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2,4-dioxo-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide
(4aS,7aR)-1-[(2-cyclohexylpyrimidin-5-yl)methyl]-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperidine
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}pyrrolidin-3-yl]acetamide
2-{2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)amino]ethyl}-1,2,3,4-tetrahydrophthalazine-1,4-dione
8-(3-fluoropyridin-4-yl)-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(3S,4R)-4-hydroxyoxolan-3-yl]-N-methyl-3-(4-methylpiperidine-1-carbonyl)benzene-1-sulfonamide
2-(4-{[2-(1-phenylethyl)-1H-imidazol-1-yl]methyl}-1,3-thiazol-2-yl)pyrimidine
N-(3-cyclopentylpropyl)-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-benzyl-5-({[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amino)azepan-2-one
3-ethyl-1-[4-(6-methoxypyridin-2-yl)phenyl]urea
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[3-(2-methoxyphenoxy)azetidin-1-yl]ethan-1-one
2-[methyl(pyridin-3-ylmethyl)amino]-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}acetamide
1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-4-(4H-1,2,4-triazol-3-yl)piperidine
4-{4-[(4-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazine-1-carbonyl}phenol
1-{[6-(5-fluoro-2-methoxyphenyl)pyridin-3-yl]methyl}-4-methylpiperazine
1-(2-fluorobenzoyl)-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-4-(1H-imidazol-1-yl)-N-methylbenzamide
methyl[1-(4-methylpyridin-2-yl)propan-2-yl](quinoxalin-2-ylmethyl)amine
5-(azonane-1-carbonyl)-2-phenylpyrimidin-4-ol
5-{1-[(2-hydroxyphenyl)methyl]pyrrolidin-2-yl}-N-[(1-methyl-1H-pyrazol-4-yl)methyl]thiophene-2-carboxamide
1-(2,3-dimethoxyphenyl)-2-(thiophene-3-carbonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-3,4-dihydro-2H-1-benzopyran-6-carboxamide
N-{[2-(azepan-1-yl)-7-fluoroquinolin-3-yl]methyl}-N-(2-methoxyethyl)furan-2-carboxamide
2-chloro-N-{[1-(cyclopropylmethyl)pyrrolidin-3-yl]methyl}-6-fluorobenzamide
N,4-dimethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1,2,5-oxadiazole-3-carboxamide
6-{4-[(3-fluorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}pyridine-2-carbonitrile
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetamide
1-{7-[cyclohexyl(methoxy)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
methyl 3-{methyl[(3-phenyl-1,2-oxazol-5-yl)methyl]carbamoyl}benzoate
2-(cyclopropylmethyl)-7-(3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
(4aS,7aR)-1-(benzenesulfonyl)-4-(2-methoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-ethyl-1-(2-fluoro-4-methoxyphenyl)-3-(2,2,2-trifluoroethyl)urea
N-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]-3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carboxamide
1-methyl-N-[(5-methylpyrazin-2-yl)methyl]-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[2-(cyclohex-1-en-1-yl)acetyl]-N-[4-(furan-2-yl)phenyl]piperidine-3-carboxamide
4-(1H-imidazol-1-yl)-N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]butanamide
1-{5-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]-2-methylphenyl}imidazolidin-2-one
ethyl 4-{[3-(pyridin-2-yl)phenyl]carbamoyl}piperazine-1-carboxylate
5-(2-{[(2-fluorophenyl)methyl]amino}ethyl)-1-(3-methylbutyl)pyrrolidin-2-one
4-(4-{1-[(2,5-difluorophenyl)methyl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
N-[2-(dimethylamino)-2-(pyridin-2-yl)ethyl]-1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
8-(2-acetylbenzoyl)-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(2-methoxyphenyl)methyl]-2-{6-oxo-7-propyl-2,7-diazaspiro[4.5]decan-2-yl}acetamide
N-(isoquinolin-5-ylmethyl)-N-methyl-3-(pyridin-3-yl)propanamide
3-[2-(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-oxoethyl]-1,3-oxazolidin-2-one
4-[3-(2-methylphenyl)piperidin-1-yl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-amine
methyl 2-(5-methyl-2-{[2-(methylsulfanyl)acetamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)benzoate
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-2-(1H-pyrazol-1-yl)butanamide