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{[1-(2-methoxyethyl)-2-(3-methylbutanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[(1-methylpiperidin-2-yl)methyl]amine
1,3-dimethyl-4-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-1H-pyrazolo[3,4-d]pyrimidine
2-ethyl-9-[(2-fluoro-4-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
4-{1-[(4-fluorophenyl)methyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}azepane
1-{2-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-oxoethyl}piperidin-2-one
6-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyrimidin-4-amine
1-[(4aR,8aS)-1-(thiophen-2-ylmethyl)-decahydro-1,6-naphthyridin-6-yl]-3-phenoxypropan-1-one
(1S,5R)-3-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-N-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
2-[2-(morpholin-4-yl)ethyl]-2H-1,2,3-benzotriazole
1-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-4-(thiophen-2-ylmethyl)piperazine
N-[3-(4-{[2-(furan-2-yl)ethyl]amino}piperidin-1-yl)phenyl]pyridine-4-carboxamide
1-({1-[(4-fluorophenyl)methyl]-3-methyl-1H-1,2,4-triazol-5-yl}methyl)-5-(trifluoromethyl)-1,2-dihydropyridin-2-one
2-[(2,3-dimethoxyphenyl)methyl]-4-[4-(oxolane-2-carbonyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
3-(4-hydroxyphenyl)-1-[(1R,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-2-(dimethylamino)-2-(2-methylphenyl)acetamide
6-(cyclopropylmethoxy)-1-[(3-methoxyphenyl)methyl]-4-(3-oxo-2,3-dihydro-1H-indene-1-carbonyl)-1,4-diazepan-2-one
4-[(4-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methyl]-3-ethylpiperazin-2-one
N-[(2R,3R)-2-(pyridin-3-ylmethoxy)-1'-(1,2,5-thiadiazole-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
ethyl 4-[(4-methoxyphenyl)methyl]-1-[3-(pyrazin-2-yl)propanoyl]piperidine-4-carboxylate
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-2-phenoxyacetamide
1-[1-(diphenylmethyl)-1H-1,2,3-triazole-4-carbonyl]-4-(2-methoxyethoxy)piperidine
2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}acetamide
1-(3-phenyl-1H-pyrazole-4-carbonyl)-4-(thian-4-yl)piperazine
1-(2,3-dihydro-1-benzofuran-5-ylmethyl)-4-[(4-fluorophenyl)methyl]-1,4-diazepan-5-one
methyl 6-(2-cyclopropylacetyl)-2-{[(4-fluorophenyl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-{4-[1-(2,2,2-trifluoroethyl)-1H-imidazol-2-yl]phenoxy}acetamide
N-(1H-imidazol-2-ylmethyl)-N-methyl-2-(phenylamino)pyrimidine-5-carboxamide
9-hydroxy-2-{[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-4H-pyrido[1,2-a]pyrimidin-4-one
2-{2-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]phenyl}ethan-1-amine
1-butanoyl-N-[3-(1H-indol-2-yl)phenyl]piperidine-3-carboxamide
1-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-yl]-4-(2-fluorophenyl)piperazine
4-[3-(3-methylpiperidin-1-yl)-3-oxopropyl]piperazin-2-one
N-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
2-methyl-1-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidine
1-{[3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}piperidine-4-carboxamide
1-tert-butyl-4-({4-oxo-3H,4H-pyrido[4,3-d]pyrimidin-3-yl}methyl)pyrrolidin-2-one
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N-methyl-2-(1H-pyrazol-1-yl)-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
3-(5-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,2,4-oxadiazol-3-yl)pyridine
1-(furan-2-carbonyl)-N-[4-(3-methoxyphenyl)phenyl]pyrrolidine-2-carboxamide
{[5-(methoxymethyl)furan-2-yl]methyl}(methyl)[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amine
4-(4-methyl-1H-pyrazol-1-yl)-1-[2-(2-oxopyrrolidin-1-yl)propanoyl]piperidine-4-carboxylic acid
2-methoxy-1-(1'-{spiro[2.4]heptane-1-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)ethan-1-one
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-1,2,5-thiadiazole-3-carboxamide
2-ethyl-4-({2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-1-(propan-2-yl)piperazine
(2-ethoxy-5-{[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]methyl}phenyl)methanol
4-{1-[2-(1H-imidazol-4-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}pyridine
4-{4-[(3-chlorophenyl)methyl]piperazine-1-carbonyl}-1-methylimidazolidin-2-one
5-(2,4-dimethoxyphenyl)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-1,2,4-triazin-3-amine