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2-(2,5-dioxoimidazolidin-1-yl)-N-{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}acetamide
[(2-fluoro-5-methoxyphenyl)methyl](methyl)[(2-methyl-1,3-thiazol-4-yl)methyl]amine
5-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2,4-dimethyl-1,3-thiazole
2-{4-[2-amino-6-(thiophen-2-ylsulfanyl)pyrimidin-4-yl]-1-methylpiperazin-2-yl}ethan-1-ol
N-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-1-phenyl-5-(trifluoromethyl)-1H-pyrazole-4-carboxamide
5-{[4-(methylsulfanyl)phenyl]methyl}-5-{3-oxo-3-[(2R,6S)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]propyl}pyrrolidin-2-one
4-(3-fluorophenoxy)-1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidine-4-carboxylic acid
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}benzamide
1-(cyclohexylmethyl)-4-oxo-N3-(propan-2-yl)-N5-[2-(pyridin-3-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
4-{[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyridine
1-[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]cyclopropane-1-carboxamide
N-[(2-chlorophenyl)methyl]-4-(3-hydroxy-3-methylbutyl)-N-(2-hydroxyethyl)benzamide
N-[(3S,7S,8aS)-3-[(2S)-butan-2-yl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-ethylbenzamide
6,7-dimethoxy-3-{[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
ethyl 2-{[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]amino}acetate
N,N,4-trimethyl-5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}pyrimidin-2-amine
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]ethan-1-one
1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-3-(pyridin-3-yl)propan-1-one
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-(cyclopropylsulfamoyl)-5-(2,3-dihydro-1-benzofuran-7-yl)benzoic acid
2-[(4aR,7aS)-4-[(2-fluorophenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
7-chloro-N-[2-(4-methoxyphenyl)ethyl]-3,5-dimethyl-1-benzofuran-2-carboxamide
1-[(3-fluorophenyl)methyl]-4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperazine
3-cyclohexyl-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-4-carboxamide
3-(1-{[2-(difluoromethoxy)phenyl]methyl}piperidin-3-yl)-N-(4-fluoro-2-methylphenyl)propanamide
1-[(3-chlorophenyl)methyl]-5-(2-{[(4-fluorophenyl)methyl]amino}ethyl)pyrrolidin-2-one
6-[(diethylamino)methyl]-N-(4-fluoro-2-methylphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N2-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-N4,6-dimethylpyrimidine-2,4-diamine
7-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}-2-oxa-7-azaspiro[4.5]decan-8-one
3-[({4-benzyl-5-[1-(thiophen-3-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}sulfanyl)methyl]pyridine
2-(3,4-difluorophenyl)-5-methylpyrimidin-4-amine
N-[2-(2-chloro-6-methylphenoxy)ethyl]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-ethyl-4-(1-ethyl-5-methyl-1H-pyrazole-4-sulfonamidomethyl)-4-hydroxyazepane-1-carboxamide
N-[(3S,4R)-4-propyl-1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}pyrrolidin-3-yl]acetamide
6-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)isoquinolin-3-amine
[(1-cyclohexylpiperidin-3-yl)methyl][(3-fluorophenyl)methyl](pyridin-3-ylmethyl)amine
N,N-dimethyl-2-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)acetamide
2-(dimethylamino)-N-methyl-N-(2-phenyl-1-{1-[4-(1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}ethyl)acetamide
N-[2-(2-chlorophenyl)ethyl]-5-(3-methoxyphenyl)-1,2,4-triazin-3-amine
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(3,3,3-trifluoropropyl)piperidine
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-(2-methoxyethyl)-N-propylacetamide
6-(3-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-3-oxopropyl)-2,3-dihydropyridazin-3-one
N,N-dimethyl-5-(4-methylpiperidin-1-yl)-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(2-ethyl-1H-imidazol-1-yl)-N-[3-methyl-1-(propan-2-yl)-1H-pyrazol-5-yl]acetamide
4-chloro-1-methyl-3-{[3-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}-1H-indazole
2-[(4aR,7aS)-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-(1,2-oxazol-3-ylmethyl)acetamide
1-{3-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
N-(4-methoxy-2-methylphenyl)-3-[1-(4-oxo-4-phenylbutanoyl)piperidin-3-yl]propanamide