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3-[(7R,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(5-acetyl-2-ethoxyphenyl)urea
methyl 4-[5-({methyl[2-(oxan-2-yl)ethyl]amino}methyl)-1,2,4-oxadiazol-3-yl]benzoate
3-methoxy-1-[3-(2-methoxyphenoxy)azetidin-1-yl]propan-1-one
3,5-dimethyl-N-[(5-oxopyrrolidin-2-yl)methyl]-N-(propan-2-yl)-1-benzofuran-2-carboxamide
2-(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)acetic acid
1-(azocan-1-yl)-3-[2-methoxy-5-({[3-(1H-pyrazol-1-yl)propyl]amino}methyl)phenoxy]propan-2-ol
5-(2,6-difluorophenoxymethyl)-N-(oxan-4-ylmethyl)-1,2-oxazole-3-carboxamide
(1S,5R)-6-[3-(2-fluorophenyl)-1H-pyrazole-4-carbonyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane
3-(4-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}piperazin-1-yl)-1,2-dihydropyrazin-2-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methylpiperidin-3-amine
(2S,4S,5R)-4-[(2-methoxyethyl)carbamoyl]-1-methyl-2-(2-methylpropyl)-5-(pyridin-3-yl)pyrrolidine-2-carboxylic acid
4-[1-(3-chlorophenyl)-1H-pyrazol-4-yl]-N-(pyridin-4-ylmethyl)pyrimidin-2-amine
4-[1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]morpholine
N-(7-chloro-2-ethyl-3-methyl-1-benzofuran-5-yl)-4-(4H-1,2,4-triazol-4-yl)piperidine-1-carboxamide
6-[3-(1H-pyrazol-1-yl)benzoyl]-N-(thiophen-2-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
N-(2-phenylethyl)-3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl](ethyl){[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amine
2-{5-[6-(piperidine-1-carbonyl)pyrazin-2-yl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
{4-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-1,4-oxazepan-6-yl}methanol
1-(4-methoxyphenyl)-4-{1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidin-3-yl}piperazine
(3R,4S)-4-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl](methyl)amino}oxolan-3-ol
2-(pyridin-3-ylmethyl)-9-[(2,3,4-trifluorophenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
cyclopentyl 4-({[2-(1-methyl-1H-pyrazol-5-yl)ethyl]carbamoyl}amino)benzoate
6-{[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
methyl 4-(5-{[4-(oxolane-2-carbonyl)piperazin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
N-{[2-(4-methoxy-2-methylphenyl)phenyl]methyl}propanamide
1-{2-oxo-2-[3-(phenylamino)piperidin-1-yl]ethyl}pyrrolidin-2-one
4-{3-[({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)amino]butyl}phenol
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[4-(5-methylpyrimidin-4-yl)piperidin-1-yl]ethan-1-one
2-hydroxy-1-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
N,N-dimethyl-6-[3-(piperidin-1-ylmethyl)piperidin-1-yl]pyrimidin-4-amine
5-[1-(5-aminopyrazin-2-yl)-1H-imidazol-2-yl]thiophene-2-carboxylic acid
8-[(1S,3R)-3-aminocyclopentanecarbonyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[3-(2H-1,3-benzodioxol-5-yl)-4-methoxyphenyl]ethan-1-amine
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-3-propyl-1H-pyrazole-5-carboxamide
1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-3-amine
(2S)-3-phenyl-2-({2-[(prop-2-en-1-yl)amino]phenyl}formamido)propanamide
N'-(3,5-dimethylphenyl)-N-[(1R,2S)-2-phenylcyclopropyl]propanediamide
9-(dimethyl-1,2-oxazole-4-carbonyl)-1-methyl-4-(oxolan-3-ylmethyl)-1,4,9-triazaspiro[5.5]undecane
(3S,4R)-1-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-N,N-dimethyl-4-propylpyrrolidin-3-amine
1-(7-{[4-(benzyloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[3-(methylsulfanyl)propyl]piperidine
N-(3,3-diphenylpropyl)-6-[(6-methylpyridin-2-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
2,8-dimethyl-4-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}quinoline
4-[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]thiomorpholine
(2S,4S)-1-[(2-chlorophenyl)methyl]-4-[(pentan-3-yl)amino]-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-(1-methyl-1H-pyrazole-5-carbonyl)piperidine
5-({5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-phenyl-1H-imidazol-1-yl}methyl)-3-ethyl-4,5-dihydro-1,2-oxazole
4-{4-[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]piperidin-1-yl}pyrimidine