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3-{[(2,2-difluoroethyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-(pyrimidin-2-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-3-amine
methyl 4-[2-(4-methylpentyl)morpholin-4-yl]-4-oxobutanoate
N-{3-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-3-oxopropyl}methanesulfonamide
1-[(4-chlorophenyl)methyl]-4-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]piperazine
3-[1-(2-acetylbenzoyl)piperidin-4-yl]-1-(4-ethylpiperazin-1-yl)propan-1-one
N-[(3,4-dimethylphenyl)(pyridin-3-yl)methyl]-1H-imidazole-2-carboxamide
2-[4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-(3-methylbutyl)piperazin-2-yl]ethan-1-ol
3-[1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-3-yl]propanamide
{2-oxo-2-[6-oxo-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]ethyl}urea
7-(5-methylthiophen-2-yl)-4-(oxane-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{2-fluoro-5-[({[1-(phenoxymethyl)cyclopropyl]methyl}carbamoyl)amino]phenyl}acetamide
methyl 2-{[(4-chlorophenyl)methyl]sulfamoyl}-6-(2,2-dimethylpropanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl})methylamine
(3aR,6aR)-2-cyclopentyl-5-[2-(3-methoxyphenoxy)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-benzyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1,3-thiazole-4-carboxamide
(1S,4S)-2-[2-(2-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-2-azabicyclo[2.2.1]heptane
2-{[4-(1-methoxypropan-2-yl)piperidin-1-yl]methyl}benzonitrile
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1-(9H-purin-6-yl)piperidin-4-amine
2-[2-(thiophen-2-yl)ethyl]-1-(1H-1,2,3-triazole-5-carbonyl)piperidine
3-{4-[(3-methoxyphenyl)methyl]piperazine-1-carbonyl}-1-phenylpyrrolidin-2-one
2-{[(2-chlorophenyl)methyl]sulfanyl}-1-(6-hydroxy-1,4-oxazepan-4-yl)ethan-1-one
N,N,3-trimethyl-4-[({2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}carbamoyl)amino]benzamide
4-(4-benzyl-1H-pyrazol-5-yl)-1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]piperidine
2-(1,4-dimethyl-1H-indole-2-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
1-(2-{2-[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]-1H-imidazol-1-yl}ethyl)imidazolidin-2-one
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}[(1-benzylpiperidin-4-yl)methyl]methylamine
1-butyl-5-(2-propyl-1,3-thiazol-4-yl)-1H-1,2,4-triazole
2,2-dimethylpropyl N-[(3R,5S)-5-(5-oxo-1,4-diazepane-1-carbonyl)pyrrolidin-3-yl]carbamate
N-cyclopropyl-5-(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
1-(2-chlorophenyl)-3-{1-[1-(2-methylpropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
3-(2-methoxyethyl)-3-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(4-methyl-2-oxo-2H-chromen-7-yl)urea
5-ethyl-2-methyl-4-[3-(pyridin-3-ylmethyl)piperidin-1-yl]pyrimidine
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-{3-[(cyclopentylamino)methyl]-4-methoxyphenyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
2-hydroxy-4-(methylsulfanyl)-1-[4-(naphthalen-2-yl)piperazin-1-yl]butan-1-one
9-(4-hydroxy-3-methylbenzoyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-({2-[cyclopentyl(methyl)amino]ethyl}(methyl)amino)acetic acid
2-(1,3-benzoxazol-2-yl)-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]acetamide
4-[3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine-1-carbonyl]-6-(2-methylpropyl)pyrimidin-2-amine
N-[(3-chlorophenyl)methyl]-3-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-4-yl}propanamide
N-({1-[(2-aminopyrimidin-5-yl)methyl]pyrrolidin-3-yl}methyl)-2,4-dimethylbenzamide
N-[4-(2-fluorophenoxy)phenyl]-1-(pyrazine-2-carbonyl)piperidine-2-carboxamide
5-methanesulfonyl-1'-(2-methylpyridin-4-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]urea
N-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}-4-(1H-pyrazol-4-yl)butanamide
N-[(2R,3R)-2-methoxy-1'-(pyridin-3-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(thiophen-2-yl)acetamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(piperidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[5-(naphthalen-2-yl)-1H-imidazol-2-yl]-1-(propan-2-yl)pyrrolidin-2-one
1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-2-(2-methyl-1H-1,3-benzodiazol-1-yl)ethan-1-one