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2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(morpholin-4-yl)ethyl]acetamide
N-(2-{7-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-fluorobenzamide
N-[(3R,4S)-1-[3-(dimethylsulfamoyl)propyl]-4-phenylpyrrolidin-3-yl]acetamide
4-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-3,4-dihydro-2H-1,4-benzoxazin-3-one
2-(1-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-1,3-benzothiazole
4-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}-2-(4-methylphenyl)pyridine
3-[(1-cyclopentanecarbonylpiperidin-4-yl)oxy]-N-(pyridin-2-ylmethyl)benzamide
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-(2-methylpropyl)pyrimidin-2-amine
2-({3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}methyl)-5-methoxypyridin-4-ol
N-(2-chlorophenyl)-6-oxo-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decane-2-carboxamide
2,2-dimethyl-N-{1-[1-(2-phenoxypropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl][(5-methylthiophen-2-yl)methyl]amine
methyl({[5-(oxan-2-yl)furan-2-yl]methyl})(1,3-thiazol-2-ylmethyl)amine
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
3-(2-methylphenyl)-1-(1H-1,2,3-triazole-5-carbonyl)pyrrolidin-3-ol
7-(3-chlorophenyl)-9-methoxy-4-[5-(methoxymethyl)furan-2-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(3,5-dimethyl-1-benzofuran-2-carbonyl)-4-(piperidin-1-yl)piperidine-4-carboxamide
2-{5-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-3-(furan-2-yl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
3-(3-hydroxy-3-methylbutyl)-N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}benzamide
1-[(1R,3R,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octan-8-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
N-cyclopentyl-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-[(2-methylphenyl)methyl]acetamide
(3aS,6aS)-2-cyclopropanecarbonyl-5-[(pyridin-3-yl)carbamoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}pyridine-2-carbonitrile
7-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinoxalin-2-one
1-[2-chloro-5-(morpholine-4-carbonyl)phenyl]-3-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]urea
4-(benzenesulfonyl)-2-(2-phenylethyl)morpholine
(3S,9aR)-3-ethyl-8-(2-fluorobenzenesulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(8-{[4-(2-methylpropyl)phenyl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]acetamide
5-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-5-[(2-fluorophenyl)methyl]imidazolidine-2,4-dione
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-3-(1H-pyrazol-1-ylmethyl)benzamide
3-(azetidine-1-carbonyl)-N-methyl-N-(thian-4-yl)benzene-1-sulfonamide
1-{1-[6-(6-aminopyridin-3-yl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
2-(azepan-1-yl)-1-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)ethan-1-one
4-({2-cyclopentyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}methyl)benzoic acid
4-(5-fluoro-3-methyl-1H-indol-2-yl)-1-methyl-3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4-({3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenol
(3S)-3-amino-3-{cyclopropyl[(4-ethoxyphenyl)methyl]carbamoyl}propanoic acid
2-methyl-2-{4-[3-(pyrrolidin-1-yl)pyrazin-2-yl]phenyl}propanenitrile
N-[2-(ethanesulfonyl)ethyl]-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
(2S)-4-(benzyloxy)-2-[(1-methyl-1H-indol-6-yl)formamido]butanoic acid
5-(2,3-dihydro-1H-inden-2-yl)-N-(3-methoxypropyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(2-ethylpyrimidin-4-yl)methyl]-2-(3-fluorophenyl)azepane
1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
(2S)-2-amino-3-(1H-imidazol-4-yl)-1-[4-(pyrrolidin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]propan-1-one
1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]-3-(4-hydroxy-2-methylquinolin-3-yl)propan-1-one
N-{3-[(3R,4S)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]-3-oxopropyl}methanesulfonamide
(1R,5S,6R)-3-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
(2S,4R)-4-amino-1-[2-(2,3-dimethylphenoxy)acetyl]-N,N-diethylpyrrolidine-2-carboxamide
5-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-4-methyl-1H-imidazole
N-[(2,6-dimethoxyphenyl)methyl]-4-(pyrrolidin-3-yl)benzamide