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1-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(morpholin-4-yl)-N-propyl-1H-1,3-benzodiazole-5-carboxamide
N-[2-(1H-indol-1-yl)ethyl]-3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}propanamide
4-{1-[ethyl(methyl)sulfamoyl]piperidin-3-yl}benzoic acid
N-[1-(pyrazin-2-yl)propan-2-yl]-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
2-{2-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-5,6-dimethyl-2,3-dihydropyridazin-3-one
1-[(4-ethyl-1,3-thiazol-2-yl)methyl]-4-(1,3-thiazol-2-yl)-1H-1,2,3-triazole
(3aS,6aS)-2-acetyl-5-[(4-fluorophenyl)methanesulfonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
8-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-2-butyl-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(1,3-benzoxazol-2-ylsulfanyl)ethyl]-5-(1H-pyrazol-1-ylmethyl)furan-2-carboxamide
N-{[8-(cyclohexylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
[(5-chloro-2,3-dimethoxyphenyl)methyl](methyl)(1,2-oxazol-3-ylmethyl)amine
1-(2-methylphenyl)-4-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]-1,4-diazepane
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(2-phenylethyl)piperazine
N-(2-{[6-(aminomethyl)-2-methylpyrimidin-4-yl]amino}ethyl)acetamide
methyl 3-benzamido-5-{[(2,3-dimethoxyphenyl)methyl]amino}-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}amine
1-[(2,5-dimethylphenyl)methyl]-3-(1,3,4-thiadiazol-2-yl)urea
2-ethyl-4-phenyl-9-(pyridine-2-carbonyl)-2,9-diazaspiro[5.5]undecane
1-{2-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-2-oxoethyl}-2-methyl-1,4-dihydroquinolin-4-one
2-[4-(cyclopropylmethyl)piperazin-1-yl]-2-(2,6-dimethylphenyl)acetic acid
1-benzyl-N-{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-amine
1-[3-(2-fluorophenoxy)azetidin-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
4-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]-7,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline
3-[(2-ethoxyphenyl)methyl]-N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-phenyl-4-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperazin-2-one
4-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-methyl-1-(2-methylpropyl)piperazin-2-one
3-[(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
4-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}morpholine
1-[ethyl({2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl})amino]-3-phenoxypropan-2-ol
2,5-dimethyl-N-[(5-methylpyrazin-2-yl)methyl]-1-phenyl-1H-pyrrole-3-carboxamide
2-{2-[4-(1-tert-butyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]ethyl}-6-fluoro-1H-1,3-benzodiazole
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-3H,3aH,4H,5H,9bH-cyclopenta[c]quinoline-4-carboxamide
4-{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}morpholine
(3R,4R)-4-cyclobutyl-3-methyl-1-(1,3-thiazol-2-ylmethyl)piperidin-4-ol
1-(4-benzylpiperidin-1-yl)-3-[1-(2-methoxyacetyl)piperidin-4-yl]propan-1-one
2-{5-[(2-methyl-1,3-thiazol-4-yl)methyl]-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-3-yl}pyridine
(3R,5S)-5-(3-fluorophenoxymethyl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-N-[3-(morpholin-4-yl)propyl]piperidine-3-carboxamide
2-methyl-4-{4-[3-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]phenyl}butan-2-ol
1-{1-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-3-yl}-2-phenylethan-1-one
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]({[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl})methylamine
6-(2,4-dimethoxyphenyl)-1,3-benzothiazol-2-amine
(1R,5R)-6-[(6-methylpyridin-2-yl)methyl]-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-cyclobutaneamido-N-(2-hydroxy-2-phenylethyl)benzamide
(4aR,7aS)-1-benzyl-4-(1H-imidazol-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{1-[2-methyl-2-(piperidin-1-yl)propyl]azetidin-3-yl}-1H-1,3-benzodiazole
3-chloro-4-fluoro-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1-benzothiophene-2-carboxamide
8-fluoro-2-{[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]methyl}quinolin-4-ol
5-{2-[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
N-(1-ethyl-1H-pyrazol-5-yl)-2-{4-[4-(1H-imidazol-1-ylmethyl)phenyl]-1H-pyrazol-1-yl}acetamide