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3-[(2R,3R,6R)-5-(5-fluoro-2-methylbenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-[4-(1-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1H-imidazol-2-yl)phenyl]acetamide
methyl (2S)-2-{[2-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]formamido}-2-phenylacetate
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-3-(thiophen-2-yl)propanamide
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
1-(1-benzothiophene-5-carbonyl)-4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
2-[4-(2-methoxy-5-sulfamoylbenzoyl)morpholin-3-yl]acetic acid
4-[3-(2-methoxybenzoyl)piperidin-1-yl]-2-methylpyrimidine
ethyl 2-[1-(2-methoxypyridine-4-carbonyl)piperidin-2-yl]acetate
1-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}ethan-1-one
1-{2-ethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-4-(1H-pyrrole-2-carbonyl)piperazine
3,3-diethyl-1-{[(2S,4S)-4-fluoro-1-(4-methylpiperazine-1-carbonyl)pyrrolidin-2-yl]methyl}urea
(2S,4S)-4-(3-methoxypropanamido)-N,1-dimethyl-N-(propan-2-yl)pyrrolidine-2-carboxamide
methyl 3-methoxy-5-{2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}benzoate
ethyl 4-{2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamido}piperidine-1-carboxylate
2-amino-6-(4-hydroxyphenyl)-4-[3-(1H-pyrazol-1-yl)phenyl]pyridine-3-carbonitrile
N-(2,1,3-benzothiadiazol-5-ylmethyl)-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
2-[1-(2,3-dihydro-1H-inden-2-yl)pyrrolidin-3-yl]benzoic acid
1-[2-(dimethylamino)acetyl]-N-[4-(2-fluorophenoxy)phenyl]piperidine-2-carboxamide
2-[1-(4-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-[2-(dimethylamino)ethyl]acetamide
2-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
4-oxo-N-[2-(propan-2-yl)phenyl]-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxamide
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)acetamide
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-3-phenoxypropan-1-one
(4aR,7aS)-1-(cyclopropylmethyl)-4-[(4-hydroxy-3,5-dimethylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[3-(4-chlorophenoxy)propyl]-N-methyl-1,9-dioxaspiro[5.5]undecan-4-amine
4-({methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]carbamoyl}amino)-N-(oxolan-2-ylmethyl)benzamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclopentanamine
3-(dimethyl-1,2-oxazol-4-yl)-N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}propanamide
N-(butan-2-yl)-N-cyclopentyl-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
4-{1-[2-(2,3-difluoro-6-methoxyphenyl)-1H-imidazol-1-yl]ethyl}pyrimidine
N-benzyl-1-[(diethylcarbamoyl)methyl]-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
6-(hydroxymethyl)-N-[3-methoxy-5-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-1,4-oxazepane-4-carboxamide
2-(2-aminoethyl)-N-cyclopentyl-N-(prop-2-en-1-yl)quinazolin-4-amine
3-[(cyclopropylamino)methyl]-3-hydroxy-1-[(3-methylphenyl)methyl]piperidin-2-one
N-[(4,6-dimethylpyridin-2-yl)methyl]-N,1,3-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
1-[3-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]-3-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]urea
1-(2-ethoxyethyl)-5-(4-methylpiperazine-1-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
(1S,5R)-6-methyl-3-(3-{[5-(pyridin-4-yl)-1,3,4-oxadiazol-2-yl]sulfanyl}propanoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}-5-methoxypyridin-4-ol
N-methyl-3-(2-oxoazepan-1-yl)-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
3-[3-(morpholin-4-yl)propyl]-1-{3-[(trifluoromethyl)sulfanyl]phenyl}urea
N-tert-butyl-2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carboxamide
1,5,6-trimethyl-N-[(3-methylphenyl)methyl]-2-oxo-N-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
N-cyclohexyl-N-methyl-2-{2-[(4-phenylpiperazin-1-yl)methyl]-4-(pyrimidin-2-yl)phenoxy}acetamide
N-cyclopropyl-4-methoxy-3-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]benzamide
2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}-5-(oxolan-3-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine
3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}propanamide
2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]acetamide