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2-(2-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methoxy}phenoxy)acetamide
5-[3-(2-methoxyphenyl)phenyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-[benzyl({[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl})amino]ethan-1-ol
3-{[1-ethyl-3-(4-phenylpiperazine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}phenol
5-{1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-2-yl}-N-(pyridin-4-ylmethyl)thiophene-2-carboxamide
2-methoxy-N-[2-methyl-3-({methyl[2-(methylsulfanyl)ethyl]carbamoyl}amino)phenyl]acetamide
N-[(3R,4S)-4-cyclopropyl-1-(2-methanesulfonylethyl)pyrrolidin-3-yl]-3,5-dimethyl-1,2-oxazole-4-carboxamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]propanamide
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
1-[6-(morpholin-4-yl)pyridine-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
3-[2-(dimethylamino)ethyl]-5-[1-(3,5-dimethylbenzoyl)piperidin-4-yl]-5-[(3-fluorophenyl)methyl]imidazolidine-2,4-dione
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
3-({[2-(2-ethyl-1H-imidazol-1-yl)ethyl]carbamoyl}amino)-2-methylbenzamide
4-chloro-3-[4-(3,6-dimethylpyrazin-2-yl)piperazine-1-carbonyl]-1H-pyrazol-5-amine
N-[4-(2-fluorophenoxy)phenyl]-1-(3-methylbut-2-en-1-yl)piperidine-4-carboxamide
1-{[1-(4-methylphenyl)pyrrolidin-3-yl]methyl}-3-[1-(2,2,2-trifluoroethyl)-1H-pyrazol-4-yl]urea
{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}(methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
6-acetyl-2-amino-4-(6-methyl-2H-1,3-benzodioxol-5-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-{4-[(3-cyclopropyl-1H-1,2,4-triazol-5-yl)methoxy]phenyl}-1H-1,2,3,4-tetrazole
4-methyl-N-(2-{7-[(4-phenylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-methyl-N-(quinoxalin-6-ylmethyl)benzamide
4-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1-{[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}piperidin-4-ol
3-[3-(oxolan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]pyridine
4-methyl-N-{[8-methyl-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}-1,3-oxazole-5-carboxamide
3-(2-ethoxyphenyl)-5-{imidazo[1,2-a]pyridine-2-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3,5-dimethyl-N-[2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-1,2-oxazole-4-carboxamide
2,3-dimethyl-N-[2-(N-methylmethanesulfonamido)ethyl]-1H-indole-7-carboxamide
3-(2,1,3-benzothiadiazol-5-ylmethyl)-6-fluoro-3,4-dihydroquinazolin-4-one
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[2-(methylsulfanyl)ethyl]benzamide
1-[(4-chlorophenyl)methyl]-N-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
N-[1-(4-methylphenyl)ethyl]-2-{[(4-sulfamoylphenyl)methyl]amino}acetamide
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-(quinoline-2-carbonyl)pyrrolidin-3-yl]methanol
1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methoxypiperidine
methyl 3-(2,5-difluorobenzoyl)-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-{4-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
ethyl[(4-ethylphenyl)methyl](pyridin-3-ylmethyl)amine
1-(3,5-dimethylphenyl)-4-[3-(pyridin-3-yl)propanoyl]piperazin-2-one
5-fluoro-N4-methyl-N2-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}pyrimidine-2,4-diamine
2-methanesulfonyl-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}acetamide
1-[(1-ethyl-1H-imidazol-5-yl)methyl]-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-benzyl-1-methyl-5-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(1S,5R)-6-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-cyclohexyl-3-(cyclopropylmethyl)-N-(3-hydroxy-3-methylbutyl)-N-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-cyclobutanecarbonyl-N-[1-(pyridin-4-yl)propan-2-yl]piperidine-4-carboxamide
5-{[benzyl(methyl)amino]methyl}-N-ethyl-N-(oxan-2-ylmethyl)-1,2-oxazole-3-carboxamide
3-[1-(5-acetylthiophene-3-carbonyl)piperidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide