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2-cyclopentyl-1-[4-(3-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]ethan-1-one
N-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-1-(6-methyl-2-propylpyrimidin-4-yl)piperidin-4-amine
4-[(3-hydroxy-2-oxo-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-3-yl)methyl]-1,4-diazepan-2-one
(3S,9aR)-3-[(4-hydroxyphenyl)methyl]-8-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-methoxy-1-[3-(phenylamino)piperidin-1-yl]ethan-1-one
4-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-3,4-dihydro-2H-1,4-benzothiazin-3-one
[1-(5-chlorothiophene-2-carbonyl)-3-(2-phenylethyl)piperidin-3-yl]methanol
4-hydroxy-N-(2-methoxyethyl)-2-methyl-N-(1,3-thiazol-2-ylmethyl)pyrimidine-5-carboxamide
N-methyl-3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}-N-(oxan-4-yl)benzamide
N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
N-methyl-4-{4-[(methylsulfanyl)methyl]piperidine-1-carbonyl}pyridin-2-amine
2-{[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]amino}-N-(2-methylphenyl)acetamide
[1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3-(2-phenylethyl)piperidin-3-yl]methanol
1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
{2-[4-(2H-1,3-benzodioxol-4-ylmethyl)morpholin-2-yl]ethyl}dimethylamine
1-{4-[5-(4-methoxyphenyl)furan-2-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-2-methylpropan-1-ol
3-hydroxy-3-(morpholin-4-ylmethyl)-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
methyl (2S,4S,5R)-4-[(2-methoxy-2-oxoethyl)(methyl)carbamoyl]-1,2-dimethyl-5-(2-methylphenyl)pyrrolidine-2-carboxylate
3-(1H-pyrazol-1-ylmethyl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}benzamide
1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine
ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl){[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}amine
1-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-3-phenylpiperazine
4-(hydroxymethyl)-1-[4-(4-propylphenyl)benzoyl]azepan-4-ol
N-[2-(3-methoxyphenyl)ethyl]-3-(piperidin-4-ylmethyl)benzamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(pyridin-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
2-chloro-N-(1-hydroxybutan-2-yl)-3-methyl-N-(thiophen-3-ylmethyl)benzamide
1-(2-methylpropyl)-4-oxo-N-(propan-2-yl)-5-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
1-[3-(5-benzyl-2-methylpyrimidin-4-yl)piperidin-1-yl]-4-(thiophen-2-yl)butan-1-one
(4aR,6R,8aS)-2-(3-fluoropyridin-2-yl)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinoline
1-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(1H-1,2,4-triazol-1-yl)propan-1-one
N3-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]piperidine-1,3-dicarboxamide
2-methyl-6-[1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-4-yl]pyrimidin-4-ol
1-(4-carboxy-3,5-dimethyl-1H-pyrrole-2-carbonyl)-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
2-methyl-N-[1-(pyrazin-2-yl)propan-2-yl]pyrido[2,3-d]pyrimidin-4-amine
(3S,5S)-5-(4-methylpiperazine-1-carbonyl)-1-(pyridin-4-ylmethyl)piperidine-3-carboxylic acid
4-{[6-ethyl-2-(piperidin-1-yl)pyrimidin-4-yl]amino}-1λ6-thiane-1,1-dione
3-({4-[3-(4-ethoxypiperidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
N-cyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}ethane-1-sulfonamide
2-ethyl-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-7-(2-methoxybenzamido)-N,1-dimethyl-1H-1,3-benzodiazole-5-carboxamide
1-ethyl-N-methyl-N-(2-phenylethyl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(cyclopropylmethyl)-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
N-[furan-2-yl(phenyl)methyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
4-(4-methoxyphenyl)-2-methyl-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperazine
1-[2-(phenylamino)pyrimidine-5-carbonyl]-1,4-diazepan-6-ol
1-{[4-(furan-2-yl)phenyl]methyl}-4-methoxypiperidine
ethyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}){[2-(propan-2-yl)pyrimidin-4-yl]methyl}amine
2-({2-[(1-hydroxy-2-methylpropan-2-yl)carbamoyl]phenyl}amino)acetic acid
N-[2-(1-{[(4-methylphenyl)carbamoyl]methyl}-1,2,3,6-tetrahydropyridin-4-yl)ethyl]acetamide