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2-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-ethyl-2-{methyl[(1-phenyl-1H-pyrazol-4-yl)methyl]amino}pyridine-4-carboxamide
5-chloro-N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-1H-1,2,4-triazole-3-carboxamide
1-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]ethan-1-one
7-[3-(furan-2-yl)-3-phenylpropanoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-methyl-2-(3-methyl-2-oxo-1,2-dihydroquinoxalin-1-yl)-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}acetamide
2-({[5-(1-cyclobutanecarbonylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)ethan-1-ol
N,3-dimethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}furan-2-carboxamide
2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]-4-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}morpholine
N3-(1,3-benzothiazol-2-ylmethyl)-1-cyclohexyl-N3,N5-dimethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-[(6-chloropyridin-3-yl)methyl]-4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazine
(3R,4R)-4-cyclobutyl-1-[1-(2-methoxyethyl)piperidine-4-carbonyl]-3-methylpiperidin-4-ol
1-{4-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
(4aS,7aR)-1-[3-(4-hydroxyphenyl)-1H-pyrazole-5-carbonyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-amino-6-(1H-indol-3-yl)-4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
1-{1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidin-3-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
3-[5-(2-methylpropyl)-4H-1,2,4-triazol-3-yl]-1-[(4-phenyl-1,3-thiazol-2-yl)methyl]urea
methyl 3-{[(2-fluorophenyl)formamido]methyl}-5-(pyridine-4-amido)benzoate
(2R,3R)-3-amino-1'-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
6-(3-chlorophenyl)-2-(4-fluoropiperidine-1-carbonyl)-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
5-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-4-propylpyrimidine
N-[(5-methylthiophen-2-yl)methyl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
1-(cyclohexylmethyl)-3-(pyrrolidin-1-yl)piperidine
2-methyl-4-(2-methylphenyl)-1-(2-propyl-1,3-thiazole-4-carbonyl)piperazine
[(2-chloro-4-fluorophenyl)methyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
(1S,5R)-3-(3-methyl-1H-pyrazole-5-carbonyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]acetamide
(2S,4R)-4-amino-N-ethyl-1-(2-methyl-1-benzofuran-7-carbonyl)pyrrolidine-2-carboxamide
9-[(2-chloro-6-fluorophenyl)methyl]-6-oxa-9-azaspiro[4.5]decane
N-[(1R)-1-(3-methoxyphenyl)ethyl]-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(6-methylpyridine-3-carbonyl)piperidine-2-carboxamide
ethyl 4-(cyclopropylmethyl)-1-(6-ethyl-2-methylquinoline-4-carbonyl)piperidine-4-carboxylate
8-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
(3R)-N-(5-acetamido-2-fluorophenyl)-3-hydroxypyrrolidine-1-carboxamide
1-[1-(2-chloro-6-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(pyridin-3-yl)propan-1-one
2-[1-(4,6-dimethylpyrimidin-2-yl)-1H-pyrazol-4-yl]-6-fluoro-N,N-dimethylquinoline-4-carboxamide
1-cyclopentyl-5-[4-(2,4-dimethylphenyl)piperazine-1-carbonyl]-N-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
N-(1-{1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
N-tert-butyl-2-(2-oxo-5,5-diphenylpiperidin-1-yl)acetamide
2-{4-[4-(azepane-1-carbonyl)-6,8-dimethylquinolin-2-yl]-1H-pyrazol-1-yl}ethan-1-ol
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]propanamide
2-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidine-1-carbonyl]-4-methylphenol
(2S)-1-{4-[3-(3-methoxyphenyl)-1,2,4-oxadiazol-5-yl]butanoyl}pyrrolidine-2-carboxylic acid
3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidine
1-(4-{[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl)amino}piperidin-1-yl)ethan-1-one
(3S,4R)-1-[(4-methylpiperazin-1-yl)sulfonyl]-4-phenylpyrrolidine-3-carboxylic acid
N-ethyl-3-methoxy-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-[(1-methylpiperidin-4-yl)oxy]benzamide
N-[3-(4-methylpiperazin-1-yl)butyl]quinoxaline-6-carboxamide
7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane
2-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}acetamide