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8-methoxy-5-[5-(morpholin-4-ylmethyl)pyridin-2-yl]quinoline
5-[1-(2,6-dimethylhept-5-en-1-yl)piperidin-4-yl]-5-propyl-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
2-[3-(2-hydroxyethyl)-4-methylpiperazin-1-yl]-4,6-dimethylpyridine-3-carbonitrile
1-cyclohexyl-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}piperidine-4-carboxamide
(2E)-1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-3-(pyridin-4-yl)prop-2-en-1-one
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-6-methoxypyrimidin-4-amine
4-[2-(1H-pyrazol-1-yl)ethyl]-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperidine
3-[(3R,4S)-1-(4-fluoro-2-methylbenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
(1S,5R)-3-[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[1-(1,2-oxazole-3-carbonyl)-4-phenylpiperidin-4-yl]ethan-1-one
N-{1-[6-ethyl-2-(piperidin-1-yl)pyrimidin-4-yl]pyrrolidin-3-yl}-N-methylacetamide
2-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}-4-(propan-2-yl)-1,3-thiazole
2-{[4-(2-methoxy-5-methylphenyl)-5-(1H-pyrazol-5-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
3-{1-[2-(1H-imidazol-4-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}-2-methoxyquinoline
N-[(4-fluorophenyl)methyl]-3-methyl-N-(prop-2-en-1-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
5-[(2-fluoro-5-methoxyphenyl)methyl]-5-(3-oxo-3-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}propyl)pyrrolidin-2-one
N-[(3R,4R)-1-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
1-(2-hydroxyethyl)-N-[(1-methanesulfonylpiperidin-3-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
3-(morpholine-4-sulfonyl)-N-[3-(1H-1,2,4-triazol-1-yl)propyl]benzamide
[(3R,4R)-1-(2-amino-5,6,7,8-tetrahydroquinazoline-4-carbonyl)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
6-(4-fluorophenyl)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-[3-(1-methyl-1H-pyrazol-3-yl)phenyl]benzonitrile
2-(4-{[3-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}phenoxy)acetic acid
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-2-(3-fluorophenyl)-1,3-benzoxazole-5-carboxamide
N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-4-(2-methylpyrrolidine-1-carbonyl)benzene-1-sulfonamide
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-3-(1-methyl-1H-pyrazol-4-yl)propanamide
3-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-4,5,6,7-tetrahydro-1H-indazole
8-methyl-N-(3-phenylpropyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
methyl 4-[(2-chloro-4-fluoro-5-methylphenyl)carbamoyl]piperazine-1-carboxylate
N-[(3S,4R)-1-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
1-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-hydroxy-4-methylpentan-1-one
4-(4-fluoro-2-methylphenoxy)-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine-4-carboxylic acid
dimethyl(2-{2-[1-(quinoline-6-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
3-chloro-4-{[1-(cyclohexylmethyl)piperidin-4-yl]oxy}-N-[2-(dimethylamino)ethyl]benzamide
N-(1H-indol-2-ylmethyl)-2-(3-methyl-1,2-oxazol-5-yl)acetamide
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(prop-2-en-1-yl)acetamide
{[4-(1H-imidazol-1-yl)phenyl]methyl}(methyl)[1-(pyridin-2-yl)ethyl]amine
2-(2-methyl-1,3-thiazole-4-carbonyl)-6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinoline
2-[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]-4-methyl-1H-1,3-benzodiazole
N-[2-methoxy-2-(thiophen-2-yl)ethyl]-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
N-tert-butyl-5-chloro-2-{[1-(3-methylbut-2-en-1-yl)piperidin-4-yl]oxy}benzamide
N-methyl-N-(2-phenylethyl)-5-(thiomorpholin-4-ylmethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-(4-methoxy-3-pentanamidophenyl)-3-(propan-2-yl)-1H-pyrazole-4-carboxamide
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}(ethyl)[2-(pyrrolidin-1-yl)ethyl]amine
{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]amine
5-(1-propylpyrrolidin-2-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]thiophene-2-carboxamide
2-ethyl-6-methyl-N-[1-(piperidin-1-ylmethyl)cyclopropyl]pyrimidin-4-amine
(3R,4R)-1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-4-(morpholin-4-yl)piperidin-3-ol
4-[(2-{1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-1H-imidazol-1-yl)methyl]pyridine
7-(2,3-dimethylbenzoyl)-N2,N2,N4,N4-tetramethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine