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(2,1,3-benzothiadiazol-5-ylmethyl)({5-[(2E)-but-2-en-1-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methylamine
3-{2-[4-hydroxy-4-(pyridin-2-yl)piperidin-1-yl]-2-oxoethyl}-4-[(5-methylfuran-2-yl)methyl]piperazin-2-one
2-(morpholin-2-yl)-1-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]ethan-1-one
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[2-(7-methyl-1H-1,3-benzodiazol-2-yl)ethyl]acetamide
1-(5-ethyl-1,3,4-oxadiazol-2-yl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
3-(1,2-oxazinan-2-yl)-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]propanamide
5-ethyl-N4-{3-[(5-methylpyridin-2-yl)amino]propyl}pyrimidine-2,4-diamine
7-(3-chlorophenyl)-4-(prop-2-en-1-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
[2-(6-methoxypyridazin-3-yl)phenyl]methanol
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-4-phenylbutane-1,2-dione
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(5-oxopyrrolidin-2-yl)acetamide
2-({3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-1H-indole
2-(3-methoxyphenyl)-N-[2-(methylsulfanyl)phenyl]pyrrolidine-1-carboxamide
1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-3-hydroxypropan-1-one
1-{[2-(2-methoxyethyl)pyrimidin-5-yl]methyl}-N-[3-(3-methylphenyl)phenyl]piperidine-3-carboxamide
5-(4-{[4-(1H-imidazol-1-yl)phenyl]methyl}piperazin-1-yl)-2-methyl-2,3-dihydropyridazin-3-one
N-(3-methylphenyl)-3-[1-(6-oxo-1,6-dihydropyridine-2-carbonyl)piperidin-4-yl]propanamide
methyl 5-cyano-2-methyl-6-[methyl({[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl})amino]pyridine-3-carboxylate
3-methyl-1-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}butan-1-one
(3aR,6aR)-2-ethyl-5-[4-methyl-6-(methylamino)pyrimidin-2-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[4-methyl-6-(methylamino)pyrimidin-2-yl]pyrrolidin-3-yl]acetamide
2-[4-(2H-1,3-benzodioxol-5-yl)-2-[(3-methylpiperidin-1-yl)methyl]phenoxy]-N-(1,3-thiazol-2-ylmethyl)acetamide
1-[1-(2-chloro-6-fluorobenzoyl)piperidin-4-yl]-N-cyclopropylpiperidine-4-carboxamide
(4aR,8aR)-2-cyclopentanecarbonyl-7-[(4-methyl-1H-imidazol-2-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-2-phenoxyacetamide
N-(1,3-dihydroxypropan-2-yl)-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]acetamide
N-(dicyclopropylmethyl)-2-(2-methoxyethyl)-N-methyl-1,3-dioxo-2,3-dihydro-1H-isoindole-5-carboxamide
methyl 4-[(3-{2-[(4-fluorophenyl)formamido]ethyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl)methyl]benzoate
N-methyl-5-({4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}methyl)-1,2,4-oxadiazole-3-carboxamide
5-(piperidin-1-yl)-2-(3,3,3-trifluoro-2-hydroxypropyl)-2,3-dihydropyridazin-3-one
N-[1-(2,4-dimethoxyphenyl)ethyl]-N-methyl-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
1-(4-fluorophenyl)-3-{2-[4-(propan-2-yl)morpholin-2-yl]ethyl}urea
3-methoxy-1-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
4-[3-(1H-1,3-benzodiazol-2-yl)azetidine-1-carbonyl]benzene-1-sulfonamide
3-({4-[3-(pyrrolidin-1-yl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
2-(2-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl)pyridine
3-(azocan-1-yl)-N-{1-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}propanamide
4-[(2-methyl-1H-imidazol-4-yl)methyl]-2-(piperidin-1-ylmethyl)-1,4-oxazepane
1-(1-benzothiophen-2-ylmethyl)-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
6-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-2,3-dimethylquinoxaline
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
5-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-2,3-dihydro-1H-pyrazol-3-one
[2-(1-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}piperidin-2-yl)ethyl]dimethylamine
5-[2-(furan-2-yl)pyrrolidine-1-carbonyl]-2-(propan-2-yl)pyrimidine
3-[5-(5-acetylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]propanamide
4-hydroxy-N-[(3-propyl-1,2-oxazol-5-yl)methyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
3-{2-[4-(2-hydroxyphenyl)piperazin-1-yl]-2-oxoethyl}-4-[(4-methylphenyl)methyl]piperazin-2-one
1-[(1-propyl-1H-pyrazol-4-yl)methyl]-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
3,3-dimethyl-1-[(3S,4R)-1-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}-4-(propan-2-yl)pyrrolidin-3-yl]urea
9-[(3-hydroxyphenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one