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N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-3-(1H-indol-3-yl)propanamide
N-(1-benzylpyrrolidin-3-yl)-3-[1-(pyridine-3-carbonyl)piperidin-4-yl]propanamide
1-({5-[(4-ethoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
2-(2-methylpropyl)-8-(pyridine-3-sulfonyl)-2,8-diazaspiro[4.5]decan-3-one
N3-(1,3-benzothiazol-2-ylmethyl)-N5-tert-butyl-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-{3-[2-(4-methoxyphenyl)ethyl]piperidin-1-yl}but-2-yn-1-one
4-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-1λ6-thiane-1,1-dione
methyl 2-[(1-methoxypropan-2-yl)sulfamoyl]-6-(4-phenylbutanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-benzyl-N,N-dimethyl-5-[methyl(thiophen-2-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-{[1-(butan-2-yl)piperidin-4-yl]oxy}-3-chloro-N-[2-(dimethylamino)ethyl]benzamide
1-methyl-4-(2-propylpyridine-4-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
(3S,7S,8aS)-3-benzyl-7-{[(2,4-difluorophenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
6-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyrimidine-2,4-diamine
1-(3,5-dimethylphenyl)-4-[2-(pyridin-3-yl)acetyl]piperazin-2-one
1-benzyl-8-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
{[3-cyclopropyl-1-(4-fluorophenyl)-1H-1,2,4-triazol-5-yl]methyl}(methyl)amine
1-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-3-yl]-4-(2-fluorophenyl)piperazine
2-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-4-methyl-1H-imidazole
4-{4-[(2-methoxynaphthalen-1-yl)methyl]piperazin-1-yl}-2-[(4-methoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
methyl (2S)-1-{4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}pyrrolidine-2-carboxylate
5-cyclopropanecarbonyl-1'-(1-ethyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[2-(cyclohex-1-en-1-yl)ethyl]-6-(3-phenylprop-2-ynoyl)-6-azaspiro[2.5]octane-1-carboxamide
8-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-butyl-2-[methyl({4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl})amino]acetamide
(3aR,6aS)-5-[4-(hydroxymethyl)benzoyl]-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[4-(furan-2-yl)phenyl]-1-(5-methyl-1,3-oxazole-4-carbonyl)piperidine-3-carboxamide
N-(2-hydroxyethyl)-N-[(5-methylthiophen-2-yl)methyl]-2-(phenylamino)pyrimidine-5-carboxamide
1-[4-(5,6-dimethylpyrimidin-4-yl)piperazin-1-yl]-2-[1-(propan-2-yl)piperidin-4-yl]ethan-1-one
1-methyl-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]azepane-2-carboxamide
7-(2-methoxyacetamido)-1-methyl-N-[(4-methylphenyl)methyl]-2-phenyl-1H-1,3-benzodiazole-5-carboxamide
1-[4-(3-fluorophenoxy)piperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
[(5-tert-butyl-1H-pyrazol-3-yl)methyl]({[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl})amine
2-(2,4-dichlorophenoxy)-N-(oxan-3-yl)acetamide
1-methyl-8-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
4-{4-[3-(4-ethylpiperazin-1-yl)-3-oxopropyl]piperidine-1-carbonyl}-N,N-dimethylpiperidine-1-carboxamide
(3S,4S)-1-[(2-chloro-6-fluorophenyl)methyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(pyridin-3-yloxy)propyl]acetamide
N-(2-hydroxyethyl)-5-methyl-2-phenyl-N-propyl-1H-imidazole-4-carboxamide
ethyl 1-(2,8-dimethylquinoline-4-carbonyl)-4-(2-phenylethyl)piperidine-4-carboxylate
2-(pyridin-4-yl)-N-[3-(1H-1,2,4-triazol-1-yl)propyl]quinoline-4-carboxamide
6-(4-carbamoylphenyl)-N,N-dimethylpyridine-2-carboxamide
2-methanesulfonamido-N-[(3R,4S)-4-propyl-1-(pyridazin-3-yl)pyrrolidin-3-yl]acetamide
5-methanesulfonyl-2-(3-methylbutyl)-4-(piperidin-3-yl)pyrimidine
2-(3-hydroxyphenyl)-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
5-ethyl-4-{4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}pyrimidin-2-amine
N-[2-(4,5-dimethyl-1H-imidazol-1-yl)ethyl]-2-(2,4-dioxo-1,3-diazinan-1-yl)benzamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-ol
N-[4-(4-{[(2,6-dimethoxyphenyl)formamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]furan-3-carboxamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-(pyridin-2-yl)propanamide