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3-{[4-(4-methylbenzenesulfonyl)piperazin-1-yl]methyl}piperidin-3-ol
[(3R,5R)-1-(3-methylpyrazin-2-yl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
N-{5-[(4-chlorophenyl)methyl]-1,3,4-thiadiazol-2-yl}-1,1-dioxo-1λ6-thiomorpholine-4-carboxamide
3-oxo-N-[3-(pyridin-3-yl)propyl]-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
5-(3,5-dimethoxyphenyl)-1,2,3,4-tetrahydroisoquinoline
2-[3-cyclopropyl-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]phenol
ethyl 2-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]acetate
1-{4-[hydroxy(pyridin-2-yl)methyl]piperidin-1-yl}-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethan-1-one
3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-{2-methylthieno[3,2-d]pyrimidin-4-yl}piperidine
N-[(2,3-dimethoxyphenyl)methyl]-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
7-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-2-oxa-7-azaspiro[4.5]decan-8-one
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(4-methoxyphenyl)acetamide
(4aR,7aS)-1-[2-(2-chloro-4-fluoro-3-methylphenoxy)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(3-methylphenyl)methyl]-N-(oxolan-2-ylmethyl)-3-(pyridin-4-yl)propanamide
3,4-difluoro-N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)benzene-1-sulfonamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)quinoline-2-carboxamide
N-[3,3-dimethyl-1-(pyridin-3-yl)butyl]-5-methyl-1,3,4-oxadiazol-2-amine
4-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}phenyl)-1-phenyl-1H-imidazole
N-[(4-methoxyphenyl)(pyridin-4-yl)methyl]imidazo[1,2-a]pyridine-6-carboxamide
N-cyclopentyl-2-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propanamide
1-(4-benzoylpiperazin-1-yl)-2-(morpholin-2-yl)ethan-1-one
3-fluoro-4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}pyridine
2-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrazine
methyl 3-(1,3-dimethyl-1H-pyrazole-5-amido)-5-{[(5-methyl-3-phenyl-1,2-oxazol-4-yl)formamido]methyl}benzoate
(1S,5R)-6-(3,5-difluoropyridine-2-carbonyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(2S)-2-[2-(2-methyl-1,3-thiazol-4-yl)acetamido]pentanoic acid
1-(2,3-dimethoxybenzoyl)-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
1-benzyl-N3-cyclopropyl-N5-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl}-2,8-diazaspiro[4.5]decane
(2S,4S)-4-{4-[4-(2,3-dihydro-1H-isoindol-2-ylmethyl)phenyl]-1H-1,2,3-triazol-1-yl}-N-methylpyrrolidine-2-carboxamide
(1-{5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}piperidin-3-yl)methanol
1-cyclopentanecarbonyl-N-(2-methoxyethyl)-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[(1-methyl-1H-pyrazol-4-yl)methyl]amine
1-[1-(2-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(pyridin-2-yl)propan-1-one
(5-{[methyl(quinolin-5-ylmethyl)amino]methyl}furan-2-yl)methanol
N-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-4-(trifluoromethyl)benzamide
methyl (1R,3S,3aR,6aS)-5-methyl-4,6-dioxo-1-(propan-2-yl)-3-[2-(propan-2-yl)pyrimidin-4-yl]-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
2-(4-{[4-(difluoromethoxy)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-1-(dimethylamino)propan-2-ol
3-(2-{[5-(4-cyclohexylphenyl)-1,2,4-triazin-3-yl]amino}ethyl)-1,3-oxazolidin-2-one
2-methyl-6-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
4-methyl-9-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-2H,3H,4H,6H,7H,8H,9H-[1,4]oxazino[2,3-g]quinoline-3,7-dione
N-[(3-methoxyphenyl)methyl]-6-methyl-N-(prop-2-en-1-yl)imidazo[2,1-b][1,3]thiazole-5-carboxamide
2-methyl-4-(5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}furan-2-yl)but-3-yn-2-ol
ethyl 1-({4-[(thiophen-2-ylmethyl)amino]quinazolin-2-yl}methyl)piperidine-3-carboxylate
(3S)-3-[({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)amino]azepan-2-one
5-(3,4-dimethylphenyl)-3-methyl-1H-1,2,4-triazole
(1R,5S,8S)-3-[(5-chlorofuran-2-yl)methyl]-N,N-dimethyl-3-azabicyclo[3.2.1]octan-8-amine
2-methoxy-N-(4-{1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)acetamide
N-(cyclopentylmethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
N-methyl-4-(pyridin-3-yl)-N-(1,3-thiazol-2-ylmethyl)pyrimidin-2-amine