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2-(1H-1,3-benzodiazol-1-ylmethyl)-N-(2-hydroxyethyl)-1,3-oxazole-4-carboxamide
1-[3-(4-methoxyphenyl)phenyl]-N-(pyridin-4-ylmethyl)piperidin-4-amine
N-cyclopropyl-6-methyl-N-[(5-methylthiophen-2-yl)methyl]-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
1-{5-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}-2-methyl-1,4-diazepan-5-one
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(3-methylfuran-2-carbonyl)-2,7-diazaspiro[4.5]decane
N,N-diethyl-1-{4-[4-(oxane-4-amido)-1H-pyrazol-1-yl]benzoyl}piperidine-3-carboxamide
1-(diphenylmethyl)-4-[(1-ethyl-1H-imidazol-2-yl)methyl]piperazine
5-[(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}propyl)sulfanyl]-1-phenyl-1H-1,2,3,4-tetrazole
3-methoxy-N-(2-methoxyethyl)-N-{[6-methyl-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}benzamide
{3-[(4-fluorophenyl)methyl]-1-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}piperidin-3-yl}methanol
8-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-[3-(naphthalene-1-carbonyl)piperidine-1-carbonyl]benzaldehyde
N-(2-oxoazepan-3-yl)-3-(4H-1,2,4-triazol-4-yl)benzamide
7-chloro-3-{[(1-hydroxy-2-methylpropan-2-yl)amino]methyl}-1-(2-phenoxyethyl)-1,2-dihydroquinolin-2-one
3-methyl-2-[2-(4H-1,2,4-triazol-4-yl)propyl]pyridine
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-methyl-N-[(5-methylfuran-2-yl)methyl]acetamide
2-(3-hydroxypropyl)-8-(6-phenylpyridazin-3-yl)-2,8-diazaspiro[5.5]undecan-3-one
N,N-bis(1,3-oxazol-4-ylmethyl)-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-9-(furan-2-carbonyl)-1-methyl-1,4,9-triazaspiro[5.5]undecane
N,N-diethyl-2-(4-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1H-1,2,3-triazol-1-yl)acetamide
N-methyl-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-2,3-dihydro-1-benzothiophene-2-carboxamide
6-[(diethylamino)methyl]-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(2,3,6-trifluorophenyl)ethan-1-one
4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,2,3,4-tetrahydroquinolin-2-one
N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-1-[3-(1H-pyrazol-1-yl)propyl]piperidine-3-carboxamide
2-{4-[(4-ethoxyphenyl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
4-{2-[3-ethyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-N-methylbenzene-1-sulfonamide
N-{3-[ethyl(phenyl)carbamoyl]phenyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
N-methyl-N-[2-phenyl-1-(1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-4-yl)ethyl]thiophene-3-carboxamide
(3aR,6aR)-2-cyclopropanecarbonyl-5-{[4-(3-hydroxyprop-1-yn-1-yl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-benzyl-N,2-dimethyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-sulfonamide
5-acetyl-N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)thiophene-2-carboxamide
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-3-(4-methylpiperazin-1-yl)propanamide
N-[(3R,4S)-4-cyclopropyl-1-(2-methanesulfonylethyl)pyrrolidin-3-yl]-3-ethyl-1H-pyrazole-5-carboxamide
(3S,4R)-4-methyl-1-[4-(trifluoromethyl)pyridin-2-yl]piperidine-3,4-diol
1-methyl-2-phenyl-4-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperazine
3-[(2-methylphenyl)methyl]-1-(pyrimidin-2-yl)piperidine-3-carboxylic acid
1-[(diethylcarbamoyl)methyl]-N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
3-fluoro-N,6-dimethyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}imidazo[1,2-a]pyridine-2-carboxamide
N-[(1S,2R)-2-(cycloheptylamino)cyclobutyl]-4-methyl-1,2,5-oxadiazole-3-carboxamide
8-(5-hydroxypyridine-2-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
N2-cyclopropyl-7-methyl-N4-[(2-methyl-1,3-thiazol-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
{[2-(4-fluorophenyl)-6-methylquinolin-3-yl]methyl}(methyl)(1,2-oxazol-5-ylmethyl)amine
7-(2-methoxyethyl)-2-(oxan-4-yl)-2,7-diazaspiro[4.5]decane
2-(2-{1-[2-(phenylsulfanyl)ethyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
N3-cyclohexyl-1-cyclopropyl-4-oxo-N5-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
N-{1-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]pyrrolidin-3-yl}acetamide
3-{[(furan-3-ylmethyl)carbamoyl]methyl}-N-(2-methoxyethyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-{[(3R,4R)-1-(furan-3-ylmethyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
N-(2-methoxyethyl)-3-(5-methylthiophen-2-yl)-N-(1,3-thiazol-2-ylmethyl)-1H-pyrazole-5-carboxamide