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2-methyl-2-(methylamino)-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)propanamide
3-ethyl-3-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1-[3-(1H-pyrazol-5-yl)phenyl]urea
2-methyl-6-[3-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2,3-dihydropyridazin-3-one
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-1-(3-hydroxyazetidin-1-yl)propan-1-one
5-{[4-(2-fluorophenoxy)piperidin-1-yl]methyl}-2-(pyridin-2-yl)pyrimidine
2-{1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]azetidin-3-yl}pyridine
4-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridin-6-yl]-2-methyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
cyclohexyl({4-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl})methanol
3-[(2-ethoxyphenyl)methyl]-9-methoxy-N-[(2-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-(2-methanesulfonamidoethyl)-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
2-{4-phenyl-5-[4-(trifluoromethyl)phenyl]-1H-imidazol-1-yl}ethan-1-ol
(4aS,8aS)-2-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-decahydroisoquinolin-4a-ol
5-(oxan-2-yl)-3-(thiophen-2-ylmethyl)-1,2,4-oxadiazole
(1s,4s)-N1-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}cyclohexane-1,4-diamine
N5-(2,2-dimethyloxan-4-yl)-N6-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
5-benzyl-N-(oxolan-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
4-[2-(3,4-dichlorophenyl)morpholin-4-yl]-6-methoxypyrimidin-2-amine
2-(morpholin-4-yl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]benzamide
2-{3-cyclopentyl-5-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[(1-methyl-5-oxopyrrolidin-2-yl)methyl]-1H-pyrazole-3-carboxamide
9-(4-ethylbenzoyl)-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopentyl-2-{4-[2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]morpholin-3-yl}acetamide
5-fluoro-2-{1-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
methyl 4-{3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}-4-oxobutanoate
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-[(2,6-difluorophenyl)methyl]-1H-pyrazole-4-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-N-methylthian-4-amine
(3R,4R)-4-amino-1-(3,5-dichloropyridin-2-yl)piperidin-3-ol
4-({4-methyl-5-[1-(3-phenylpropyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
3-[(3R,4S)-4-(dimethylamino)-1-[4-(2-methylphenyl)benzoyl]piperidin-3-yl]propan-1-ol
1-(carbamoylmethyl)-N-{[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]methyl}piperidine-4-carboxamide
[(2E)-3-(furan-2-yl)prop-2-en-1-yl](2-methylpropyl)(pyridin-2-ylmethyl)amine
1-[(4,5-dimethylfuran-2-yl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3,6-diazabicyclo[3.2.2]nonane
1-[5-(2,4-difluorophenoxymethyl)-1H-pyrazole-3-carbonyl]-3-(methoxymethyl)piperidine
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-methyl-1,2,3-thiadiazole-5-carboxamide
1-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)acetamide
1-(cyclopropylmethyl)-5-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-({[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}(thiophen-2-ylmethyl)amino)butan-1-ol
N-(1H-imidazol-2-ylmethyl)-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
2-(1H-indol-3-yl)-1-(3-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-1-yl)ethan-1-one
N-cyclopropyl-2,3-dimethyl-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)-1H-indole-7-carboxamide
2-(2-methoxy-5-{[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}phenoxy)acetic acid
3-benzyl-5-[4-methoxy-3-(methoxymethyl)phenyl]-1H-1,2,4-triazole
5-chloro-2-[3-(2-phenylethyl)-1,2-oxazole-5-carbonyl]-1,2,3,4-tetrahydroisoquinoline
1-methyl-4-[6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]-1,4-diazepane
2-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-N-(pyridin-2-ylmethyl)acetamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-1-methyl-1H-pyrrole-2-carboxamide
1-[(2,3-dichloro-6-fluorophenyl)methyl]-5-methylpyrrolidin-2-one
1-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}-4-(thiophene-2-carbonyl)piperazine