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2-[5-({2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)-1,2-oxazol-3-yl]pyridine
3,5-dimethyl-4-({3-[3-(1,3-thiazol-2-yl)phenyl]-1H-pyrazol-1-yl}methyl)-1,2-oxazole
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-2-propyl-1,3-thiazole-4-carboxamide
4-[4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carbonyl]-1λ6-thiomorpholine-1,1-dione
5-(5-chloro-2-methylphenoxy)-1-azabicyclo[3.2.1]octane
2-[(3,4-dihydro-2H-1-benzopyran-3-ylformamido)methyl]-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-(1-{7-[(4-chlorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
7-[2-(2-cyclopropyl-1H-1,3-benzodiazol-1-yl)acetyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
4-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
(2S,4R)-4-amino-N,N-diethyl-1-(2-methoxyacetyl)pyrrolidine-2-carboxamide
2-(adamantan-1-yl)-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]acetamide
2-(2-{[(1R,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenoxy)acetic acid
2-cyclopentyl-8-(5-oxo-2,5-dihydro-1H-pyrazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
4-[1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperazine-1-sulfonamide
3-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}pyridin-2-amine
4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1λ6-thiane-1,1-dione
2-{[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl](methyl)amino}-N,N-dimethylacetamide
4-benzyl-1-(2,3-difluoro-4-methylbenzoyl)-3-ethyl-1,4-diazepan-5-one
2-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]pyrimidine
4-{4-[2-(pyrrolidine-1-carbonyl)piperazine-1-carbonyl]phenyl}phenol
1'-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-{2-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindol-1-one
N-[2-(dimethylamino)ethyl]-5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
5-chloro-N-(2-methylpropyl)-6-oxo-N-(3-phenylprop-2-yn-1-yl)-1,6-dihydropyridine-3-carboxamide
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-sulfonyl}-2,1,3-benzothiadiazole
(2S,4R)-4-amino-N,N-diethyl-1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)pyrrolidine-2-carboxamide
1-(cyclohexylmethyl)-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N-methyl-6-oxopiperidine-3-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N'-(2-methylphenyl)propanediamide
1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(3-methylpyridin-2-yl)piperazine
2,5-dimethyl-N-[1-(2-phenylethyl)piperidin-3-yl]furan-3-carboxamide
1-{2-[(2,3-dimethoxyphenyl)formamido]ethyl}-N-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
3-{2-oxo-2-[2-(pyridin-2-yl)piperidin-1-yl]ethyl}-3-phenyl-1-(thiophen-2-ylmethyl)pyrrolidine-2,5-dione
N-({3-[(2-fluorophenyl)methoxy]-4-methoxyphenyl}methyl)-N-(pyridin-4-ylmethyl)acetamide
N-(3-fluorophenyl)-3-[methyl(2-phenylethyl)amino]piperidine-1-carboxamide
N-[(1-phenylcyclopentyl)methyl]-6-[(2E)-3-phenylprop-2-enoyl]-6-azaspiro[2.5]octane-1-carboxamide
4-methoxy-N-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
(1S,5R)-3-cyclobutanecarbonyl-6-(dimethyl-1,3-thiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
6-methyl-5-[5-(2-methyl-1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
6,6-dimethyl-1-(2-methylphenyl)-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
2-(2-methoxyethyl)-8-(5-phenyl-1,2,4-oxadiazol-3-yl)-2,8-diazaspiro[5.5]undecan-3-one
1-[(4-fluorophenyl)methyl]-4-(pyridin-2-ylmethyl)-1,4-diazepane
3-(4-methyl-1,3-thiazol-5-yl)-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}propanamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-[2-(1H-pyrrol-1-yl)ethyl]acetamide
3-[6-amino-5-cyano-4-(6-methoxy-2,3-dihydro-1H-inden-5-yl)pyridin-2-yl]-1H-pyrazole-5-carboxylic acid
3-{5-[(4-methoxy-2,3-dimethylphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}pyridine
9-(3-amino-3-phenylpropanoyl)-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 4-(1-{[4-(methylsulfanyl)phenyl]carbamoyl}-6-azaspiro[2.5]octan-6-yl)-4-oxobutanoate
N-(3-chloro-4-methoxyphenyl)-6-[(3-ethoxy-4-methoxyphenyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
4-(1-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)morpholine