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3-{[cyclohexyl(methyl)amino]methyl}-1-[(2,3-difluorophenyl)methyl]-3-hydroxypiperidin-2-one
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]quinoline-5-carboxamide
1-{1-[2-(thiophen-2-yl)pyrimidine-5-carbonyl]piperidin-4-yl}piperidin-3-ol
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2,5-dimethyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
5,7-dimethyl-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}pyrazolo[1,5-a]pyrimidine-2-carboxamide
ethyl 4-({4-[3-oxo-3-(pyrrolidin-1-yl)propyl]piperidin-1-yl}methyl)-1H-pyrazole-3-carboxylate
5-(2-chlorophenyl)-N-[1-(4-propyl-4H-1,2,4-triazol-3-yl)ethyl]furan-2-carboxamide
13-benzyl-4,6-dimethyl-3,7,8,10-tetraazatricyclo[7.4.0.02,7]trideca-1,3,5,8-tetraen-11-one
{1-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
N-methyl-N-(1-{1-[2-(morpholin-4-yl)propanoyl]piperidin-4-yl}-2-phenylethyl)thiophene-3-carboxamide
4-cyano-N-[(3R,4S)-4-(propan-2-yl)-1-(pyridin-4-yl)pyrrolidin-3-yl]oxane-4-carboxamide
1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
N-methyl-2-(3-methyl-2-oxo-1,2-dihydroquinoxalin-1-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)acetamide
2-methyl-6-(piperidin-4-yl)-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]pyrimidin-4-amine
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
ethyl 3-[(2-fluorophenyl)methyl]-1-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}piperidine-3-carboxylate
5-({4-[(2-methylphenyl)methyl]piperazin-1-yl}methyl)-2,1,3-benzoxadiazole
(1S,5R)-3-benzyl-6-(2,3-difluoro-6-methoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonane
(2E)-3-(4-methoxyphenyl)-N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)prop-2-enamide
8-benzyl-1-ethyl-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(1-benzothiophen-5-ylmethyl)-1-cycloheptyl-6-oxopiperidine-3-carboxamide
N-cyclohexyl-4-{[2-(dimethylamino)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-[3-(dimethylamino)propyl]-N-methyl-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
2-{[2-(furan-2-yl)azepan-1-yl]methyl}benzonitrile
7-cyclohexyl-2-(oxane-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-tert-butyl-6-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]-1,2-dihydropyrimidin-2-one
1-[2-({[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-(thiophen-2-ylmethyl)piperidine-4-carboxylic acid
N-ethyl-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-(pyridin-4-ylmethyl)propanamide
2-methyl-8-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-2-methoxy-N-methylpyridine-3-carboxamide
2-(3,4-dimethylphenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
1-[1-(5-methyl-1,3-oxazole-4-carbonyl)piperidin-3-yl]-3-phenylpropan-1-one
4-[(2-methylphenyl)methyl]-3-[2-(morpholin-4-yl)-2-oxoethyl]piperazin-2-one
2-methyl-6-({5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-4H-pyran-4-one
methyl 2-{N-methyl-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamido}acetate
3-(2H-1,3-benzodioxole-5-carbonyl)-1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperidine
3-methyl-8-{[3-(trifluoromethyl)phenyl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[(cycloheptylamino)methyl]-2-methoxy-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-(1-benzylpyrrolidin-3-yl)-3-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]propanamide
3-[3-({[cyclopropyl(3-methylpyridin-2-yl)methyl]carbamoyl}amino)phenyl]-N,N-dimethylpropanamide
1'-(1-acetylpiperidine-3-carbonyl)-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
3-propyl-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazole-5-carboxamide
1-(furan-2-carbonyl)-4-(3-phenylbutyl)-1,4-diazepane
2-(4-{5-[(phenylsulfanyl)methyl]furan-2-carbonyl}morpholin-3-yl)acetamide
(1S,5R)-6-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane
3-methyl-8-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl 4-[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxylate
6-(2-{[3-(trifluoromethyl)phenyl]methyl}morpholine-4-carbonyl)pyridin-3-ol