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5-({2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)-2-(pyrrolidin-1-yl)pyrimidine
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
2-[5-(3-phenyl-1,2,4-oxadiazol-5-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
15-methyl-9-(3-methylthiophen-2-yl)-N-[2-(morpholin-4-yl)ethyl]-13-oxo-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
1-[2-({[2-(ethylamino)pyrimidin-5-yl]methyl}(methyl)amino)ethyl]cyclopentan-1-ol
N-(2-{7-[(3,5-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
1-{5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-4-ol
7-(cyclobutylmethyl)-2-(3-methylpyrazin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
5-[1-(4-methyl-1,3-thiazole-5-carbonyl)pyrrolidin-2-yl]-N-(2-methylpropyl)thiophene-2-carboxamide
(1S,5R)-3-benzyl-6-[(2-fluoro-5-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
3-[1-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]benzoic acid
1-[cyclohexyl(methyl)amino]-3-(3-{[4-(2-methoxyethoxy)piperidin-1-yl]methyl}phenoxy)propan-2-ol
N-tert-butyl-2-({2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)acetamide
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-1-[3-(4-methylphenoxymethyl)piperidin-1-yl]propan-1-one
methyl (2S,4S)-1-[(4-methoxy-3-methylphenyl)methyl]-4-[2-(1H-pyrazol-1-yl)benzamido]pyrrolidine-2-carboxylate
2-[3-(furan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-5-methyl-1,3-benzoxazole
(2S)-N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(2-methoxyacetyl)pyrrolidine-2-carboxamide
ethyl 1-[(3-{[1-(quinoline-8-sulfonyl)piperidin-4-yl]oxy}phenyl)methyl]piperidine-2-carboxylate
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]benzamide
(2R,3R)-3-amino-1'-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-(1H-1,3-benzodiazol-2-yl)-2-({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}amino)acetamide
9-(pent-2-yn-1-yl)-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(1-{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-1,4-diazepan-5-one
[(3R,4R)-1-[(4-chloro-3-fluorophenyl)methyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
5-{[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-2-ethoxypyridine
4-methoxy-N-{2-[7-(quinolin-7-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}benzamide
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-propoxyacetamide
1-{2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}pyrrolidin-3-ol
N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1,3-benzothiazol-5-amine
1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-(oxan-4-yl)piperazine
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-3-amine
2-methyl-8-[(4-methyl-2-oxo-2H-chromen-7-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-cyclopentyl-5-(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)piperidin-2-one
(4aS,7aR)-1-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
6-(3-chlorophenyl)-N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
(3aS,6aR)-3-[(2-methoxyphenyl)methyl]-N,N-dimethyl-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-sulfonamide
4-[1-(2,3-dihydro-1H-inden-4-yl)-1H-imidazol-2-yl]pyridine
N-({1-[3-(morpholin-4-yl)propanoyl]piperidin-3-yl}methyl)-1-phenylmethanesulfonamide
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-butoxyethan-1-one
N-[(4-hydroxyazepan-4-yl)methyl]-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
2-{5-[(dimethyl-1,3-thiazol-5-yl)methyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}-4-methylpyridine
5-({3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}methyl)-N-methylfuran-2-carboxamide
1-[2-({[3-(trifluoromethyl)pyridin-2-yl]amino}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]ethan-1-one
1-methanesulfonyl-N-[2-(3-phenylpiperidin-1-yl)ethyl]piperidin-4-amine
ethyl 3-[(3-chlorophenyl)methyl]-1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidine-3-carboxylate
1-cyclobutanecarbonyl-N-methyl-N-(pyrazin-2-ylmethyl)piperidine-4-carboxamide