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methyl[(4-methyl-1H-imidazol-5-yl)methyl]{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-ethyl-1-{[3-(prop-2-en-1-yl)-4-(prop-2-en-1-yloxy)phenyl]methyl}pyrrolidine-3-carboxamide
N-[1-(2-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-2-oxoethyl)-1H-pyrazol-4-yl]furan-2-carboxamide
2-{2-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]ethoxy}ethan-1-ol
methyl 6-[(4-acetylpiperazin-1-yl)methyl]-3-cyclohexaneamidothieno[2,3-b]pyridine-2-carboxylate
(3S,4S)-4-(naphthalen-2-yl)-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-ol
3-chloro-6-[4-(1-ethylpiperidin-4-yl)piperazin-1-yl]pyridine-2-carboxylic acid
1-(cyclohexylmethyl)-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-3,5-dimethylfuran-2-carboxamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-5-chloro-6-oxo-1,6-dihydropyridine-3-carboxamide
1-[4-(diphenylmethyl)piperazin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
4-{[3-(4-propylpiperazine-1-carbonyl)-1,2-oxazol-5-yl]methyl}morpholine
(2S,3S)-3-methyl-2-({1-[3-(trifluoromethyl)phenyl]propan-2-yl}amino)pentan-1-ol
ethyl[(1-methyl-1H-imidazol-2-yl)methyl][(3S)-3-phenylbutyl]amine
2-[5-(2,5-difluorophenyl)-1H-indazol-1-yl]-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
N-ethyl-4-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-1,3-thiazole-5-carboxamide
(3S,4S)-1-[2-(methylamino)pyridine-4-carbonyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
N-[(3S,4R)-1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
1-[5-(5-ethyl-1,3,4-oxadiazol-2-yl)-2-methoxyphenyl]-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]urea
1-[2-(dimethylamino)-4-(methylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
2-{[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]methyl}-4,5,6,7-tetrahydro-1,3-benzothiazole
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
5-(ethylsulfanyl)-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}thiophene-2-carboxamide
4-(1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)thiomorpholine
methyl 5-[(2,1,3-benzothiadiazol-5-ylmethyl)amino]-1-(2-methoxyethyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-1,9-dioxaspiro[5.5]undecan-4-amine
(1R,5R)-6-(cyclopropylmethyl)-3-(dimethyl-1,3-oxazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N,1-dimethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-ethyl-1-methyl-3-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(5-fluoro-2-methoxyphenyl)methyl]-3-methoxypiperidine
1-(4-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}phenyl)imidazolidine-2,4-dione
N-(2-methoxyethyl)-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-(1,3-thiazol-2-ylmethyl)propanamide
5-[1-(2,5-dimethylphenyl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-3,4-dihydropyrimidin-4-one
(4aR,7aS)-1-acetyl-4-[(3,4-difluorophenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{1-[(2,5-dimethylphenyl)methyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
N,6-dimethyl-N-[1-(3-phenylpropyl)piperidin-3-yl]pyridine-3-carboxamide
N'-(2,4-dimethylphenyl)-N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylpropanediamide
4-benzyl-3-ethyl-1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,4-diazepan-5-one
2-amino-N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
3-({4-[2-(2,6-difluoro-4-methoxyphenyl)-1H-imidazol-1-yl]piperidin-1-yl}methyl)pyridine
4-(1H-imidazol-1-ylmethyl)-1-[(3-phenyloxolan-3-yl)methyl]piperidin-4-ol
4-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
(1S,5R)-6-(2-methoxyethyl)-N-[(2-methylphenyl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-(4-fluorophenyl)-2-{2-[1-(propan-2-yl)piperidin-4-yl]acetamido}acetic acid
N-ethyl-5-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl]pyrimidin-2-amine
(5S,9aS,9bS)-5-(4-methoxy-3-methylphenyl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-[1-(2-hydroxyethyl)-5-(1-{3-oxo-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-2-yl}ethyl)-1H-1,2,4-triazol-3-yl]acetamide
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
2-cyclopropyl-N-[2-(3,4-dimethoxyphenyl)ethyl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide