline-3-carboxamide
2-methyl-4-(5-{[4-(3-methylpyridin-2-yl)piperazin-1-yl]methyl}thiophen-2-yl)but-3-yn-2-ol
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]amine
(3aR,6aR)-2-acetyl-5-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(propan-2-yl)-5-(1H-pyrazol-3-yl)-1,3-benzoxazole
7-[3-(4-ethylphenyl)propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-(4-methyl-1H-pyrazol-1-yl)-1-[5-(3-methylbut-2-en-1-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]ethan-1-one
3-(2-methoxyethyl)-1-[8-(trifluoromethyl)quinolin-4-yl]piperidine-3-carboxylic acid
2-tert-butyl-5-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]pyrimidin-4-ol
9-[(3-methylphenyl)methyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[2-({5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)ethyl]-1,3-oxazolidin-2-one
3-{1-[1-(4-fluoro-2-methylphenyl)piperidin-4-yl]piperidin-3-yl}-1-(pyrrolidin-1-yl)propan-1-one
2-ethyl-4-{[4-(pyridin-3-yl)piperazin-1-yl]methyl}pyrimidine
4-[6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]thiomorpholine
3-(5-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
(2S)-3-{[(4-hydroxy-6-methylquinolin-2-yl)methyl]amino}propane-1,2-diol
N-(1-{1-[(4-hydroxy-3,5-dimethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
4-methyl-2-(2-oxo-2-{4-[2-(oxolan-2-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethyl)-1,2-dihydrophthalazin-1-one
4-{4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperazin-1-yl}-2-methyl-6-propylpyrimidine
2-[(4-chlorophenyl)methyl]-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,3-benzoxazole-5-carboxamide
2-(2-chlorophenyl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-[6-hydroxy-4-(1H-indol-7-ylmethyl)-1,4-diazepan-1-yl]pyridine-3-carbonitrile
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)cyclobutanecarboxamide
({4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-1,4-oxazepan-6-yl}methyl)dimethylamine
2-(4-{[2-(difluoromethoxy)phenyl]methyl}-1-[(4-methylphenyl)methyl]piperazin-2-yl)ethan-1-ol
3-(2-{6-methyl-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-oxoethyl)-2,3-dihydro-1H-isoindol-1-one
2-(hydroxymethyl)-N-[phenyl(pyridin-4-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]piperidine-2-carboxamide
2-{4-[(3-chloropyridin-4-yl)methyl]piperazin-1-yl}-N-(prop-2-en-1-yl)pyridine-3-carboxamide
N-methyl-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-4-propylpyrimidine-5-carboxamide
methyl (2S,4R)-1-[(2-ethoxyphenyl)methyl]-4-(4-methylbenzamido)pyrrolidine-2-carboxylate
N-[2-(4-phenylpyrimidin-2-yl)ethyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
6-{4-[(4-methoxy-2,5-dimethylphenyl)methyl]piperazin-1-yl}pyrimidine-2,4-diamine
2-oxo-N-{[5-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
N-cyclobutyl-3-[(5-oxo-1-propylpyrrolidin-3-yl)sulfamoyl]benzamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}benzamide
[(2S,6S)-4-[1-(2-methoxyethyl)piperidine-4-carbonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
2-(3-chlorophenoxy)-1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]ethan-1-one
1-(2,6-dimethylpyrimidine-4-carbonyl)-N-[3-(3-methylphenyl)phenyl]piperidine-3-carboxamide
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-[2-(trifluoromethyl)benzoyl]piperidine
2-(1H-imidazol-2-yl)-N-methyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}benzamide
1-({4-[2-(1H-pyrazol-1-ylmethyl)pyrrolidine-1-carbonyl]phenyl}methyl)piperidine
10-methoxy-N-(2-methyl-1,3-benzothiazol-5-yl)-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carboxamide
N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-1-(propan-2-yl)piperidine-4-carboxamide
1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3-(1H-imidazol-1-ylmethyl)piperidine
N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)naphthalene-1-carboxamide