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2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[(3-methylpyridin-2-yl)methyl]acetamide
[(3R,4R)-1-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
7-(2-ethylbutyl)-3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
3-(2-{4-[1-(dimethylamino)ethyl]phenyl}-1H-imidazol-1-yl)-1-(pyrrolidin-1-yl)propan-1-one
ethyl 3-benzyl-1-{[2-(methylsulfanyl)phenyl]carbamoyl}piperidine-3-carboxylate
{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[3-(morpholin-4-yl)propyl]amine
8-chloro-2-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]quinoline
N-[(2-methyl-6-oxo-1,6-dihydropyrimidin-4-yl)methyl]-9-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
N-({4-[(4-fluorophenyl)methoxy]phenyl}methyl)-4-(2-oxopyrrolidin-1-yl)-N-(pyridin-3-ylmethyl)benzamide
[5-({methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}methyl)furan-2-yl]methanol
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1-ethyl-3-methyl-N-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-[1-(2,5-difluorophenyl)cyclopropyl]-1-methylazepane-2-carboxamide
1-(4-{4-chloro-2-[4-(methoxymethyl)piperidine-1-carbonyl]phenoxy}piperidin-1-yl)ethan-1-one
2-amino-4-(2-aminopyrimidin-5-yl)-6-(3,4-dimethylphenyl)pyridine-3-carbonitrile
2-{1-[(2-cyclohexylpyrimidin-5-yl)methyl]-1,4-diazepan-6-yl}acetic acid
(1R,9aR)-1-({[2-(ethylsulfanyl)ethyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
5-{2-[4-(1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-(morpholin-4-ylmethyl)-N-{2-[(trifluoromethyl)sulfanyl]ethyl}furan-3-carboxamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-oxo-1-phenylpyrrolidine-3-carboxamide
3-(1-propyl-1H-1,2,4-triazol-3-yl)-1-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]urea
(2S,4S)-4-amino-N-(propan-2-yl)-1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}pyrrolidine-2-carboxamide
6-[(1R,5S,8S)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]-2-methylpyrimidin-4-amine
1-(6-hydroxy-1,4-oxazepan-4-yl)-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-2-(2,5-dioxoimidazolidin-4-yl)-N-methylacetamide
1-[3-(morpholin-4-yl)propyl]-6-oxo-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
9-[(2-chloro-3,4-dimethoxyphenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
3-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carboxamide
1-[1-(5-chloro-2,3-dihydro-1H-indole-2-carbonyl)piperidin-4-yl]piperidin-4-ol
1-(2-methoxyethyl)-N-methyl-6-oxo-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)piperidine-3-carboxamide
5-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1,2-dihydropyridin-2-one
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}thiophene-3-carboxamide
N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-3-oxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
4-[(4-fluorophenyl)methyl]-1-(1,2-oxazole-3-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
N-cyclopentyl-N'-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}butanediamide
(1S,5R)-6-(2-methoxyethyl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-N-(1-methyl-1H-pyrazol-4-yl)acetamide
N-benzyl-3-[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]-N-methylpropanamide
8-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-(3-methoxypropyl)-8-[(3-methylquinoxalin-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
4-(1-{6-[(3-methoxyphenyl)methoxy]-4-(2-methylpropyl)-3-oxo-1,4-diazepan-1-yl}-1-oxopropan-2-yl)-1,2-dihydrophthalazin-1-one
(4aS,8aR)-1-(2-aminoethyl)-6-(2,5-dimethylfuran-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-[2-(dimethylamino)ethyl]-7-(5-methylthiophene-2-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-6-(4H-1,2,4-triazol-4-yl)pyridine
2-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1,2-dihydrophthalazin-1-one
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2,2-dimethylpropanamide
1-{3-methyl-5-[2-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-1-yl}butan-2-ol
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-[(4-methylphenyl)amino]-2-phenylpropanamide
1-{2-[1-(3-chloro-2-fluorophenyl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]ethyl}pyrrolidin-2-one
N-(2-{[1-(4-methoxyphenyl)-2,2-dimethylcyclopropyl]formamido}ethyl)pyridine-3-carboxamide