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N-(4-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-4-oxobutyl)acetamide
1-(2-hydroxyethyl)-4-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1,4-diazepan-6-ol
(1R,3s,6r,8S)-4-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-4-azatricyclo[4.3.1.13,8]undecane
2-(adamantan-1-yl)-N-[(2-aminopyrimidin-5-yl)methyl]-N-methylacetamide
6-[1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-2-methylpyrimidin-4-ol
4-{3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-4-oxobutanamide
4-({3-[4-(piperazin-1-ylmethyl)phenyl]phenyl}methyl)morpholine
N-(1-{7-[(3,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2,5-difluorobenzamide
N-(2-phenylethyl)-6-(thiophene-2-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
N-ethyl-N-methyl-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
2-(4-chlorophenyl)-2-{[3-(5-methylfuran-2-yl)-1H-pyrazol-5-yl]formamido}acetic acid
1-ethyl-4-[4-(4-methylphenoxy)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
N-(2-methylprop-2-en-1-yl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
3-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
(3R,4R)-1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-4-ethylpiperidine-3,4-diol
2-{4-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
(3R,5S)-N3-(4-fluorophenyl)-N5-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)piperidine-3,5-dicarboxamide
N,N,2-trimethyl-7-(3,4,5-trimethoxybenzoyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(4-methyl-1H-imidazole-5-carbonyl)piperidine
6-{3-[1-(but-2-yn-1-yl)-1H-pyrazol-3-yl]phenyl}-N,N-dimethylpyridazin-3-amine
4-hydroxy-N-[(1S)-2-hydroxy-1-phenylethyl]-2-(phenoxymethyl)pyrimidine-5-carboxamide
2-(2-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-2-oxoethyl)-2-azaspiro[4.5]decan-3-one
2-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-2-oxoethyl}-4-methyl-1,2-dihydrophthalazin-1-one
4-(1,3-benzothiazol-2-yl)-2-{[4-(piperidin-1-yl)piperidin-1-yl]methyl}phenol
benzyl[(2-butyl-1H-imidazol-4-yl)methyl](1,3-thiazol-2-ylmethyl)amine
2,4-dimethyl-N-[4-(4-{[2-(methylsulfanyl)ethyl]amino}piperidin-1-yl)phenyl]benzamide
tert-butyl(1H-imidazol-2-ylmethyl)(thiophen-3-ylmethyl)amine
2-(2-{[2-(2-hydroxyethyl)pyrrolidin-1-yl]methyl}phenoxy)ethan-1-ol
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
N-cyclohexyl-1-methyl-2-oxo-6-(propan-2-yl)-N-(pyridin-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
5-{[4-(3-fluorophenoxy)piperidin-1-yl]methyl}-N-propylpyrimidin-2-amine
2-{[5-(2,3-dimethylphenyl)-4-methyl-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-[2-(dimethylamino)ethyl]-3-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}propanamide
4-(1H-imidazol-1-ylmethyl)-1-[2-(pyrrolidin-3-yl)benzoyl]piperidin-4-ol
N-[3-(3-fluorophenyl)phenyl]-1-methanesulfonylpiperidine-4-carboxamide
2-cyclopropyl-8-(5-fluoropentyl)-2,8-diazaspiro[5.5]undecan-3-one
1-{[1-(1-phenyl-1H-1,2,3-triazole-5-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
1-benzyl-8-cyclohexyl-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 4-({4-[(3-fluorophenyl)methyl]-1,4-diazepan-1-yl}methyl)thiophene-2-carboxylate
N-(1-benzyl-1H-pyrazol-3-yl)-2-[4-(pyridin-2-yl)-1H-pyrazol-1-yl]acetamide
[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl](methyl)[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]amine
2-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-1-(pyridin-3-yl)ethan-1-ol
N-[2-(dimethylamino)ethyl]-N-{[2-(4-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
6-[3-(1H-pyrazol-1-yl)benzoyl]-5,6,7,8-tetrahydro-1,6-naphthyridine
(1R,2R,4R)-N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}bicyclo[2.2.1]hept-5-ene-2-carboxamide
1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
3-[1-(2-ethoxypyridine-3-carbonyl)piperidin-4-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl 3-acetamido-1-[2-(4-methoxyphenyl)ethyl]-5-[(pentan-3-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-[(2,6-dimethylpyridin-3-yl)oxy]-1-(pyrrolidine-1-carbonyl)piperidine-4-carboxylic acid
5-[(4-ethylpiperazin-1-yl)methyl]-N-methyl-N-(2-phenylethyl)-1,2-oxazole-3-carboxamide