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(1R,2S)-2-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-N-methylcyclohexane-1-carboxamide
1-cyclopropyl-N-(2-methylpropyl)-6-oxo-N-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxamide
N-[(3R,4R)-1-(3-chloropyridin-2-yl)-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
1-{[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]methyl}-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
3-(4-fluorophenoxymethyl)-1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)piperidine
(4aR,8aR)-4-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-octahydro-2H-1,4-benzoxazine
1-(2-fluorophenyl)-N-[(3-methylphenyl)methyl]-N-(propan-2-yl)cyclopropane-1-carboxamide
1-[5-(1H-imidazol-2-yl)imidazo[2,1-b][1,3]thiazole-6-carbonyl]-4-methyl-1,4-diazepane
N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-4-oxo-4H-chromene-2-carboxamide
methyl({[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
1-[5-(3-fluorophenyl)-1,2,4-triazin-3-yl]azepane
5-phenyl-1-(7-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)pentan-1-one
N-({3,5-dimethoxy-4-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-3,4-difluoro-N-[(3S)-2-oxoazepan-3-yl]benzene-1-sulfonamide
5-{[4-(3-ethylmorpholine-4-carbonyl)-1,3-oxazol-2-yl]methoxy}-2-methyl-1,3-benzothiazole
3-acetyl-N-{2-[2-(trifluoromethyl)phenyl]ethyl}-1H-pyrazole-5-carboxamide
2-methoxy-6-methyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}benzamide
(2-{2-[1-(4-fluoro-2-methylbenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
4-[(2-methyl-1,3-thiazol-4-yl)methyl]-N-[2-(1H-pyrazol-1-yl)phenyl]piperazine-1-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-6-oxo-1,6-dihydropyridine-3-carboxamide
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
2-{1-[(4-methylphenyl)methyl]-4-(quinoxalin-5-ylmethyl)piperazin-2-yl}ethan-1-ol
1-({1-[2-(1H-imidazol-5-yl)ethyl]-3-(phenoxymethyl)-1H-1,2,4-triazol-5-yl}methyl)pyrrolidin-2-one
2-benzyl-9-[2-(4-fluorophenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1-(4,6,7-trimethylquinazolin-2-yl)piperidin-4-amine
5-{[4-(methylsulfanyl)phenyl]methyl}-2-(3,4,5-trimethoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepin-4-one
2-{[8-(3-methoxypropyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]methyl}benzonitrile
N-(isoquinolin-5-ylmethyl)-N,1-dimethylazepane-2-carboxamide
(3aS,6aS)-5-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(2-methoxyethyl)-N-methyl-N-[(3-methylthiophen-2-yl)methyl]-6-oxopiperidine-3-carboxamide
3-(1,2-oxazolidin-2-yl)-1-[3-(4-phenylbenzoyl)piperidin-1-yl]propan-1-one
(3aR,6aR)-2-(3-acetylbenzoyl)-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(2-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}-2-oxoethyl)-1,2-dihydrophthalazin-1-one
2-(1H-imidazol-1-yl)-1-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]ethan-1-one
5-(3-fluorophenyl)-3-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]-1,2,4-triazine
2-{1-methyl-4-[(3-methyl-1H-indol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
4-(4-methylphenoxy)-1-[(2R)-oxolane-2-carbonyl]piperidine
7-methyl-2-[(2E)-3-(1-methyl-1H-pyrazol-4-yl)prop-2-enoyl]-2,7-diazaspiro[4.5]decan-6-one
(2-ethoxy-5-{1-[2-(pyrazin-2-yl)ethyl]-1H-imidazol-2-yl}phenyl)methanol
1-(2-chloroprop-2-en-1-yl)-3-{[(2,2-dimethyloxan-4-yl)amino]methyl}-6,7-dimethoxy-1,2-dihydroquinolin-2-one
(2-{2-[1-(3,5-difluoropyridine-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
2-{[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-4-yl]oxy}-N-tert-butyl-5-chlorobenzamide
N-[2-methoxy-5-({[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]carbamoyl}amino)phenyl]propanamide
3-(1-methyl-1H-1,2,4-triazol-3-yl)-1-{2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl}urea
N,N-diethyl-2-{[4-(1H-indole-5-carbonyl)-2-oxo-1-(2-phenylethyl)-1,4-diazepan-6-yl]oxy}acetamide
N-[(3R,4R)-1-cyclohexyl-3-hydroxypiperidin-4-yl]pyridine-4-carboxamide
1-[4-(4-{[methyl(quinolin-6-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]-2-phenylethan-1-one
3-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-1-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}urea
2-(2-aminopyrimidin-5-yl)-N-ethyl-8-methyl-N-(pyridin-2-ylmethyl)quinoline-4-carboxamide
2-ethyl-4-methyl-N-[2-(pyrrolidin-1-yl)ethyl]-1,3-oxazole-5-carboxamide
7-fluoro-2-methyl-4-[1-(pyridin-4-ylmethyl)-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]quinoline