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1-(6-{6-[(pyridin-4-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-3-yl)ethan-1-one
methyl (2R,4S)-1-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]acetyl}-4-hydroxypiperidine-2-carboxylate
7-methyl-3-[5-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]quinolin-2-ol
3-benzyl-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-1,2-oxazole-5-carboxamide
1-(2-hydroxyethyl)-4-[4-(methoxymethyl)benzoyl]-1,4-diazepan-6-ol
9-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{3-[cyclopentyl(methyl)amino]propyl}-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
6-methoxy-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)hexanamide
N,1,3-trimethyl-6-(pyridin-2-yl)-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}-N-methylcyclohexanamine
N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)-2-(4-propanoylphenoxy)acetamide
N-[(cyclopropylcarbamoyl)methyl]-2-(dimethylamino)-2-(2-fluorophenyl)acetamide
3-[4-(4-fluorophenyl)-1,4-diazepane-1-carbonyl]piperidine-1-carboxamide
methyl 4-[5-methyl-4-({methyl[1-(4-methyl-1,3-thiazol-2-yl)ethyl]amino}methyl)-1,3-oxazol-2-yl]benzoate
1-(cyclopropylmethyl)-5-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-(1-propyl-1H-pyrazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(5-methoxypyrimidin-2-yl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
N-(1-hydroxybutan-2-yl)-N-(thiophen-3-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
3-(2-chlorophenyl)-1-[2-(dimethylamino)ethyl]-3-[2-(2-methyl-4-phenylpiperazin-1-yl)-2-oxoethyl]pyrrolidine-2,5-dione
3-(1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carbonyl}piperidin-3-yl)benzoic acid
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-(2-ethoxyethyl)-1,2-oxazole-3-carboxamide
1-benzyl-5-{[(4-chlorophenyl)methyl]amino}-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-2-(3-fluorophenyl)-N-(pyridin-3-ylmethyl)acetamide
9-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
N-(1-ethyl-1H-indazol-3-yl)-2-(2-methyl-1H-imidazol-1-yl)acetamide
(1R,7S)-N-(2-hydroxyethyl)-N-methyl-3-[(5-methylpyrazin-2-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
6-[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]-5-chloropyridine-3-carboxylic acid
(1-{1-[(6-chloro-2-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methanamine
2-methoxy-3-[3-(1H-pyrazol-3-yl)phenyl]pyrazine
3-[1-(propan-2-yl)-5-[(propan-2-yl)sulfamoyl]-1H-1,3-benzodiazol-2-yl]propanamide
N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
3-{1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]piperidin-3-yl}-N-[(3-methoxyphenyl)methyl]propanamide
5-(3-methoxyphenyl)-2-(pyridin-4-yl)-4-[1-(thiophen-3-ylmethyl)piperidin-4-yl]pyrimidine
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(4,6-dimethylpyrimidin-2-yl)ethyl]amine
3-[(1R,5S)-6-azabicyclo[3.2.1]octane-6-carbonyl]-N-[(3-methyloxetan-3-yl)methyl]benzene-1-sulfonamide
1-[5-(hydroxymethyl)furan-2-carbonyl]-4-(3-methylbut-2-en-1-yl)-1,4-diazepan-6-ol
1-[2-methoxy-4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)urea
3-{3-[methyl(2-methylpropyl)amino]propyl}-8-[(2-methyl-1,3-oxazol-4-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{4-[(5-cyclopentylthiophen-2-yl)methyl]-1-(1-methylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
4-[4-(quinolin-2-ylmethyl)piperazin-1-yl]quinazoline
N-[1-(cyclohex-1-en-1-yl)ethyl]-2-(1H-1,2,3,4-tetrazol-5-yl)acetamide
4-{2,6-dioxo-1H,2H,5H,6H,7H,8H-[1,3]oxazolo[4,5-g]quinolin-8-yl}-N-methylbenzene-1-sulfonamide
2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[(4-methyl-1H-imidazol-2-yl)methyl]benzamide
8-({7-chloro-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-[2-(quinolin-8-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]phenol
4-{[2-(3-fluorophenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}-2,6-dimethoxyphenol
1-methyl-4-[(1-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methyl]piperazine
N-({1-[2-(phenylsulfanyl)acetyl]piperidin-3-yl}methyl)furan-2-carboxamide
1-[5-(azepan-1-ylmethyl)-2-methoxyphenoxy]-3-(diethylamino)propan-2-ol
1-(3-{[3-(dimethylamino)propyl](methyl)amino}piperidin-1-yl)-2-(2,3-dimethylphenoxy)ethan-1-one