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(4aR,7aS)-1-acetyl-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S,4R)-4-amino-1-[(2-chloro-6-fluoro-3-methylphenyl)methyl]-N-methylpyrrolidine-2-carboxamide
2-[4-(propan-2-yl)phenyl]-N-(4H-1,2,4-triazol-4-yl)acetamide
1-[1-(2-cyclooctyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)piperidine-4-carbonyl]-N,N-diethylpiperidine-3-carboxamide
4-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-1λ6-thiomorpholine-1,1-dione
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methyl-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
ethyl(methyl){[5-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}amine
1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(pyrrolidin-1-yl)ethan-1-one
1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine
5-{4-[(2-methylphenyl)methyl]piperazine-1-carbonyl}-2-(pyridin-3-yl)pyrimidine
4-[(3,5-dimethoxyphenyl)methyl]-9-methoxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]pyridine
2-{3-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-3-oxopropyl}-2,3-dihydro-1H-isoindol-1-one
N-ethyl-1-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}-N-(pyridin-4-ylmethyl)piperidin-3-amine
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-[(2-methyl-1-benzothiophen-3-yl)methyl]piperidin-4-ol
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-5-(2-methylphenyl)-1,2,4-triazin-3-amine
4-acetyl-N-ethyl-N-{[3-(prop-2-en-1-yloxy)phenyl]methyl}benzamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}benzamide
1-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-2-(1,3-thiazol-2-yl)piperidine
2-[1-(2,3-dihydro-1H-inden-2-yl)-1H-pyrazol-4-yl]-N,N-dimethylquinoline-4-carboxamide
2-(4-methoxy-2-methylphenyl)-5-(pyrrolidin-1-ylmethyl)pyridine
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
5-chloro-3-(pyridin-4-ylmethyl)-3,4-dihydroquinazolin-4-one
2-(2,5-dioxoimidazolidin-1-yl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
(3R)-4-{[2-(propan-2-yloxy)naphthalen-1-yl]methyl}morpholine-3-carboxylic acid
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
N-[(3S)-1-benzylpiperidin-3-yl]-[1,2,4]triazolo[4,3-a]pyridine-7-carboxamide
5-(adamantan-1-ylmethyl)-3-[(methylsulfanyl)methyl]-1,2,4-oxadiazole
(2S,4S)-4-amino-1-methyl-N-(5,6,7,8-tetrahydronaphthalen-2-ylmethyl)pyrrolidine-2-carboxamide
N,6-dimethyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]pyridine-2-carboxamide
2-(2-chloro-4-fluorophenoxymethyl)-N-(2-oxopiperidin-3-yl)-1,3-oxazole-4-carboxamide
1-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}-2-(piperidin-1-yl)ethan-1-one
4-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}thiomorpholine
2-(4-chloro-2-fluorophenyl)-1-[2-(1H-imidazol-1-yl)ethyl]-1H-imidazole
2-[(2-{[(1-hydroxycyclohexyl)methyl]carbamoyl}phenyl)amino]acetic acid
methyl 4-[({1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}amino)methyl]benzoate
2-{methyl[(4-methylphenyl)methyl]amino}-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]ethan-1-one
4-{[1-(1-ethyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]oxy}-N-(2-phenylethyl)benzamide
N-(2-{1-[(4-chlorophenyl)methanesulfonyl]piperidin-2-yl}ethyl)acetamide
N-[1,3-dihydroxy-2-(hydroxymethyl)propan-2-yl]-2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-propyl-N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}-1,3-thiazole-4-carboxamide
8-(2-ethylpyrimidine-5-carbonyl)-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(4-{[(3S,4S)-3-hydroxy-4-(piperidin-1-yl)pyrrolidin-1-yl]methyl}phenoxy)acetic acid
N-[1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine
2-(2H-indazol-2-yl)-1-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
N-(2-chloropyridin-3-yl)-3-(3-methoxyphenoxymethyl)piperidine-1-carboxamide
5-(2-cyclopentylacetamido)-1-methyl-2-(oxolan-2-yl)-N-(thiophen-3-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
5-phenyl-N-(pyrrolidin-2-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
2-{[3-({[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}carbamoyl)phenyl]amino}acetic acid